| The inhibition of cysteine proteases rhodesain and TbCatB: A valuable approach to treat Human African Trypanosomiasis R Ettari, S Previti, L Tamborini, G Cullia, S Grasso, M Zappalà Mini reviews in medicinal chemistry 16 (17), 1374-1391, 2016 | 62 | 2016 |
| Inspired by Nature: The 3‐Halo‐4, 5‐dihydroisoxazole Moiety as a Novel Molecular Warhead for the Design of Covalent Inhibitors A Pinto, L Tamborini, G Cullia, P Conti, C De Micheli ChemMedChem 11 (1), 10-14, 2016 | 30 | 2016 |
| Simple rules govern the diversity of bacterial nicotianamine-like metallophores C Laffont, C Brutesco, C Hajjar, G Cullia, R Fanelli, L Ouerdane, ... Biochemical Journal 476 (15), 2221-2233, 2019 | 22 | 2019 |
| Selectivity of 3-bromo-isoxazoline inhibitors between human and Plasmodium falciparum glyceraldehyde-3-phosphate dehydrogenases S Bruno, M Margiotta, A Pinto, G Cullia, P Conti, C De Micheli, ... Bioorganic & Medicinal Chemistry 24 (12), 2654-2659, 2016 | 22 | 2016 |
| Control by metals of staphylopine dehydrogenase activity during metallophore biosynthesis C Hajjar, R Fanelli, C Laffont, C Brutesco, G Cullia, M Tribout, D Nurizzo, ... Journal of the American Chemical Society 141 (13), 5555-5562, 2019 | 20 | 2019 |
| Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity TC Eadsforth, A Pinto, R Luciani, L Tamborini, G Cullia, C De Micheli, ... Journal of medicinal chemistry 58 (20), 7938-7948, 2015 | 18 | 2015 |
| Covalent Inhibitors of Plasmodium falciparum Glyceraldehyde 3-Phosphate Dehydrogenase with Antimalarial Activity in Vitro G Cullia, S Bruno, S Parapini, M Margiotta, L Tamborini, A Pinto, ... ACS Medicinal Chemistry Letters 10 (4), 590-595, 2019 | 17 | 2019 |
| 3-Bromo-isoxazoline derivatives inhibit GAPDH enzyme in PDAC cells triggering autophagy and apoptotic cell death R Pacchiana, N Mullappilly, A Pinto, S Bova, S Forciniti, G Cullia, ... Cancers 14 (13), 3153, 2022 | 16 | 2022 |
| Bicyclic γ-amino acids as inhibitors of γ-aminobutyrate aminotransferase A Pinto, L Tamborini, E Pennacchietti, A Coluccia, R Silvestri, G Cullia, ... Journal of Enzyme Inhibition and Medicinal Chemistry 31 (2), 295-301, 2016 | 15 | 2016 |
| 3-Carboxy-pyrazolinalanine as a new scaffold for developing potent and selective NMDA receptor antagonists L Tamborini, A Pinto, F Mastronardi, MC Iannuzzi, G Cullia, B Nielsen, ... European Journal of Medicinal Chemistry 68, 33-37, 2013 | 13 | 2013 |
| Folates in Trypanosoma brucei: Achievements and Opportunities G Cullia, L Tamborini, P Conti, C De Micheli, A Pinto ChemMedChem 13 (20), 2150-2158, 2018 | 12 | 2018 |
| Targeting NOX2 via p47/Phox-p22/Phox inhibition with novel triproline mimetics JB Garsi, B Komjáti, G Cullia, I Fejes, M Sipos, Z Sipos, E Fördős, ... ACS Medicinal Chemistry Letters 13 (6), 949-954, 2022 | 9 | 2022 |
| Identification of a 2, 4-diaminopyrimidine scaffold targeting Trypanosoma brucei pteridine reductase 1 from the LIBRA compound library screening campaign P Linciano, G Cullia, C Borsari, M Santucci, S Ferrari, G Witt, S Gul, ... European Journal of Medicinal Chemistry 189, 112047, 2020 | 9 | 2020 |
| Synthesis and pharmacological evaluation of conformationally constrained glutamic acid higher homologues L Tamborini, G Cullia, B Nielsen, C De Micheli, P Conti, A Pinto Bioorganic & Medicinal Chemistry 24 (22), 5741-5747, 2016 | 3 | 2016 |
| Synthesis of Two Epimers of Pseudopaline G Cullia, R Fanelli, R Voulhoux, P Arnoux, F Cavelier European Journal of Organic Chemistry 2020 (26), 3975-3980, 2020 | | 2020 |
| Development of covalent inhibitors of Plasmodium falciparum glyceraldehyde-3-phosphate dehydrogenase with antiparasitic activity in vitro A Galbiati, G Cullia, S Bruno, M Margiotta, S Parapini, D Taramelli, ... Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry …, 2018 | | 2018 |
| ENZYME INHIBITORS AS POTENTIAL ANTIPARASITIC AGENTS G Cullia Università degli Studi di Milano, 2017 | | 2017 |
| Design, synthesis and biological characterization of PfGAPDH inhibitors G Cullia, A Pinto, S Bruno, S Parapini, L Tamborini, A Mozzarelli, ... | | 2016 |
| Synthesis and biological evaluation of new ligands designed to selectively interact with kainate receptors G Cullia, F Mastronardi, A Pinto, L Tamborini, L Marconi, C De Micheli, ... | | 2016 |
| Design and synthesis of novel enzyme inhibitors as potential antiparasitic agents G Cullia | | 2016 |
