Design of radioiodinated pharmaceuticals: structural features affecting metabolic stability towards in vivo deiodination L Cavina, D van der Born, PHM Klaren, MC Feiters, OC Boerman, ... European journal of organic chemistry 2017 (24), 3387-3414, 2017 | 74 | 2017 |
Versatile Picklocks To Access All Opioid Receptors: Tuning the Selectivity and Functional Profile of the Cyclotetrapeptide c[Phe-d-Pro-Phe-Trp] (CJ-15,208) R De Marco, A Bedini, S Spampinato, L Cavina, E Pirazzoli, L Gentilucci Journal of Medicinal Chemistry 59 (19), 9255-9261, 2016 | 22 | 2016 |
Stable pantothenamide bioisosteres: novel antibiotics for Gram-positive bacteria PAM Jansen, DA van Der Krieken, PNM Botman, RH Blaauw, L Cavina, ... The Journal of Antibiotics 72 (9), 682-692, 2019 | 21 | 2019 |
Easy preparation of dehydroalanine building blocks equipped with oxazolidin-2-one chiral auxiliaries, and applications to the stereoselective synthesis of substituted tryptophans R De Marco, L Cavina, A Greco, L Gentilucci Amino Acids 46, 2823-2839, 2014 | 16 | 2014 |
Orthoflaviviral Inhibitors in Clinical Trials, Preclinical In Vivo Efficacy Targeting NS2B-NS3 and Cellular Antiviral Activity via Competitive Protease Inhibition L Cavina, MJ Bouma, D Gironés, MC Feiters Molecules 29 (17), 4047, 2024 | | 2024 |
Opioid activity profiles of peptides containing overlapping portions of CJ-15,208 and CycloEM, and identification of the bioactive conformations R DE MARCO, E Pirazzoli, L Cavina, A Tolomelli, A Bedini, S Spampinato, ... Programme and Abstracts, O8-O8, 2013 | | 2013 |