Design of a stable cyclic peptide analgesic derived from sunflower seeds that targets the κ-opioid receptor for the treatment of chronic abdominal pain E Muratspahić, N Tomašević, J Koehbach, L Duerrauer, S Hadžić, ... Journal of medicinal chemistry 64 (13), 9042-9055, 2021 | 24 | 2021 |
Plant-derived cyclotides modulate κ-opioid receptor signaling E Muratspahić, N Tomašević, S Nasrollahi-Shirazi, J Gattringer, ... Journal of Natural Products 84 (8), 2238-2248, 2021 | 17 | 2021 |
Design and structural validation of peptide–drug conjugate ligands of the kappa-opioid receptor E Muratspahić, K Deibler, J Han, N Tomašević, KB Jadhav, AL Olivé-Marti, ... Nature communications 14 (1), 8064, 2023 | 16 | 2023 |
In vitro Inhibition of HIV-1 by Cyclotide-Enriched Extracts of Viola tricolor C Conzelmann, E Muratspahić, N Tomašević, J Münch, CW Gruber Frontiers in Pharmacology 13, 888961, 2022 | 14 | 2022 |
Development of a selective peptide κ-opioid receptor antagonist by late-stage functionalization with cysteine staples E Muratspahić, AM White, CI Ciotu, N Hochrainer, N Tomašević, ... Journal of Medicinal Chemistry 66 (17), 11843-11854, 2023 | 7 | 2023 |
Flipping the GPCR switch: Structure-based development of selective cannabinoid receptor 2 inverse agonists M Kosar, RC Sarott, DA Sykes, AEG Viray, RM Vitale, N Tomašević, X Li, ... ACS Central Science 10 (5), 956-968, 2024 | 6 | 2024 |
Design, synthesis, conformational analysis, and biological activity of Cα1-to-Cα6 1,4- and 4,1-disubstituted 1H-[1,2,3]triazol-1-yl-bridged oxytocin analogues F Nuti, M Larregola, A Staśkiewicz, B Retzl, N Tomašević, L Macchia, ... Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2254019, 2023 | 2 | 2023 |
Discovery and development of macrocyclic peptide modulators of the cannabinoid 2 receptor N Tomašević, FS Emser, E Muratspahić, J Gattringer, S Hasinger, ... Journal of Biological Chemistry 300 (6), 107330, 2024 | 1 | 2024 |
Chemical synthesis of grafted cyclotides using a “plug and play” approach J Koehbach, E Muratspahić, ZM Ahmed, AM White, N Tomašević, T Durek, ... RSC Chemical Biology, 2024 | 1 | 2024 |