| A strategy for the diversity-oriented synthesis of macrocyclic scaffolds using multidimensional coupling HSG Beckmann, F Nie, CE Hagerman, H Johansson, YS Tan, D Wilcke, ... Nature Chemistry 5 (10), 861-867, 2013 | 132 | 2013 |
| Fragment-based covalent ligand screening enables rapid discovery of inhibitors for the RBR E3 ubiquitin ligase HOIP H Johansson, YC Isabella Tsai, K Fantom, CW Chung, S Kümper, ... Journal of the American Chemical Society 141 (6), 2703-2712, 2019 | 124 | 2019 |
| Greening the synthesis of peptide therapeutics: an industrial perspective V Martin, PHG Egelund, H Johansson, ST Le Quement, F Wojcik, ... RSC advances 10 (69), 42457-42492, 2020 | 104 | 2020 |
| 3-Substituted 2-phenyl-indoles: privileged structures for medicinal chemistry H Johansson, TB Jørgensen, DE Gloriam, H Bräuner-Osborne, ... RSC Advances 3 (3), 945-960, 2013 | 75 | 2013 |
| Harnessing polarity and viscosity to identify green binary solvent mixtures as viable alternatives to DMF in solid-phase peptide synthesis V Martin, S Jadhav, PHG Egelund, R Liffert, HJ Castro, T Krüger, ... Green Chemistry 23 (9), 3295-3311, 2021 | 52 | 2021 |
| Azide‐and alkyne‐derivatised α‐amino acids H Johansson, DS Pedersen European Journal of Organic Chemistry 2012 (23), 4267-4281, 2012 | 48 | 2012 |
| Replacing DMF in solid-phase peptide synthesis: varying the composition of green binary solvent mixtures as a tool to mitigate common side-reactions S Jadhav, V Martin, PHG Egelund, HJ Castro, T Krüger, F Richner, ... Green Chemistry 23 (9), 3312-3321, 2021 | 44 | 2021 |
| Fmoc-removal with pyrrolidine expands the available solvent space in green solid-phase peptide synthesis PHG Egelund, S Jadhav, V Martin, H Johansson Castro, F Richner, ... ACS Sustainable Chemistry & Engineering 9 (42), 14202-14215, 2021 | 30 | 2021 |
| Selective allosteric antagonists for the G protein-coupled receptor GPRC6A based on the 2-phenylindole privileged structure scaffold H Johansson, MW Boesgaard, L Nørskov-Lauritsen, I Larsen, S Kuhne, ... Journal of medicinal chemistry 58 (22), 8938-8951, 2015 | 27 | 2015 |
| Probing the Existence of a Metastable Binding Site at the β2-Adrenergic Receptor with Homobivalent Bitopic Ligands BI Gaiser, M Danielsen, E Marcher-Rørsted, K Røpke Jørgensen, ... Journal of medicinal chemistry 62 (17), 7806-7839, 2019 | 25 | 2019 |
| A scalable method for regioselective 3-acylation of 2-substituted indoles under basic conditions H Johansson, A Urruticoechea, I Larsen, D Sejer Pedersen The Journal of Organic Chemistry 80 (1), 471-481, 2015 | 23 | 2015 |
| Single-domain antibodies as crystallization chaperones to enable structure-based inhibitor development for RBR E3 ubiquitin ligases YCI Tsai, H Johansson, D Dixon, S Martin, C Chung, J Clarkson, D House, ... Cell chemical biology 27 (1), 83-93. e9, 2020 | 18 | 2020 |
| Synthesis of the calcilytic ligand NPS 2143 H Johansson, T Cailly, ARB Thomsen, H Bräuner-Osborne, DS Pedersen Beilstein Journal of Organic Chemistry 9 (1), 1383-1387, 2013 | 14 | 2013 |
| Exploring endoperoxides as a new entry for the synthesis of branched azasugars S Domeyer, M Bjerregaard, H Johansson, DS Pedersen Beilstein Journal of Organic Chemistry 13 (1), 644-647, 2017 | 7 | 2017 |
| Revisiting Bromohexitols as a Novel Class of Microenvironment‐Activated Prodrugs for Cancer Therapy H Johansson, O Hussain, SJ Allison, TV Robinson, RM Phillips, ... ChemMedChem 15 (2), 228-235, 2020 | | 2020 |
| ALLOSTERIC ANTAGONISTS OF GPRC6a AND THEIR USE IN MITIGATING PROTEINOPATHIES DC Lee, DS Pedersen, H Bräuner-Osborne, DE Gloriam, S Kuhne, ... US Patent App. 16/461,716, 2019 | | 2019 |
| Design and Synthesis of Allosteric Modulators for the G Protein-coupled Receptor GPRC6A: PhD Thesis H Johansson Faculty of Health and Medical Sciences, University of Copenhagen, 2014 | | 2014 |
| Taming the G protein-coupled receptor GPRC6A H Johansson, H Brauner-Osborne, DS Pedersen ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 245, 2013 | | 2013 |