Следене
Alessia Bono
Alessia Bono
Dipartimento STEBICEF - University of Palermo
Потвърден имейл адрес: community.unipa.it
Заглавие
Позовавания
Позовавания
Година
Targeting SARS-CoV-2 main protease for treatment of COVID-19: Covalent inhibitors structure–activity relationship insights and evolution perspectives
G La Monica, A Bono, A Lauria, A Martorana
Journal of medicinal chemistry 65 (19), 12500-12534, 2022
1042022
Quinoline anticancer agents active on DNA and DNA-interacting proteins: From classical to emerging therapeutic targets
A Lauria, G La Monica, A Bono, A Martorana
European Journal of Medicinal Chemistry 220, 113555, 2021
692021
Antiproliferative activity predictor: a new reliable in silico tool for drug response prediction against NCI60 panel
A Martorana, G La Monica, A Bono, S Mannino, S Buscemi, ...
International Journal of Molecular Sciences 23 (22), 14374, 2022
92022
Off-target-based design of selective hiv-1 protease inhibitors
G La Monica, A Lauria, A Bono, A Martorana
International Journal of Molecular Sciences 22 (11), 6070, 2021
92021
mai n protease for treatment of COVID-19: covalent inhibitors structure–activit y relationship insights and evolution perspectives
G La Monica, A Bono, A Lauria, A Martorana
J. Med. Chem 65, 12500-12534, 2022
82022
In silico mixed ligand/structure-based design of new CDK-1/PARP-1 dual inhibitors as anti-breast cancer agents
A Bono, G La Monica, F Alamia, F Mingoia, C Gentile, D Peri, A Lauria, ...
International Journal of Molecular Sciences 24 (18), 13769, 2023
62023
In Silico Design of New Dual Inhibitors of SARS-CoV-2 MPRO through Ligand- and Structure-Based Methods
A Bono, A Lauria, G La Monica, F Alamia, F Mingoia, A Martorana
International Journal of Molecular Sciences 24 (9), 8377, 2023
62023
Synthesis of new antiproliferative 1, 3, 4-substituted-pyrrolo [3, 2-c] quinoline derivatives, biological and in silico insights
F Mingoia, C Di Sano, C D'Anna, M Fazzari, L Minafra, A Bono, ...
European Journal of Medicinal Chemistry 258, 115537, 2023
52023
Bioisosteric heterocyclic analogues of natural bioactive flavonoids by scaffold-hopping approaches: State-of-the-art and perspectives in medicinal chemistry
G La Monica, A Bono, F Alamia, A Lauria, A Martorana
Bioorganic & Medicinal Chemistry, 117791, 2024
42024
Design and Synthesis of Novel Thieno[3,2-c]quinoline Compounds with Antiproliferative Activity on RET-Dependent Medullary Thyroid Cancer Cells
G La Monica, G Pizzolanti, C Baiamonte, A Bono, F Alamia, F Mingoia, ...
ACS omega 8 (38), 34640-34649, 2023
32023
Scaffold-hopping strategies in aurone optimization: A comprehensive review of synthetic procedures and biological activities of nitrogen and sulfur analogues
G La Monica, F Alamia, A Bono, A Lauria, A Martorana
Molecules 29 (12), 2813, 2024
22024
One pot-like regiospecific access to 1-aryl-1H-pyrazol-3 (2H)-one derivatives and evaluation of the anticancer activity
F Mingoia, G Panzeca, MC Vitale, G La Monica, A Bono, A Lauria, ...
Arkivoc 2022, 191-203, 2022
22022
Antiproliferative properties and g-quadruplex-binding of symmetrical naphtho [1, 2-b: 8, 7-b’] dithiophene derivatives
A Lauria, G La Monica, A Terenzi, G Mannino, R Bonsignore, A Bono, ...
Molecules 26 (14), 4309, 2021
22021
A novel in silico approach for identifying multi-target JAK/STAT inhibitors as anticancer agents
A Bono, G La Monica, F Alamia, A Lauria, A Martorana
Journal of Molecular Graphics and Modelling 135, 108913, 2025
2025
Design, Synthesis, and In Silico Insights of new 4‐Piperazinylquinolines as Antiproliferative Agents against NCI Renal Cancer Cell Lines
G La Monica, A Bono, F Alamia, A Martorana, A Lauria
ChemistryOpen, e202400518, 2025
2025
Novel Antibacterial 4-Piperazinylquinoline Hybrid Derivatives Against Staphylococcus aureus: Design, Synthesis, and In Vitro and In Silico Insights
G La Monica, A Gallo, A Bono, F Alamia, A Lauria, R Alduina, A Martorana
Molecules 30 (1), 28, 2024
2024
In Silico Design of Dual Estrogen Receptor and Hsp90 Inhibitors for ER-Positive Breast Cancer Through a Mixed Ligand/Structure-Based Approach
G La Monica, F Alamia, A Bono, F Mingoia, A Martorana, A Lauria
Molecules 29 (24), 6040, 2024
2024
Targeting the SARS-CoV-2 MPRO through covalent and non-covalent inhibition: molecular modeling and synthetic procedures for the development of new antiviral molecules
A Bono
Università degli Studi di Palermo, 2024
2024
Innovative In Silico Method for Discovering Multi-Target JAK/STAT Inhibitors as Potential Anticancer Therapies
A Bono, G LA MONICA, F Alamia, A Lauria, A Martorana
Atti del Congresso Congiunto 2024 delle Sezioni Sicilia e Calabria della …, 2024
2024
Machine learning model for predicting molecular activity using Molecular Descriptors and ElectroShape Descriptors-FL051
A Bono, A Asad, M Albanese, RI Cooper, A Lauria, G LA MONICA, ...
Proceedings of the Merck Young Chemists’ Symposium XXIII edition, 2024
2024
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