A synthetic approach for the rapid preparation of BODIPY conjugates and their use in imaging of cellular drug uptake and distribution S Krajcovicova, J Stankova, P Dzubak, M Hajduch, M Soural, M Urban Chemistry–A European Journal 24 (19), 4957-4966, 2018 | 54 | 2018 |
Solid-phase synthesis for thalidomide-based proteolysis-targeting chimeras (PROTAC) S Krajcovicova, R Jorda, D Hendrychova, V Krystof, M Soural Chemical Communications 55 (7), 929-932, 2019 | 52 | 2019 |
Modulation of FLT3-ITD and CDK9 in acute myeloid leukaemia cells by novel proteolysis targeting chimera (PROTAC) E Řezníčková, S Krajčovičová, M Peřina, M Kovalová, M Soural, V Kryštof European Journal of Medicinal Chemistry 243, 114792, 2022 | 25 | 2022 |
Triterpenic azines, a new class of compounds with selective cytotoxicity to leukemia cells CCRF-CEM J Pokorny, S Krajcovicova, M Hajduch, M Holoubek, S Gurska, P Dzubak, ... Future Medicinal Chemistry 10 (5), 483-491, 2018 | 22 | 2018 |
Diastereoselective flexible synthesis of carbocyclic C-nucleosides L Maier, P Khirsariya, O Hylse, SK Adla, L Černová, M Poljak, ... The Journal of Organic Chemistry 82 (7), 3382-3402, 2017 | 19 | 2017 |
Tryptophan in Multicomponent Petasis Reactions for Peptide Stapling and Late‐Stage Functionalisation S Krajcovicova, DR Spring Angewandte Chemie International Edition 62 (34), e202307782, 2023 | 17 | 2023 |
1, 4, 6-Trisubstituted imidazo [4, 5-c] pyridines as inhibitors of Bruton’s tyrosine kinase S Krajčovičová, R Jorda, D Vanda, M Soural, V Kryštof European Journal of Medicinal Chemistry 211, 113094, 2021 | 16 | 2021 |
Solid-phase synthetic strategies for the preparation of purine derivatives S Krajcovicova, M Soural ACS Combinatorial Science 18 (7), 371-386, 2016 | 14 | 2016 |
Disulfide re-bridging reagents for single-payload antibody-drug conjugates TA King, SJ Walsh, M Kapun, T Wharton, S Krajcovicova, MS Glossop, ... Chemical Communications 59 (65), 9868-9871, 2023 | 10 | 2023 |
A stepwise approach for the synthesis of folic acid conjugates with protein kinase inhibitors S Krajčovičová, T Gucky, D Hendrychova, V Krystof, M Soural The Journal of Organic Chemistry 82 (24), 13530-13541, 2017 | 10 | 2017 |
A cell-active cyclic peptide targeting the Nrf2/Keap1 protein–protein interaction J Iegre, S Krajcovicova, A Gunnarsson, L Wissler, H Käck, A Luchniak, ... Chemical Science 14 (39), 10800-10805, 2023 | 5 | 2023 |
Scaffold hopping of the SYK inhibitor entospletinib leads to broader targeting of the BCR signalosome R Jorda, S Krajčovičová, P Králová, M Soural, V Kryštof European Journal of Medicinal Chemistry 204, 112636, 2020 | 5 | 2020 |
Configuration-dependent medium-sized ring formation: chiral molecular framework with three-dimensional architecture N Cankarova, A La Venia, S Krajcovicova, V Krchnak The Journal of Organic Chemistry 84 (2), 636-644, 2018 | 3 | 2018 |
Site-selective peptide functionalisation mediated via vinyl-triazine linchpins JD Sydenham, H Seki, S Krajcovicova, L Zeng, T Schober, T Deingruber, ... Chemical Communications 60 (6), 706-709, 2024 | 2 | 2024 |
[68Ga]Ga-DFO-c(RGDyK): Synthesis and Evaluation of Its Potential for Tumor Imaging in Mice S Krajcovicova, A Daniskova, K Bendova, Z Novy, M Soural, M Petrik International Journal of Molecular Sciences 22 (14), 7391, 2021 | 2 | 2021 |
Polymer-supported synthesis of N-substituted anthranilates as the building blocks for preparation of N-arylated 3-hydroxyquinolin-4 (1 H)-ones S Krajčovičová, J Hlaváč, K Vychodilová RSC advances 11 (16), 9362-9365, 2021 | 2 | 2021 |
Mitsunobu C-alkylation of β-alkoxycarbonyl 2-nitrobenzenesulfones and its use for the rapid synthesis of novel benzothiazine derivatives M Drabikova, S Krajčovičová, M Soural Tetrahedron 73 (44), 6296-6306, 2017 | 2 | 2017 |
Ideas Behind the Tryptophan‐Mediated Petasis Reaction (TMPR) Concept for Peptide Stapling S Krajcovicova ChemMedChem, e202400148, 2024 | 1 | 2024 |