Sledovat
Attila Keresztes
Název
Citace
Citace
Rok
Cannabis sativa terpenes are cannabimimetic and selectively enhance cannabinoid activity
JE LaVigne, R Hecksel, A Keresztes, JM Streicher
Scientific reports 11 (1), 8232, 2021
1102021
Analgesic potential of terpenes derived from Cannabis sativa
E Liktor-Busa, A Keresztes, J LaVigne, JM Streicher, TM Largent-Milnes
Pharmacological reviews 73 (4), 1269-1297, 2021
772021
Repeated morphine treatment-mediated hyperalgesia, allodynia and spinal glial activation are blocked by co-administration of a selective cannabinoid receptor type-2 agonist
S Tumati, TM Largent-Milnes, A Keresztes, J Ren, WR Roeske, ...
Journal of neuroimmunology 244 (1-2), 23-31, 2012
562012
New endomorphin analogues containing alicyclic β-amino acids: Influence on bioactive conformation and pharmacological profile
A Keresztes, M Szucs, A Borics, KE Kövér, E Forro, F Fülöp, ...
Journal of Medicinal Chemistry 51 (14), 4270-4279, 2008
552008
Design of novel neurokinin 1 receptor antagonists based on conformationally constrained aromatic amino acids and discovery of a potent chimeric opioid agonist-neurokinin 1 …
S Ballet, D Feytens, K Buysse, NN Chung, C Lemieux, S Tumati, ...
Journal of medicinal chemistry 54 (7), 2467-2476, 2011
542011
Synthesis and evaluation of a novel bivalent selective antagonist for the mu-delta opioid receptor heterodimer that reduces morphine withdrawal in mice
KM Olson, A Keresztes, JK Tashiro, LV Daconta, VJ Hruby, JM Streicher
Journal of medicinal chemistry 61 (14), 6075-6086, 2018
492018
Recent advances in endomorphin engineering
A Keresztes, A Borics, G Tóth
ChemMedChem 5 (8), 1176-1196, 2010
492010
Novel molecular strategies and targets for opioid drug discovery for the treatment of chronic pain
KM Olson, W Lei, A Keresztes, J LaVigne, JM Streicher
The Yale journal of biology and medicine 90 (1), 97, 2017
472017
Tachykinin NK1 receptor antagonist co-administration attenuates opioid withdrawal-mediated spinal microglia and astrocyte activation
S Tumati, TM Largent-Milnes, AI Keresztes, T Yamamoto, TW Vanderah, ...
European journal of pharmacology 684 (1-3), 64-70, 2012
422012
Design, synthesis, pharmacological evaluation, and structure− activity study of novel endomorphin analogues with multiple structural modifications
JR Mallareddy, A Borics, A Keresztes, KE Kövér, D Tourwé, G Tóth
Journal of medicinal chemistry 54 (5), 1462-1472, 2011
412011
Analgesic properties of opioid/NK1 multitarget ligands with distinct in vitro profiles in naive and chronic constriction injury mice
J Starnowska, R Costante, K Guillemyn, K Popiolek-Barczyk, NN Chung, ...
ACS chemical neuroscience 8 (10), 2315-2324, 2017
382017
Preparation of bivalent agonists for targeting the mu opioid and cannabinoid receptors
S Dvorácskó, A Keresztes, A Mollica, A Stefanucci, G Macedonio, ...
European journal of medicinal chemistry 178, 571-588, 2019
362019
Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist–neurokinin-1 antagonist peptidomimetics
K Guillemyn, P Kleczkowska, A Lesniak, J Dyniewicz, O Van der Poorten, ...
European journal of medicinal chemistry 92, 64-77, 2015
352015
Structural basis of small molecule targetability of monomeric tau protein
R Kiss, G Csizmadia, K Solti, A Keresztes, M Zhu, M Pickhardt, ...
ACS Chemical Neuroscience 9 (12), 2997-3006, 2018
312018
Synthesis and pharmacology of a novel μ–δ opioid receptor heteromer-selective agonist based on the carfentanyl template
A Faouzi, R Uprety, I Gomes, N Massaly, AI Keresztes, V Le Rouzic, ...
Journal of medicinal chemistry 63 (22), 13618-13637, 2020
302020
New endomorphin analogs with mu-agonist and delta-antagonist properties
G Tóth, A Keresztes, C Tömböly, A Péter, F Fülöp, D Tourwe, ...
Pure and applied chemistry 76 (5), 951-957, 2004
292004
Influence of ring substitution on the conformation and β-turn mimicry of 4-amino-1, 2, 4, 5-tetrahydro-2-benzazepin-3-one peptide mimetics
R De Wachter, L Brans, S Ballet, I Van den Eynde, D Feytens, A Keresztes, ...
Tetrahedron 65 (11), 2266-2278, 2009
252009
Antagonism of the mu-delta opioid receptor heterodimer enhances opioid antinociception by activating Src and calcium/calmodulin-dependent protein kinase II signaling
A Keresztes, K Olson, P Nguyen, MA Lopez-Pier, R Hecksel, NK Barker, ...
Pain 163 (1), 146-158, 2022
232022
Dual alleviation of acute and neuropathic pain by fused opioid agonist-neurokinin 1 antagonist peptidomimetics
C Betti, J Starnowska, J Mika, J Dyniewicz, L Frankiewicz, A Novoa, ...
ACS Medicinal Chemistry Letters 6 (12), 1209-1214, 2015
232015
Investigation of receptor binding and functional characteristics of hemopressin (1–7)
S Dvorácskó, C Tömböly, R Berkecz, A Keresztes
Neuropeptides 58, 15-22, 2016
212016
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Články 1–20