Novel 1,2,3-Triazole Derivatives for Use against Mycobacterium tuberculosis H37Rv (ATCC 27294) Strain N Boechat, VF Ferreira, SB Ferreira, MLG Ferreira, FC da Silva, ... Journal of medicinal chemistry 54 (17), 5988-5999, 2011 | 323 | 2011 |
The clinically approved antiviral drug sofosbuvir inhibits Zika virus replication CQ Sacramento, GR de Melo, CS de Freitas, N Rocha, LVB Hoelz, ... Scientific reports 7 (1), 40920, 2017 | 249 | 2017 |
Yellow fever virus is susceptible to sofosbuvir both in vitro and in vivo CS de Freitas, LM Higa, CQ Sacramento, AC Ferreira, PA Reis, ... PLoS neglected tropical diseases 13 (1), e0007072, 2019 | 112 | 2019 |
In vitro antiviral activity of the anti-HCV drugs daclatasvir and sofosbuvir against SARS-CoV-2, the aetiological agent of COVID-19 CQ Sacramento, N Fintelman-Rodrigues, JR Temerozo, APD Da Silva, ... Journal of Antimicrobial Chemotherapy 76 (7), 1874-1885, 2021 | 110 | 2021 |
Beyond Members of the Flaviviridae Family, Sofosbuvir Also Inhibits Chikungunya Virus Replication AC Ferreira, PA Reis, CS de Freitas, CQ Sacramento, L Villas Bôas Hoelz, ... Antimicrobial agents and chemotherapy 63 (2), 10.1128/aac. 01389-18, 2019 | 103 | 2019 |
New Trifluoromethyl Triazolopyrimidines as Anti-Plasmodiumfalciparum Agents N Boechat, LCS Pinheiro, TS Silva, ACC Aguiar, AS Carvalho, MM Bastos, ... Molecules 17 (7), 8285-8302, 2012 | 74 | 2012 |
Efavirenz a nonnucleoside reverse transcriptase inhibitor of first-generation: Approaches based on its medicinal chemistry MM Bastos, CCP Costa, TC Bezerra, FC da Silva, N Boechat European journal of medicinal chemistry 108, 455-465, 2016 | 62 | 2016 |
Pyrroles as privileged scaffolds in the search for new potential HIV inhibitors MCAD Bianco, DILF Marinho, LVB Hoelz, MM Bastos, N Boechat Pharmaceuticals 14 (9), 893, 2021 | 54 | 2021 |
Novel Selective Inhibitor of Leishmania (Leishmania) amazonensis Arginase ER da Silva, N Boechat, LCS Pinheiro, MM Bastos, CCP Costa, ... Chemical biology & drug design 86 (5), 969-978, 2015 | 54 | 2015 |
Design, synthesis and pharmacological evaluation of HIV-1 reverse transcriptase inhibition of new indolin-2-ones N Boechat, WB Kover, V Bongertz, MM Bastos, NC Romeiro, ... Medicinal Chemistry 3 (6), 533-542, 2007 | 51 | 2007 |
New pentasubstituted pyrrole hybrid atorvastatin–quinoline derivatives with antiplasmodial activity RCC Carvalho, WA Martins, TP Silva, CR Kaiser, MM Bastos, ... Bioorganic & medicinal chemistry letters 26 (8), 1881-1884, 2016 | 50 | 2016 |
Design, synthesis, and biological evaluation of new 3-hydroxy-2-oxo-3-trifluoromethylindole as potential HIV-1 reverse transcriptase inhibitors N Boechat, WB Kover, MM Bastos, NC Romeiro, ASC Silva, FC Santos, ... Medicinal Chemistry Research 15, 492-510, 2007 | 43 | 2007 |
Repurposing strategies for Chagas disease therapy: the effect of imatinib and derivatives against Trypanosoma cruzi MR Simões-Silva, JS De Araújo, RB Peres, PB Da Silva, MM Batista, ... Parasitology 146 (8), 1006-1012, 2019 | 34 | 2019 |
O uso de porfirinas em terapia fotodinâmica no tratamento da leishmaniose cutânea MM Bastos, N Boechat, ATPC Gomes, MG Neves, JAS Cavaleiro Revista Virtual de Química 4 (3), 257-267, 2012 | 32 | 2012 |
Trifluoromethylation of carbonyl compounds N Boechat, MM Bastos Current Organic Synthesis 7 (5), 403-413, 2010 | 27 | 2010 |
N-Acyl-3, 3-difluoro-2-oxoindoles as versatile intermediates for the preparation of different 2, 2-difluorophenylacetic derivatives N Boechat, WB Kover, MM Bastos, AC Pinto, LC Maciel, LMU Mayer, ... Journal of the Brazilian Chemical Society 19, 445-457, 2008 | 26 | 2008 |
Quimioterapia antileishmania: uma revisão da literatura MM Bastos, N Boechat, LVB Hoelz, AP de Oliveira Revista Virtual de Química 8 (6), 2072-2104, 2016 | 22 | 2016 |
New imatinib derivatives with antiproliferative activity against A549 and K562 cancer cells A Oliveira, S Moura, L Pimentel, J Neto, R Dantas, F Silva-Jr, M Bastos, ... Molecules 27 (3), 750, 2022 | 19 | 2022 |
Imatinib derivatives as inhibitors of K562 cells in chronic myeloid leukemia LD Azevedo, MM Bastos, FC Vasconcelos, LVB Hoelz, FPS Junior, ... Medicinal Chemistry Research 26, 2929-2941, 2017 | 17 | 2017 |
Antimalarial and anti-inflammatory activities of new chloroquine and primaquine hybrids: Targeting the blockade of malaria parasite transmission N Boechat, RCC Carvalho, GF Maria de Lourdes, JP Coutinho, PM Sa, ... Bioorganic & Medicinal Chemistry 28 (24), 115832, 2020 | 16 | 2020 |