| Discovery and structure–activity relationships of a highly selective butyrylcholinesterase inhibitor by structure-based virtual screening SN Dighe, GS Deora, E De la Mora, F Nachon, S Chan, MO Parat, ... Journal of medicinal chemistry 59 (16), 7683-7689, 2016 | 159 | 2016 |
| Novel N-indolylmethyl substituted olanzapine derivatives: Their design, synthesis and evaluation as PDE4B inhibitors DR Gorja, S Mukherjee, CLT Meda, GS Deora, K Lalith Kumar, A Jain, ... Org. Biomol. Chem. 11, 2075-2079, 2013 | 72 | 2013 |
| Synthesis and pharmacological evaluation of pyrazolo [4, 3-< i> c</i>] cinnoline derivatives as potential anti-inflammatory and antibacterial agents RK Tonk, S Bawa, G Chawla, GS Deora, S Kumar, V Rathore, ... European Journal of Medicinal Chemistry 57, 176-184, 2012 | 71 | 2012 |
| Synthesis and evaluation of 3-amino/guanidine substituted phenyl oxazoles as a novel class of LSD1 inhibitors with anti-proliferative properties B Dulla, KT Kirla, V Rathore, GS Deora, S Kavela, S Maddika, K Chatti, ... Organic & biomolecular chemistry 11, 3103, 2013 | 66 | 2013 |
| Spiro heterocycles as potential inhibitors of SIRT1: Pd/C-mediated synthesis of novel N-indolylmethyl spiroindoline-3, 2′-quinazolines D Rambabu, G Raja, BY Sreenivas, GPK Seerapu, KL Kumar, GS Deora, ... Bioorganic & medicinal chemistry letters 23 (5), 1351-1357, 2013 | 54 | 2013 |
| Synthesis of some coumarinyl chalcones and their antiproliferative activity against breast cancer cell lines K Patel, C Karthikeyan, V Raja Solomon, N S. Hari Narayana Moorthy, ... Letters in Drug Design & Discovery 8 (4), 308-311, 2011 | 54 | 2011 |
| Cu-mediated 1, 3-dipolar cycloaddition of azomethine ylides with dipolarophiles: a faster access to spirooxindoles of potential pharmacological interest SN Singh, S Regati, AK Paul, M Layek, S Jayaprakash, KV Reddy, ... Tetrahedron Letters 54 (40), 5448-5452, 2013 | 53 | 2013 |
| Design, synthesis and biological evaluation of some novel 3-cinnamoyl-4-hydroxy-2H-chromen-2-ones as antimalarial agents K Patel, C Karthikeyan, NS Hari Narayana Moorthy, GS Deora, ... Medicinal Chemistry Research 21, 1780-1784, 2012 | 50 | 2012 |
| A brain-permeable inhibitor of the neurodegenerative disease target kynurenine 3-monooxygenase prevents accumulation of neurotoxic metabolites S Zhang, M Sakuma, GS Deora, CW Levy, A Klausing, C Breda, KD Read, ... Communications biology 2 (1), 271, 2019 | 49 | 2019 |
| AlCl (3) mediated unexpected migration of sulfonyl groups: regioselective synthesis of 7-sulfonyl indoles of potential pharmacological interest. B Prasad, R Adepu, S Sandra, D Rambabu, GR Krishna, CM Reddy, ... Chemical communications (Cambridge, England) 48, 10434-10436, 2012 | 48 | 2012 |
| Synthesis, anti-inflammatory, analgesic, COX1/2-inhibitory activity, and molecular docking studies of hybrid pyrazole analogues MJ Alam, O Alam, SA Khan, MJ Naim, M Islamuddin, GS Deora Drug design, development and therapy, 3529-3543, 2016 | 43 | 2016 |
| Effect of the Biphenyl Neolignan Honokiol on Aβ42-Induced Toxicity in Caenorhabditis elegans, Aβ42 Fibrillation, Cholinesterase Activity, DPPH Radicals, and … S Kantham, S Chan, G McColl, JA Miles, SK Veliyath, GS Deora, ... ACS Chemical Neuroscience 8 (9), 1901-1912, 2017 | 42 | 2017 |
| Facile assembly of two 6-membered fused N-heterocyclic rings: a rapid access to novel small molecules via Cu-mediated reaction MP R Adepu, R Sunke, CLT Meda, GS Deora, D Rambabu Chemical Communications 49 (2), 190-192, 2013 | 42 | 2013 |
| Synthesis of novel benzimidazole acrylonitriles for inhibition of Plasmodium falciparum growth by dual target inhibition K Sharma, A Shrivastava, RN Mehra, GS Deora, MM Alam, MS Zaman, ... Archiv der Pharmazie 351 (1), 1700251, 2018 | 41 | 2018 |
| Multifunctional analogs of kynurenic acid for the treatment of Alzheimer’s disease: synthesis, pharmacology, and molecular modeling studies GS Deora, S Kantham, S Chan, SN Dighe, SK Veliyath, G McColl, ... ACS chemical neuroscience 8 (12), 2667-2675, 2017 | 37 | 2017 |
| Synthesis of 2, 2, 4-trimethyl-1, 2-dihydroquinolinyl substituted 1, 2, 3-triazole derivatives: Their evaluation as potential PDE 4B inhibitors possessing cytotoxic properties … KSS Praveena, S Durgadas, NS Babu, S Akkenapally, CG Kumar, ... Bioorganic Chemistry 53, 8-14, 2014 | 37 | 2014 |
| Pyrrole [2, 3< i>-b</i>] quinoxalines as inhibitors of firefly luciferase: Their Cu-mediated synthesis and evaluation as false positives in a reporter Gene Assay A Nakhi, S Rahman, R Kishore, CLT Meda, GS Deora, KVL Parsa, M Pal Bioorganic & Medicinal Chemistry Letters 22, 6433-6441, 2012 | 35 | 2012 |
| Design, synthesis and molecular modelling studies of novel 3-acetamido-4-methyl benzoic acid derivatives as inhibitors of protein tyrosine phosphatase 1B M Rakse, C Karthikeyan, GS Deora, N Moorthy, V Rathore, AK Rawat, ... European Journal of Medicinal Chemistry 70, 469-476, 2013 | 31 | 2013 |
| Ligand/PTC-free intramolecular Heck reaction: synthesis of pyrroloquinoxalines and their evaluation against PDE4/luciferase/oral cancer cell growth in vitro and zebrafish in vivo P Vijaya Babu, S Mukherjee, GS Deora, K Chennubhotla, R Medisetti, ... Organic & biomolecular chemistry 11 (39), 6680-6685, 2013 | 29 | 2013 |
| AgNO< sub> 3</sub> mediated CN bond forming reaction: Synthesis of 3-substituted benzothiazines as potential COX inhibitors D Rambabu, P Murthy, KRS Prasad, A Kandale, GS Deora, ... Tetrahedron Letters 53, 6577-6583, 2012 | 28 | 2012 |
Prof. Manojit Pal, FRSCProfessor of Organic and Medicinal ChemistryBestätigte E-Mail-Adresse bei drils.org