Παρακολούθηση
Tihomir Tomasic
Tihomir Tomasic
University of Ljubljana, Faculty of Pharmacy
Η διεύθυνση ηλεκτρονικού ταχυδρομείου έχει επαληθευτεί στον τομέα ffa.uni-lj.si - Αρχική σελίδα
Τίτλος
Παρατίθεται από
Παρατίθεται από
Έτος
Rhodanine as a privileged scaffold in drug discovery
T Tomasic, LP Masic
Current Medicinal Chemistry 16 (13), 1596-1629, 2009
3502009
Rhodanine as a scaffold in drug discovery: a critical review of its biological activities and mechanisms of target modulation
T Tomašić, L Peterlin Mašič
Expert opinion on drug discovery 7 (7), 549-560, 2012
1982012
Efflux pump inhibitors of clinically relevant multidrug resistant bacteria
A Lamut, L Peterlin Mašič, D Kikelj, T Tomašič
Medicinal Research Reviews 39 (6), 2460-2504, 2019
1802019
Discovery of benzothiazole scaffold-based DNA gyrase B inhibitors
M Gjorgjieva, T Tomasic, M Barancokova, S Katsamakas, J Ilas, ...
Journal of medicinal chemistry 59 (19), 8941-8954, 2016
1412016
Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site
T Tomasic, S Katsamakas, Z Hodnik, J Ilaš, M Brvar, T Solmajer, ...
Journal of medicinal chemistry 58 (14), 5501-5521, 2015
1352015
Prospects for developing new antibacterials targeting bacterial type IIA topoisomerases
T Tomašić, L Peterlin Masic
Current topics in medicinal chemistry 14 (1), 130-151, 2014
1342014
Xanthine oxidase inhibitors beyond allopurinol and febuxostat; an overview and selection of potential leads based on in silico calculated physico-chemical properties, predicted …
A Šmelcerović, K Tomović, Ž Šmelcerović, Ž Petronijević, G Kocić, ...
European journal of medicinal chemistry 135, 491-516, 2017
1272017
Discovery of novel 5-benzylidenerhodanine and 5-benzylidenethiazolidine-2, 4-dione inhibitors of MurD ligase
N Zidar, T Tomašić, R Šink, V Rupnik, A Kovac, S Turk, D Patin, ...
Journal of medicinal chemistry 53 (18), 6584-6594, 2010
1272010
5‐Benzylidenethiazolidin‐4‐ones as multitarget inhibitors of bacterial Mur ligases
T Tomašić, N Zidar, A Kovač, S Turk, M Simčič, D Blanot, ...
ChemMedChem: Chemistry Enabling Drug Discovery 5 (2), 286-295, 2010
942010
Synthesis and antibacterial activity of 5-ylidenethiazolidin-4-ones and 5-benzylidene-4, 6-pyrimidinediones
T Tomašić, N Zidar, M Mueller-Premru, D Kikelj, LP Mašič
European Journal of Medicinal Chemistry 45 (4), 1667-1672, 2010
872010
ATP-binding site of bacterial enzymes as a target for antibacterial drug design
V Škedelj, T Tomašić, LP Mašič, A Zega
Journal of medicinal chemistry 54 (4), 915-929, 2011
712011
N-Phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATP Competitive DNA Gyrase B Inhibitors: Design, Synthesis, and Evaluation
N Zidar, H Macut, T Tomasic, M Brvar, S Montalvao, P Tammela, ...
Journal of medicinal chemistry 58 (15), 6179-6194, 2015
692015
Synthesis and biological evaluation of hybrid quinolone-based quaternary ammonium antibacterial agents
J Fedorowicz, J Sączewski, A Konopacka, K Waleron, D Lejnowski, ...
European Journal of Medicinal Chemistry 179, 576-590, 2019
682019
Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors
Ž Jakopin, J Ilaš, M Barančoková, M Brvar, P Tammela, MS Dolenc, ...
European Journal of Medicinal Chemistry 130, 171-184, 2017
672017
Synthesis and Evaluation of N‐Phenylpyrrolamides as DNA Gyrase B Inhibitors
M Durcik, P Tammela, M Barančoková, T Tomašič, J Ilaš, D Kikelj, N Zidar
ChemMedChem 13 (2), 186-198, 2018
662018
Antioxidant and anti-inflammatory properties of 1, 2, 4-oxadiazole analogs of resveratrol
M Gobec, T Tomašič, T Markovič, I Mlinarič-Raščan, MS Dolenc, ...
Chemico-Biological Interactions 240, 200-207, 2015
652015
Dual Inhibitor of MurD and MurE Ligases from Escherichia coli and Staphylococcus aureus
T Tomašić, R Šink, N Zidar, A Fic, C Contreras-Martel, A Dessen, ...
ACS Medicinal Chemistry Letters 3 (8), 626-630, 2012
632012
Structure-Based Design of a New Series of d-Glutamic Acid Based Inhibitors of Bacterial UDP-N-acetylmuramoyl-l-alanine:d-glutamate Ligase (MurD)
T Tomašić, N Zidar, R Sink, A Kovač, D Blanot, C Contreras-Martel, ...
Journal of medicinal chemistry 54 (13), 4600-4610, 2011
632011
Synthesis and biological evaluation of new glutamic acid-based inhibitors of MurD ligase
T Tomašić, N Zidar, V Rupnik, A Kovač, D Blanot, S Gobec, D Kikelj, ...
Bioorganic & Medicinal Chemistry Letters 19 (1), 153-157, 2009
632009
Benzothiazole-based compounds in antibacterial drug discovery
M Gjorgjieva, T Tomašič, D Kikelj, LP Mašič
Current medicinal chemistry 25 (38), 5218-5236, 2018
622018
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