Articles with public access mandates - george fleetLearn more
Not available anywhere: 18
Synthesis and glycosidase inhibition of australine and its fluorinated derivatives
YX Li, Y Shimada, K Sato, A Kato, W Zhang, YM Jia, GWJ Fleet, M Xiao, ...
Organic letters 17 (3), 716-719, 2015
Mandates: National Natural Science Foundation of China
Design and synthesis of labystegines, hybrid iminosugars from LAB and calystegine, as inhibitors of intestinal α-glucosidases: binding conformation and interaction for ntSI
A Kato, ZL Zhang, HY Wang, YM Jia, CY Yu, K Kinami, Y Hirokami, Y Tsuji, ...
The Journal of organic chemistry 80 (9), 4501-4515, 2015
Mandates: National Natural Science Foundation of China
Synthesis of the enantiomers of XYLNAc and LYXNAc: comparison of β-N-acetylhexosaminidase inhibition by the 8 stereoisomers of 2-N-acetylamino-1, 2, 4-trideoxy-1, 4-iminopentitols
EV Crabtree, RF Martínez, S Nakagawa, I Adachi, TD Butters, A Kato, ...
Organic & Biomolecular Chemistry 12 (23), 3932-3943, 2014
Mandates: Cancer Research UK, UK Engineering and Physical Sciences Research Council …
3‐Hydroxyazetidine Carboxylic Acids: Non‐Proteinogenic Amino Acids for Medicinal Chemists
AFG Glawar, SF Jenkinson, AL Thompson, S Nakagawa, A Kato, ...
ChemMedChem 8 (4), 658-666, 2013
Mandates: Cancer Research UK
Synthesis from d-Altrose of (5R,6R,7R,8S)-5,7-Dihydroxy-8-hydroxymethylconidine and 2,4-Dideoxy-2,4-imino-d-glucitol, Azetidine Analogues of Swainsonine and 1,4 …
N Araújo, SF Jenkinson, RF Martínez, AFG Glawar, MR Wormald, ...
Organic letters 14 (16), 4174-4177, 2012
Mandates: Cancer Research UK, Government of Spain
Gem-difluoromethylated and trifluoromethylated derivatives of DMDP-related iminosugars: Synthesis and glycosidase inhibition
YX Li, K Kinami, Y Hirokami, A Kato, JK Su, YM Jia, GWJ Fleet, CY Yu
Organic & Biomolecular Chemistry 14 (7), 2249-2263, 2016
Mandates: National Natural Science Foundation of China
Synthesis and glycosidase inhibition of N-substituted derivatives of 1, 4-dideoxy-1, 4-imino-d-mannitol (DIM)
LF Yang, Y Shimadate, A Kato, YX Li, YM Jia, GWJ Fleet, CY Yu
Organic & Biomolecular Chemistry 18 (5), 999-1011, 2020
Mandates: National Natural Science Foundation of China
Fluorinated and Conformationally Fixed Derivatives of l-HomoDMDP: Synthesis and Glycosidase Inhibition
YX Li, Y Shimada, I Adachi, A Kato, YM Jia, GWJ Fleet, M Xiao, CY Yu
The Journal of Organic Chemistry 80 (10), 5151-5158, 2015
Mandates: National Natural Science Foundation of China
Palladium-catalyzed one-pot stereospecific synthesis of 2-deoxy aryl C-glycosides from glycals and anilines in the presence of tert-butyl nitrite
AK Singh, R Venkatesh, J Kandasamy
Synthesis 51 (22), 4215-4230, 2019
Mandates: Council of Scientific and Industrial Research, India, Department of Science …
5-C-Branched Deoxynojirimycin: Strategy for Designing a 1-Deoxynojirimycin-Based Pharmacological Chaperone with a Nanomolar Affinity for Pompe Disease
A Kato, I Nakagome, U Kanekiyo, TT Lu, YX Li, K Yoshimura, M Kishida, ...
Journal of Medicinal Chemistry 65 (3), 2329-2341, 2022
Mandates: National Natural Science Foundation of China
(3R, 4S, 5R, 6R, 7S)-3, 4, 5, 7-Tetrahydroxyconidine, an azetidine analogue of 6, 7-diepicastanospermine and a conformationally constrained d-deoxyaltronojirimycin, from l …
RF Martínez, N Araújo, SF Jenkinson, S Nakagawa, A Kato, GWJ Fleet
Bioorganic & medicinal chemistry 21 (16), 4813-4819, 2013
Mandates: Government of Spain
A stereoselective transformation of (−)-shikimic acid into (3R, 4S, 5R, 7R)-7-(hydroxymethyl) azepane-3, 4, 5-triol, a potential glycosidase inhibitor
MA Gonzalez-Castro, DL Poole, JC Estevez, GWJ Fleet, RJ Estevez
Tetrahedron: Asymmetry 26 (5-6), 320-323, 2015
Mandates: Government of Spain
Fluorinated radicamine A and B: synthesis and glycosidase inhibition
YX Li, R Iwaki, A Kato, YM Jia, GWJ Fleet, X Zhao, M Xiao, CY Yu
European Journal of Organic Chemistry 2016 (7), 1429-1438, 2016
Mandates: National Natural Science Foundation of China
Introduction of C-alkyl branches to l-iminosugars changes their active site binding orientation
A Kato, I Nakagome, K Yoshimura, U Kanekiyo, M Kishida, K Shinzawa, ...
Organic & Biomolecular Chemistry 20 (36), 7250-7260, 2022
Mandates: National Natural Science Foundation of China
An Efficient Cascade Synthesis of Ethyl 3-Amino-5-oxoisoxazolidine-4-carboxylate Derivatives
R Li, Q Wei, X Wang, Z Ge, R Li
Synthesis 49 (18), 4341-4349, 2017
Mandates: National Natural Science Foundation of China
Divergent Synthesis of Various 2-Aryl Iminocyclitols from (R)-p-Hydroxyphenylglycine
VK Jain
Synthesis 51 (24), 4635-4644, 2019
Mandates: Council of Scientific and Industrial Research, India
Design and synthesis of iso-allo-DNJ and l-isoDALDP derivatives: pursuit of potent and selective inhibitors of α-glucosidase
LF Yang, M Zhang, Y Shimadate, A Kato, TYL Hou, YX Li, YM Jia, ...
Organic & Biomolecular Chemistry 21 (16), 3453-3464, 2023
Mandates: National Natural Science Foundation of China
A Short Synthesis of (2S, 3S, 4R)-Dihydroxyhomoprolines from d-Erythrose-Derived 5, 6-Dihydro-2H-pyran-2-one
DS Freitas, J Noro, A Drogalin, MCS Fernandes, AVM Baptista, ...
Synthesis 51 (13), 2720-2728, 2019
Mandates: Fundação para a Ciência e a Tecnologia, Portugal
Available somewhere: 28
Pharmacological chaperones for human α-N-acetylgalactosaminidase
NE Clark, MC Metcalf, D Best, GWJ Fleet, SC Garman
Proceedings of the National Academy of Sciences 109 (43), 17400-17405, 2012
Mandates: US National Institutes of Health
Scalable Syntheses of Both Enantiomers of DNJNAc and DGJNAc from Glucuronolactone: The Effect of N‐Alkylation on Hexosaminidase Inhibition
AFG Glawar, D Best, BJ Ayers, S Miyauchi, S Nakagawa, ...
Chemistry–A European Journal 18 (30), 9341-9359, 2012
Mandates: Cancer Research UK, Government of Spain
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