| Crystallographic and electrophilic fragment screening of the SARS-CoV-2 main protease A Douangamath, D Fearon, P Gehrtz, T Krojer, P Lukacik, CD Owen, ... Nature communications 11 (1), 5047, 2020 | 506 | 2020 |
| A road map for prioritizing warheads for cysteine targeting covalent inhibitors P Abranyi-Balogh, L Petri, T Imre, P Szijj, A Scarpino, M Hrast, A Mitrović, ... European journal of medicinal chemistry 160, 94-107, 2018 | 130 | 2018 |
| Covalent fragment libraries in drug discovery A Keeley, L Petri, P Ábrányi-Balogh, GM Keserű Drug Discovery Today 25 (6), 983-996, 2020 | 98 | 2020 |
| Design and characterization of a heterocyclic electrophilic fragment library for the discovery of cysteine-targeted covalent inhibitors A Keeley, P Ábrányi-Balogh, GM Keserű MedChemComm 10 (2), 263-267, 2019 | 76 | 2019 |
| The synthesis of α-aryl-α-aminophosphonates and α-aryl-α-aminophosphine oxides by the microwave-assisted Pudovik reaction E Bálint, Á Tajti, A Ádám, I Csontos, K Karaghiosoff, M Czugler, ... Beilstein Journal of Organic Chemistry 13 (1), 76-86, 2017 | 57 | 2017 |
| Electrophilic warheads in covalent drug discovery: an overview N Péczka, Z Orgován, P Ábrányi-Balogh, GM Keserű Expert Opinion on Drug Discovery 17 (4), 413-422, 2022 | 55 | 2022 |
| T3P®-promoted Kabachnik–Fields reaction: An efficient synthesis of α-aminophosphonates M Milen, P Abranyi-Balogh, A Dancsó, D Frigyes, L Pongo, G Keglevich Tetrahedron Letters 54 (40), 5430-5433, 2013 | 48 | 2013 |
| Comparative reactivity analysis of small-molecule thiol surrogates L Petri, P Ábrányi-Balogh, PR Varga, T Imre, GM Keserű Bioorganic & Medicinal Chemistry 28 (7), 115357, 2020 | 39 | 2020 |
| An electrophilic warhead library for mapping the reactivity and accessibility of tractable cysteines in protein kinases L Petri, A Egyed, D Bajusz, T Imre, A Hetényi, T Martinek, ... European Journal of Medicinal Chemistry 207, 112836, 2020 | 37 | 2020 |
| A Mechanistic Study on the Tautomerism of H-Phosphonates, H-Phosphinates and Secondary Phosphine Oxides D Vincze, P Ábrányi-Balogh, P Bagi, G Keglevich Molecules 24 (21), 3859, 2019 | 35 | 2019 |
| PharmacoSTORM nanoscale pharmacology reveals cariprazine binding on Islands of Calleja granule cells S Prokop, P Ábrányi-Balogh, B Barti, M Vámosi, M Zöldi, L Barna, ... Nature communications 12 (1), 6505, 2021 | 34 | 2021 |
| Cysteine specific bioconjugation with benzyl isothiocyanates L Petri, PA Szijj, Á Kelemen, T Imre, Á Gömöry, MTW Lee, K Hegedűs, ... RSC advances 10 (25), 14928-14936, 2020 | 34 | 2020 |
| Synthesis of β-carbolines (microreview) M Milen, P Ábrányi-Balogh Chemistry of Heterocyclic Compounds 52, 996-998, 2016 | 34 | 2016 |
| Penicillin's catalytic mechanism revealed by inelastic neutrons and quantum chemical theory Z Mucsi, GA Chass, P Ábrányi-Balogh, B Jójárt, DC Fang, ... Physical chemistry chemical physics 15 (47), 20447-20455, 2013 | 31 | 2013 |
| A novel three-component reaction between isocyanides, alcohols or thiols and elemental sulfur: a mild, catalyst-free approach towards O-thiocarbamates and dithiocarbamates AG Németh, GM Keserű, P Ábrányi-Balogh Beilstein Journal of Organic Chemistry 15 (1), 1523-1533, 2019 | 29 | 2019 |
| Heterocyclic electrophiles as new MurA inhibitors A Keeley, P Ábrányi‐Balogh, M Hrast, T Imre, J Ilaš, S Gobec, GM Keserű Archiv der Pharmazie 351 (12), 1800184, 2018 | 29 | 2018 |
| Synthetic study on the T3P®-promoted one-pot preparation of 1-substituted-3, 4-dihydro-β-carbolines by the reaction of tryptamine with carboxylic acids P Abranyi-Balogh, T Földesi, A Grün, B Volk, G Keglevich, M Milen Tetrahedron Letters 57 (18), 1953-1957, 2016 | 29 | 2016 |
| Vinylation of α-Aminoazoles with Triethylamine: A General Strategy to Construct Azolo[1,5-a]pyrimidines with a Nonsubstituted Ethylidene Fragment Q Gao, Z Sun, Q Xia, R Li, W Wang, S Ma, Y Chai, M Wu, W Hu, ... Organic Letters 23 (7), 2664-2669, 2021 | 28 | 2021 |
| WIDOCK: a reactive docking protocol for virtual screening of covalent inhibitors A Scarpino, L Petri, D Knez, T Imre, P Ábrányi-Balogh, GG Ferenczy, ... Journal of Computer-Aided Molecular Design 35, 223-244, 2021 | 26 | 2021 |
| T3P®‐Mediated One‐Pot Synthesis of Bis (α‐aminophosphonates) M Milen, P Ábrányi‐Balogh, R Kangyal, A Dancso, D Frigyes, G Keglevich Heteroatom Chemistry 25 (4), 245-255, 2014 | 26 | 2014 |
