| Design and Synthesis of some new 2, 4, 6-trisubstituted quinazoline EGFR inhibitors as targeted anticancer agents HA Allam, EE Aly, AK Farouk, AM El Kerdawy, E Rashwan, SES Abbass Bioorganic Chemistry 98, 103726, 2020 | 72 | 2020 |
| Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the … HS Ibrahim, HA Allam, WR Mahmoud, A Bonardi, A Nocentini, P Gratteri, ... European Journal of Medicinal Chemistry 152, 1-9, 2018 | 69 | 2018 |
| Design and synthesis of novel coumarin derivatives as potential acetylcholinesterase inhibitors for Alzheimer's disease KM Amin, DEA Rahman, HA Allam, HH El-Zoheiry Bioorganic Chemistry 110, 104792, 2021 | 32 | 2021 |
| Synthesis and biological evaluation of some novel thiobenzimidazole derivatives as anti-renal cancer agents through inhibition of c-MET kinase HS Ibrahim, ME Albakri, WR Mahmoud, HA Allam, AM Reda, ... Bioorganic chemistry 85, 337-348, 2019 | 29 | 2019 |
| Design, synthesis and biological evaluation of some new 1, 3, 4-thiadiazine-thiourea derivatives as potential antitumor agents against non-small cell lung cancer cells FAF Ragab, SA Abdel-Aziz, M Kamel, AMA Ouf, HA Allam Bioorganic Chemistry 93, 103323, 2019 | 24 | 2019 |
| Application of hydrazino and hydrazido linkers to connect benzenesulfonamides with hydrophilic/phobic tails for targeting the middle region of human carbonic anhydrases active … HA Allam, SH Fahim, MF Abo-Ashour, A Nocentini, ME Elbakry, ... European Journal of Medicinal Chemistry 179, 547-556, 2019 | 22 | 2019 |
| Synthesis and Vasodilator Activity of Some pyridazin-3(2H)-one Based Compounds HA Allam, AA Kamel, M El-Daly, RF George Future Medicinal Chemistry 12 (1), 37-50, 2020 | 20 | 2020 |
| Design and synthesis of novel pyridopyrimidine derivatives with anchoring non-coplanar aromatic extensions of EGFR inhibitory activity AAM Eissa, KFM Aljamal, HS Ibrahim, HA Allam Bioorganic Chemistry 116, 105318, 2021 | 19 | 2021 |
| Natural inspired ligustrazine-based SLC-0111 analogues as novel carbonic anhydrase inhibitors DM Elimam, WM Eldehna, R Salem, A Bonardi, A Nocentini, ... European Journal of Medicinal Chemistry 228, 114008, 2022 | 18 | 2022 |
| Design and synthesis of some new 6-bromo-2-(pyridin-3-yl)-4-substituted quinazolines as multi tyrosine kinase inhibitors AK Farouk, HA Allam, E Rashwan, RF George, SES Abbas Bioorganic Chemistry 128, 106099, 2022 | 11 | 2022 |
| Design and synthesis of some new benzoylthioureido phenyl derivatives targeting carbonic anhydrase enzymes MAA Najm, WR Mahmoud, AT Taher, SES Abbas, FM Awadallah, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 2702-2709, 2022 | 9 | 2022 |
| 3-Methyl-imidazo [2, 1-b] thiazole derivatives as a new class of antifolates: Synthesis, in vitro/in vivo bio-evaluation and molecular modeling simulations MA Ewida, HA Ewida, MS Ahmed, HA Allam, RI ElBagary, RF George, ... Bioorganic Chemistry 115, 105205, 2021 | 9 | 2021 |
| Design and synthesis of certain 7-Aryl-2-Methyl-3-Substituted Pyrazolo {1, 5-a} Pyrimidines as multikinase inhibitors MA Al-Qadhi, HA Allam, SH Fahim, TAA Yahya, FAF Ragab European journal of medicinal chemistry 262, 115918, 2023 | 7 | 2023 |
| Design, synthesis, in vitro, and in vivo evaluation of novel phthalazinone‐based derivatives as promising acetylcholinesterase inhibitors for treatment of Alzheimer's disease MAF Ezzat, SM Abdelhamid, MA Fouad, HA Abdel‐Aziz, HA Allam Drug Development Research 84 (6), 1231-1246, 2023 | 7 | 2023 |
| Design and synthesis of some new benzoylthioureido benzenesulfonamide derivatives and their analogues as carbonic anhydrase inhibitors KH Oudah, WR Mahmoud, FM Awadallah, AT Taher, SES Abbas, ... Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 12-23, 2023 | 7 | 2023 |
| Discovery of novel quinolin-2-one derivatives as potential GSK-3β inhibitors for treatment of Alzheimer’s disease: Pharmacophore-based design, preliminary SAR, in vitro and in … EA Moustafa, HA Allam, MA Fouad, AM El Kerdawy, NNE El-Sayed, ... Bioorganic Chemistry 146, 107324, 2024 | 6 | 2024 |
| Effect of hydrophobic extension of aryl enaminones and pyrazole-linked compounds combined with sulphonamide, sulfaguanidine, or carboxylic acid functionalities on carbonic … HA Allam, ME Albakry, WR Mahmoud, A Bonardi, SA Moussa, ... Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2201403, 2023 | 6 | 2023 |
| Arylidine extensions of 3-methyl-5-oxo-4, 5-dihydro-1H-pyrazol-benzenesulfonamide derivatives: synthesis, computational simulations and biological evaluation as tumor … HM Metwally, HA Allam, F Baselious, A Bonardi, EM Seif, SA Moussa, ... Bioorganic Chemistry 135, 106492, 2023 | 5 | 2023 |
| Nanomolar potency of imidazo[2,1‐b]thiazole analogs as indoleamine 2,3‐dioxygenase inhibitors MA Ewida, HA Ewida, MS Ahmed, HA Allam, RI ElBagary, RF George, ... Archiv der Pharmazie 354 (11), 2100202, 2021 | 5 | 2021 |
| Novel VEGFR-2 inhibitors as antiangiogenic and apoptotic agents via paracrine and autocrine cascades: Design, synthesis, and biological evaluation DEA Rahman, MA Fouad, ER Mohammed, HH El-Zoheiry, HA Allam Bioorganic Chemistry 139, 106678, 2023 | 2 | 2023 |
