A mechanistic model for colibactin-induced genotoxicity AR Healy, H Nikolayevskiy, JR Patel, JM Crawford, SB Herzon Journal of the American Chemical Society 138 (48), 15563-15570, 2016 | 84 | 2016 |
Conformational constraints of cyclopentane peptide nucleic acids facilitate tunable binding to DNA H Zheng, I Botos, V Clausse, H Nikolayevskiy, EE Rastede, MF Fouz, ... Nucleic Acids Research 49 (2), 713-725, 2021 | 24 | 2021 |
Structure elucidation of secondary metabolites: Current frontiers and lingering pitfalls M DiBello, AR Healy, H Nikolayevskiy, Z Xu, SB Herzon Accounts of chemical research 56 (12), 1656-1668, 2023 | 13 | 2023 |
Reaction Kinetics Direct a Rational Synthesis of an HIV‐1 Inactivator of Nucleocapsid Protein 7 and Provide Mechanistic Insight into Cellular Metabolism and Antiviral Activity H Nikolayevskiy, MT Scerba, JR Deschamps, DH Appella Chemistry–A European Journal 24 (38), 9485-9489, 2018 | 10 | 2018 |
Emergent properties of natural products SB Herzon Synlett 29 (14), 1823-1835, 2018 | 8 | 2018 |
The structure-activity profile of mercaptobenzamides’ anti-HIV activity suggests that thermodynamics of metabolism is more important than binding affinity to the target H Nikolayevskiy, M Robello, MT Scerba, EH Pasternak, M Saha, ... European journal of medicinal chemistry 178, 818-837, 2019 | 7 | 2019 |
Inhibition of HIV maturation via selective unfolding and cross-linking of Gag polyprotein by a mercaptobenzamide acetylator LM Miller Jenkins, EL Paine, L Deshmukh, H Nikolayevskiy, GC Lyons, ... Journal of the American Chemical Society 141 (20), 8327-8338, 2019 | 7 | 2019 |
A complex stereochemical relay approach to the antimalarial alkaloid ocimicide A 1. Evidence for a structural revision H Nikolayevskiy, MKM Tun, PR Rablen, CB Mamoun, SB Herzon Chemical Science 8 (7), 4867-4871, 2017 | 5 | 2017 |
Dna alkylation and cross-linking agents as compounds and payloads for targeted therapies S Herzon, A Healy, J Crawford, M Vizcaino, H Nikolayevskiy | 1 | 2017 |
Covalent Modification of p53 by (E)-1-(4-Methylpiperazin-1-yl)-3-(5-nitrofuran-2-yl)prop-2-en-1-one K Brown, M Robello, AJ Perciaccante, JC Dinan, TK Maity, GC Lyons, ... ACS Pharmacology & Translational Science 7 (11), 3559-3572, 2024 | | 2024 |
Mechanistic Analysis of 5-Hydroxy γ-Pyrones as Michael Acceptor Prodrugs C Leung, UM Bashir, WL Karney, MG Swanson, H Nikolayevskiy The Journal of Organic Chemistry 89 (17), 12432-12438, 2024 | | 2024 |
Mechanistic Analysis of 5-Hydroxy 𝛾-Pyrones as Michael Acceptor Prodrugs C Leung, U Bashir, W Karney, M Swanson, H Nikolayevskiy | | 2024 |
Prodrug Strategy Extends the Use of Anti-HIV Sulfanylbenzamides for Application In Vivo M Robello, H Nikolayevskiy, MT Scerba, RA Nahui Palomino, V Mercurio, ... ACS Pharmacology & Translational Science 7 (1), 259-273, 2023 | | 2023 |
N-(3-amino-3-oxopropyl)-2-[(1-methyl-4-nitro-1h-imidazol-5-yl) thio] benzamide and its use for treating hiv infection DH Appella, H Nikolayevskiy, M Robello, MT Scerba US Patent App. 17/785,155, 2023 | | 2023 |
Front Cover: Reaction Kinetics Direct a Rational Synthesis of an HIV‐1 Inactivator of Nucleocapsid Protein 7 and Provide Mechanistic Insight into Cellular Metabolism and … H Nikolayevskiy, MT Scerba, JR Deschamps, DH Appella Chemistry–A European Journal 24 (38), 9436-9436, 2018 | | 2018 |
Scalable synthesis and spectroscopic analysis of mercaptobenzamide thioester (SAMT) HIV inhibitors H Nikolayevskiy, M Scerba, D Appella ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 254, 2017 | | 2017 |