Harnessing the therapeutic potential of capsaicin and its analogues in pain and other diseases S Basith, M Cui, S Hong, S Choi Molecules 21 (8), 966, 2016 | 213 | 2016 |
Exploring G protein-coupled receptors (GPCRs) ligand space via cheminformatics approaches: impact on rational drug design S Basith, M Cui, SJY Macalino, J Park, NAB Clavio, S Kang, S Choi Frontiers in pharmacology 9, 128, 2018 | 203 | 2018 |
Transient receptor potential vanilloid type 1 antagonists: a patent review (2011–2014) Y Lee, S Hong, M Cui, PK Sharma, J Lee, S Choi Expert opinion on therapeutic patents 25 (3), 291-318, 2015 | 85 | 2015 |
Transmembrane 4 L six family member 5 senses arginine for mTORC1 signaling JW Jung, SJY Macalino, M Cui, JE Kim, HJ Kim, DG Song, SH Nam, ... Cell Metabolism 29 (6), 1306-1319. e7, 2019 | 65 | 2019 |
Polymodal transient receptor potential vanilloid type 1 nocisensor: structure, modulators, and therapeutic applications M Cui, V Gosu, S Basith, S Hong, S Choi Advances in Protein Chemistry and Structural Biology 104, 81-125, 2016 | 56 | 2016 |
Discovery of potent human glutaminyl cyclase inhibitors as anti-Alzheimer’s agents based on rational design VH Hoang, PT Tran, M Cui, VTH Ngo, J Ann, J Park, J Lee, K Choi, H Cho, ... Journal of medicinal chemistry 60 (6), 2573-2590, 2017 | 50 | 2017 |
Expediting the design, discovery and development of anticancer drugs using computational approaches S Basith, M Cui, SJY Macalino, S Choi Current medicinal chemistry 24 (42), 4753-4778, 2017 | 43 | 2017 |
The cell shape-determining Csd6 protein from Helicobacter pylori constitutes a new family of L, D-carboxypeptidase HS Kim, HN Im, DR An, JY Yoon, JY Jang, S Mobashery, D Hesek, M Lee, ... Journal of Biological Chemistry 290 (41), 25103-25117, 2015 | 41 | 2015 |
TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl) propanamides TH Ha, HC Ryu, SE Kim, HS Kim, J Ann, PT Tran, VH Hoang, K Son, ... Bioorganic & medicinal chemistry 21 (21), 6657-6664, 2013 | 28 | 2013 |
In silico prediction of multiple-category classification model for cytochrome P450 inhibitors and non-inhibitors using machine-learning method JH Lee, S Basith, M Cui, B Kim, S Choi SAR and QSAR in Environmental Research 28 (10), 863-874, 2017 | 27 | 2017 |
Synthesis and Anti-Renal Fibrosis Activity of Conformationally Locked Truncated 2-Hexynyl-N6-Substituted-(N)-Methanocarba-nucleosides as A3 Adenosine … A Nayak, G Chandra, I Hwang, K Kim, X Hou, HO Kim, PK Sahu, KK Roy, ... Journal of Medicinal Chemistry 57 (4), 1344-1354, 2014 | 27 | 2014 |
N6-Substituted 5′-N-Methylcarbamoyl-4′-selenoadenosines as Potent and Selective A3 Adenosine Receptor Agonists with Unusual Sugar Puckering and … J Yu, LX Zhao, J Park, HW Lee, PK Sahu, M Cui, SM Moss, E Hammes, ... Journal of medicinal chemistry 60 (8), 3422-3437, 2017 | 26 | 2017 |
Discovery of conformationally restricted human glutaminyl cyclase inhibitors as potent anti-Alzheimer’s agents by structure-based design VH Hoang, VTH Ngo, M Cui, NV Manh, PT Tran, J Ann, HJ Ha, H Kim, ... Journal of medicinal chemistry 62 (17), 8011-8027, 2019 | 24 | 2019 |
Synthesis and biological evaluation of 3-substituted 5-benzylidene-1-methyl-2-thiohydantoins as potent NADPH oxidase (NOX) inhibitors YS Bae, S Choi, JJ Park, JH Joo, M Cui, H Cho, WJ Lee, SH Lee Bioorganic & Medicinal Chemistry 24 (18), 4144-4151, 2016 | 24 | 2016 |
5-Lipoxygenase inhibitors suppress RANKL-induced osteoclast formation via NFATc1 expression JH Kang, Z Ting, M Moon, JS Sim, JM Lee, KE Doh, S Hong, M Cui, ... Bioorganic & medicinal chemistry 23 (21), 7069-7078, 2015 | 24 | 2015 |
Structure-activity relationship investigation of Phe-Arg mimetic region of human glutaminyl cyclase inhibitors VTH Ngo, VH Hoang, PT Tran, N Van Manh, J Ann, E Kim, M Cui, S Choi, ... Bioorganic & Medicinal Chemistry 26 (12), 3133-3144, 2018 | 23 | 2018 |
Potent human glutaminyl cyclase inhibitors as potential anti-Alzheimer’s agents: Structure-activity relationship study of Arg-mimetic region VTH Ngo, VH Hoang, PT Tran, J Ann, M Cui, G Park, S Choi, J Lee, H Kim, ... Bioorganic & medicinal chemistry 26 (5), 1035-1049, 2018 | 23 | 2018 |
2-Alkyl/alkenyl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl) propanamides as highly potent TRPV1 antagonists HC Ryu, S Seo, SH Cho, HS Kim, A Jung, DW Kang, K Son, M Cui, ... Bioorganic & medicinal chemistry letters 24 (16), 4039-4043, 2014 | 20 | 2014 |
Anti‐angiogenic activity of thienopyridine derivative LCB 03‐0110 by targeting VEGFR‐2 and JAK/STAT 3 Signalling BH Kim, Y Lee, H Yoo, M Cui, S Lee, SY Kim, JU Cho, H Lee, BS Yang, ... Experimental dermatology 24 (7), 503-509, 2015 | 19 | 2015 |
2-Aryl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl) propanamides as highly potent TRPV1 antagonists HC Ryu, S Seo, MS Kim, MY Kim, HS Kim, J Ann, PT Tran, VH Hoang, ... Bioorganic & medicinal chemistry letters 24 (16), 4044-4047, 2014 | 19 | 2014 |