| 3D printing of a heterogeneous copper-based catalyst CR Tubío, J Azuaje, L Escalante, A Coelho, F Guitián, E Sotelo, A Gil Journal of Catalysis 334, 110-115, 2016 | 244 | 2016 |
| An efficient and recyclable 3D printed α-Al2O3 catalyst for the multicomponent assembly of bioactive heterocycles J Azuaje, CR Tubío, L Escalante, M Gómez, F Guitián, A Coelho, ... Applied Catalysis A: General 530, 203-210, 2017 | 113 | 2017 |
| Discovery of 3, 4-Dihydropyrimidin-2 (1 H)-ones As a Novel Class of Potent and Selective A2B Adenosine Receptor Antagonists A Crespo, A El Maatougui, P Biagini, J Azuaje, A Coelho, J Brea, MI Loza, ... ACS medicinal chemistry letters 4 (11), 1031-1036, 2013 | 82 | 2013 |
| Discovery of Potent and Highly Selective A2B Adenosine Receptor Antagonist Chemotypes A El Maatougui, J Azuaje, M Gonzalez-Gomez, G Miguez, A Crespo, ... Journal of medicinal chemistry 59 (5), 1967-1983, 2016 | 75 | 2016 |
| Integrated Ugi-Based Assembly of Functionally, Skeletally, and Stereochemically Diverse 1, 4-Benzodiazepin-2-ones J Azuaje, JM Pérez-Rubio, V Yaziji, A El Maatougui, JC González-Gomez, ... The Journal of organic chemistry 80 (3), 1533-1549, 2015 | 45 | 2015 |
| Clinical validation of blood/brain glutamate grabbing in acute ischemic stroke A da Silva‐Candal, A Pérez‐Díaz, M Santamaría, C Correa‐Paz, ... Annals of Neurology 84 (2), 260-273, 2018 | 43 | 2018 |
| Enantiospecific Recognition at the A2B Adenosine Receptor by Alkyl 2-Cyanoimino-4-substituted-6-methyl-1,2,3,4-tetrahydropyrimidine-5-carboxylates C Carbajales, J Azuaje, A Oliveira, MI Loza, J Brea, MI Cadavid, ... Journal of medicinal chemistry 60 (8), 3372-3382, 2017 | 36 | 2017 |
| Ugi-Based Approaches to Quinoxaline Libraries J Azuaje, A El Maatougui, X García-Mera, E Sotelo ACS combinatorial science 16 (8), 403-411, 2014 | 33 | 2014 |
| X‐Ray Crystallography and Free Energy Calculations Reveal the Binding Mechanism of A2A Adenosine Receptor Antagonists W Jespers, G Verdon, J Azuaje, M Majellaro, H Keränen, X García‐Mera, ... Angewandte Chemie International Edition 59 (38), 16536-16543, 2020 | 31 | 2020 |
| 3,4-Dihydropyrimidin-2(1H)-ones as Antagonists of the Human A2B Adenosine Receptor: Optimization, Structure–Activity Relationship Studies, and … M Majellaro, W Jespers, A Crespo, MJ Núñez, S Novio, J Azuaje, ... Journal of Medicinal Chemistry 64 (1), 458-480, 2020 | 30 | 2020 |
| Copper-Catalyzed Huisgen 1, 3-Dipolar Cycloaddition under Oxidative Conditions: Polymer-Assisted Assembly of 4-Acyl-1-Substituted-1, 2, 3-Triazoles PM Diz, A Coelho, A El Maatougui, J Azuaje, O Caamaño, Á Gil, E Sotelo The Journal of organic chemistry 78 (13), 6540-6549, 2013 | 29 | 2013 |
| Multicomponent Assembly of Diverse Pyrazin-2 (1 H)-one Chemotypes J Azuaje, A El Maatougui, JM Pérez-Rubio, A Coelho, F Fernández, ... The Journal of organic chemistry 78 (9), 4402-4409, 2013 | 29 | 2013 |
| Nitrogen-Walk Approach to Explore Bioisosteric Replacements in a Series of Potent A2B Adenosine Receptor Antagonists A Mallo-Abreu, R Prieto-Díaz, W Jespers, J Azuaje, M Majellaro, ... Journal of Medicinal Chemistry 63 (14), 7721-7739, 2020 | 27 | 2020 |
| Sol-Gel Entrapped Cu in a Silica Matrix: An Efficient Heterogeneous Nanocatalyst for Huisgen and Ullmann Intramolecular Coupling Reactions P Diz, Á Gil, F Guitían, A El Maatougui, J Azuaje, P Pernas, E Sotelo, ... Applied Catalysis A: Genera 502, 86-95, 2015 | 26 | 2015 |
| Supported p-toluenesulfonic acid as a highly robust and eco-friendly isocyanide scavenger J Azuaje, A Coelho, A El Maatougui, JM Blanco, E Sotelo ACS combinatorial science 13 (1), 89-95, 2010 | 26 | 2010 |
| Three-Component Assembly of Structurally Diverse 2-Aminopyrimidine-5-carbonitriles C Val, A Crespo, V Yaziji, A Coelho, J Azuaje, A El Maatougui, ... ACS combinatorial science 15 (7), 370-378, 2013 | 23 | 2013 |
| Discovery and Preliminary SAR of 5-Arylidene-2, 2-dimethyl-1, 3-dioxane-4, 6-diones as Platelet Aggregation Inhibitors A El Maatougui, J Azuaje, A Coelho, E Cano, M Yanez, C Lopez, V Yaziji, ... Combinatorial chemistry & high throughput screening 15 (7), 551-554, 2012 | 20 | 2012 |
| Trifluorinated Pyrimidine-Based A2B Antagonists: Optimization and Evidence of Stereospecific Recognition A Mallo-Abreu, M Majellaro, W Jespers, J Azuaje, O Caamano, ... Journal of Medicinal Chemistry 62 (20), 9315-9330, 2019 | 18 | 2019 |
| Computer-aided design of multi-target ligands at A1R, A2AR and PDE10A, key proteins in neurodegenerative diseases L Kalash, C Val, J Azuaje, MI Loza, F Svensson, A Zoufir, L Mervin, ... Journal of Cheminformatics 9, 1-19, 2017 | 18 | 2017 |
| Effect of Nitrogen Atom Substitution in A3 Adenosine Receptor Binding: N-(4,6-Diarylpyridin-2-yl)acetamides as Potent and Selective Antagonists J Azuaje, W Jespers, V Yaziji, A Mallo, M Majellaro, O Caamano, MI Loza, ... Journal of Medicinal Chemistry 60 (17), 7502-7511, 2017 | 18 | 2017 |
