| The versatility of boron in biological target engagement DB Diaz, AK Yudin Nature Chemistry 9 (8), 731-742, 2017 | 282 | 2017 |
| Conformational Control of Macrocycles by Remote Structural Modification: Focus Review SD Appavoo, S Huh, DB Diaz, AK Yudin Chemical reviews 119 (17), 9724-9752, 2019 | 117 | 2019 |
| Synthesis of aminoboronic acid derivatives from amines and amphoteric boryl carbonyl compounds DB Diaz, CCG Scully, SK Liew, S Adachi, P Trinchera, JD St. Denis, ... Angewandte Chemie 128 (41), 12849-12853, 2016 | 78 | 2016 |
| Nanomolar-potency small molecule inhibitor of STAT5 protein AA Cumaraswamy, AM Lewis, M Geletu, A Todic, DB Diaz, XR Cheng, ... ACS medicinal chemistry letters 5 (11), 1202-1206, 2014 | 74 | 2014 |
| Amine hemilability enables boron to mechanistically resemble either hydride or proton CF Lee, DB Diaz, A Holownia, SJ Kaldas, SK Liew, GE Garrett, T Dudding, ... Nature Chemistry 10 (10), 1062-1070, 2018 | 57 | 2018 |
| Illuminating the dark conformational space of macrocycles using dominant rotors DB Diaz, SD Appavoo, AF Bogdanchikova, Y Lebedev, TJ McTiernan, ... Nature chemistry 13 (3), 218-225, 2021 | 54 | 2021 |
| Multicomponent mapping of boron chemotypes furnishes selective enzyme inhibitors J Tan, AB Cognetta III, DB Diaz, KM Lum, S Adachi, S Kundu, BF Cravatt, ... Nature communications 8 (1), 1760, 2017 | 51 | 2017 |
| De novo design of boron-based peptidomimetics as potent inhibitors of human ClpP in the presence of human ClpX J Tan, JJ Grouleff, Y Jitkova, DB Diaz, EC Griffith, W Shao, ... Journal of Medicinal Chemistry 62 (13), 6377-6390, 2019 | 46 | 2019 |
| Carboxyboronate: a versatile C1 building block A Holownia, CH Tien, DB Diaz, RT Larson, AK Yudin Angewandte Chemie 131 (42), 15292-15297, 2019 | 38 | 2019 |
| Conformationally stable peptide macrocycles assembled using the Petasis borono-Mannich reaction A Yamaguchi, SJ Kaldas, SD Appavoo, DB Diaz, AK Yudin Chemical Communications 55 (71), 10567-10570, 2019 | 24 | 2019 |
| Reversible covalent interactions of β-aminoboronic acids with carbohydrate derivatives GE Garrett, DB Diaz, AK Yudin, MS Taylor Chemical Communications 53 (11), 1809-1812, 2017 | 23 | 2017 |
| Effect of γ-substituted proline derivatives on the performance of the peptidic catalyst H-dPro-pro-Glu-NH2 T Schnitzer, H Wennemers Synthesis 50 (22), 4377-4382, 2018 | 16 | 2018 |
| Identification and characterization of the first fragment hits for SETDB1 Tudor domain P Mader, R Mendoza-Sanchez, A Iqbal, A Dong, E Dobrovetsky, ... Bioorganic & Medicinal Chemistry 27 (17), 3866-3878, 2019 | 14 | 2019 |
| Borylated oximes: versatile building blocks for organic synthesis SK Liew, A Holownia, DB Diaz, PA Cistrone, PE Dawson, AK Yudin Chemical Communications 53 (81), 11237-11240, 2017 | 12 | 2017 |
| Navigating complex peptide structures using macrocycle conformational maps TJ McTiernan, DB Diaz, GJ Saunders, F Sprang, AK Yudin RSC Chemical Biology 3 (6), 739-747, 2022 | 11 | 2022 |
| Synthesis of Fluorinated Aminoalkylboronic Acids from Amphoteric α‐Boryl Aldehydes HS Soor, DB Diaz, KI Burton, AK Yudin Angewandte Chemie 133 (30), 16502-16507, 2021 | 7 | 2021 |
| Grafting Bis (heteroaryl) Motifs into ring structures CN Apte, DB Diaz, T Adrianov, AK Yudin European Journal of Organic Chemistry 2020 (31), 5029-5033, 2020 | 7 | 2020 |
| Solid‐phase synthesis of peptide β‐aminoboronic acids HS Soor, J Hansen, DB Diaz, S Appavoo, AK Yudin Peptide Science 111 (1), e24072, 2019 | 7 | 2019 |
| Synthesis and Application of Constrained Amidoboronic Acids Using Amphoteric Boron-Containing Building Blocks HS Soor, DB Diaz, KY Tsui, K Calvopina, M Bielinski, DJ Tantillo, ... The Journal of Organic Chemistry 87 (1), 94-102, 2021 | 5 | 2021 |
| A Boron Scan of Ethyl Acetoacetate Leads to Versatile Building Blocks A Trofimova, B White, DB Diaz, MJ Širvinskas, A Lough, T Dudding, ... Angewandte Chemie 136 (15), e202319842, 2024 | 3 | 2024 |