Discovery of an α-amino C–H arylation reaction using the strategy of accelerated serendipity A McNally, CK Prier, DWC MacMillan Science 334 (6059), 1114-1117, 2011 | 1043 | 2011 |
Enantioselective organocatalysis MJ Gaunt, CCC Johansson, A McNally, NT Vo Drug Discovery Today 12 (1-2), 8-27, 2007 | 766 | 2007 |
Palladium-catalysed C–H activation of aliphatic amines to give strained nitrogen heterocycles A McNally, B Haffemayer, BSL Collins, MJ Gaunt Nature 510 (7503), 129-133, 2014 | 539 | 2014 |
Selective functionalization of pyridines via heterocyclic phosphonium salts MC Hilton, RD Dolewski, A McNally Journal of the American Chemical Society 138 (42), 13806-13809, 2016 | 201 | 2016 |
Heterobiaryl synthesis by contractive C–C coupling via P (V) intermediates MC Hilton, X Zhang, BT Boyle, JV Alegre-Requena, RS Paton, A McNally Science 362 (6416), 799-804, 2018 | 190 | 2018 |
A general strategy for site-selective incorporation of deuterium and tritium into pyridines, diazines, and pharmaceuticals JL Koniarczyk, D Hesk, A Overgard, IW Davies, A McNally Journal of the American Chemical Society 140 (6), 1990-1993, 2018 | 176 | 2018 |
Organocatalytic C–H bond arylation of aldehydes to bis-heteroaryl ketones QY Toh, A McNally, S Vera, N Erdmann, MJ Gaunt Journal of the American Chemical Society 135 (10), 3772-3775, 2013 | 152 | 2013 |
Phosphorus-mediated sp2–sp3 couplings for C–H fluoroalkylation of azines X Zhang, KG Nottingham, C Patel, JV Alegre-Requena, JN Levy, ... Nature 594 (7862), 217-222, 2021 | 108 | 2021 |
Phosphonium Salts as Pseudohalides: Regioselective Nickel‐Catalyzed Cross‐Coupling of Complex Pyridines and Diazines X Zhang, A McNally Angewandte Chemie 129 (33), 9965-9968, 2017 | 106 | 2017 |
A counteranion triggered arylation strategy using diaryliodonium fluorides L Chan, A McNally, QY Toh, A Mendoza, MJ Gaunt Chemical Science 6 (2), 1277-1281, 2015 | 93 | 2015 |
Late-stage C–H functionalization of azines CM Josephitis, HMH Nguyen, A McNally Chemical reviews 123 (12), 7655-7691, 2023 | 86 | 2023 |
A unified approach to couple aromatic heteronucleophiles to azines and pharmaceuticals RG Anderson, BM Jett, A McNally Angewandte Chemie International Edition 57 (38), 12514-12518, 2018 | 79 | 2018 |
Cobalt-Catalyzed Alkylation of Drug-Like Molecules and Pharmaceuticals Using Heterocyclic Phosphonium Salts X Zhang, A McNally ACS catalysis 9 (6), 4862-4866, 2019 | 77 | 2019 |
A Strategy to Aminate Pyridines, Diazines, and Pharmaceuticals via Heterocyclic Phosphonium Salts C Patel, M Mohnike, MC Hilton, A McNally Organic letters 20 (9), 2607-2610, 2018 | 76 | 2018 |
4-Selective pyridine functionalization reactions via heterocyclic phosphonium salts RD Dolewski, MC Hilton, A McNally Synlett 29 (01), 08-14, 2018 | 76 | 2018 |
A Pyridine–Pyridine Cross‐Coupling Reaction via Dearomatized Radical Intermediates JL Koniarczyk, JW Greenwood, JV Alegre‐Requena, RS Paton, ... Angewandte Chemie 131 (42), 15024-15028, 2019 | 75 | 2019 |
Halogenation of the 3-position of pyridines through Zincke imine intermediates BT Boyle, JN Levy, L de Lescure, RS Paton, A McNally Science 378 (6621), 773-779, 2022 | 70 | 2022 |
Nonsymmetrical bis-azine biaryls from chloroazines: a strategy using phosphorus ligand-coupling BT Boyle, MC Hilton, A McNally Journal of the American Chemical Society 141 (38), 15441-15449, 2019 | 67 | 2019 |
Site-selective switching strategies to functionalize polyazines RD Dolewski, PJ Fricke, A McNally Journal of the American Chemical Society 140 (25), 8020-8026, 2018 | 63 | 2018 |
Selective halogenation of pyridines using designed phosphine reagents JN Levy, JV Alegre-Requena, R Liu, RS Paton, A McNally Journal of the American Chemical Society 142 (25), 11295-11305, 2020 | 60 | 2020 |