Direct synthesis of fluorinated heteroarylether bioisosteres Q Zhou, A Ruffoni, R Gianatassio, Y Fujiwara, E Sella, D Shabat, ... Angewandte Chemie 125 (14), 4041-4044, 2013 | 261 | 2013 |
Practical and regioselective amination of arenes using alkyl amines A Ruffoni, F Juliá, TD Svejstrup, AJ McMillan, JJ Douglas, D Leonori Nature Chemistry 11 (5), 426-433, 2019 | 233 | 2019 |
Synthesis of arylamines via aminium radicals TD Svejstrup, A Ruffoni, F Juliá, VM Aubert, D Leonori Angewandte Chemie 129 (47), 15144-15148, 2017 | 140 | 2017 |
Photoexcited nitroarenes for the oxidative cleavage of alkenes A Ruffoni, C Hampton, M Simonetti, D Leonori Nature 610 (7930), 81-86, 2022 | 117 | 2022 |
Divergent strain‐release amino‐functionalization of [1.1. 1] propellane with electrophilic nitrogen‐radicals JH Kim, A Ruffoni, YSS Al‐Faiyz, NS Sheikh, D Leonori Angewandte Chemie International Edition 59 (21), 8225-8231, 2020 | 117 | 2020 |
The interplay of polar effects in controlling the selectivity of radical reactions A Ruffoni, RC Mykura, M Bietti, D Leonori Nature Synthesis 1 (9), 682-695, 2022 | 84 | 2022 |
Photoinduced olefin diamination with alkylamines S Govaerts, L Angelini, C Hampton, L Malet‐Sanz, A Ruffoni, D Leonori Angewandte Chemie International Edition 59 (35), 15021-15028, 2020 | 83 | 2020 |
Visible-light-mediated reactions of electrophilic radicals with vinyl and allyl trifluoroborates D Fernandez Reina, A Ruffoni, YSS Al-Faiyz, JJ Douglas, NS Sheikh, ... ACS Catalysis 7 (6), 4126-4130, 2017 | 67 | 2017 |
Practical and Selective sp3 C−H Bond Chlorination via Aminium Radicals AJ McMillan, M Sieńkowska, P Di Lorenzo, GK Gransbury, NF Chilton, ... Angewandte Chemie 133 (13), 7208-7215, 2021 | 47 | 2021 |
Photoinduced decarboxylative azidation of cyclic amino acids DC Marcote, R Street-Jeakings, E Dauncey, JJ Douglas, A Ruffoni, ... Organic & Biomolecular Chemistry 17 (7), 1839-1842, 2019 | 43 | 2019 |
2-Amino-3-(phenylsulfanyl) norbornane-2-carboxylate: an appealing scaffold for the Design of Rac1–Tiam1 protein–protein interaction inhibitors A Ruffoni, N Ferri, SK Bernini, C Ricci, A Corsini, I Maffucci, F Clerici, ... Journal of medicinal chemistry 57 (7), 2953-2962, 2014 | 40 | 2014 |
Rational optimization of a transcription factor activation domain inhibitor S Basu, P Martínez-Cristóbal, M Frigolé-Vivas, M Pesarrodona, M Lewis, ... Nature structural & molecular biology 30 (12), 1958-1969, 2023 | 30 | 2023 |
Sulfanyl-methylene-5(4H)-oxazolones and β-sulfanyl-α-nitroacrylates as appealing dienophiles for the synthesis of conformationally constrained cysteine analogues A Ruffoni, A Casoni, S Pellegrino, ML Gelmi, R Soave, F Clerici Tetrahedron 68 (7), 1951-1962, 2012 | 30 | 2012 |
Synthesis of polysubstituted azepanes by dearomative ring expansion of nitroarenes R Mykura, R Sánchez-Bento, E Matador, VK Duong, A Varela, L Angelini, ... Nature Chemistry, 1-9, 2024 | 29 | 2024 |
Model peptides containing the 3-sulfanyl-norbornene amino acid, a conformationally constrained cysteine analogue effective inducer of 3 10-helix secondary structures A Ruffoni, A Contini, R Soave, LL Presti, I Esposto, I Maffucci, D Nava, ... RSC Advances 5 (41), 32643-32656, 2015 | 23 | 2015 |
A Photochemical Strategy for the Conversion of Nitroarenes into Rigidified Pyrrolidine Analogues E Matador, MJ Tilby, I Saridakis, M Pedrón, D Tomczak, J Llaveria, ... Journal of the American Chemical Society 145 (50), 27810-27820, 2023 | 21 | 2023 |
Self-assembled hydrophobic Ala-Aib peptide encapsulating curcumin: a convenient system for water insoluble drugs S Locarno, S Argentiere, A Ruffoni, D Maggioni, R Soave, R Bucci, E Erba, ... RSC advances 10 (17), 9964-9975, 2020 | 17 | 2020 |
Aqueous self-assembly of short hydrophobic peptides containing norbornene amino acid into supramolecular structures with spherical shape A Ruffoni, MV Cavanna, S Argentiere, S Locarno, S Pellegrino, ML Gelmi, ... RSC advances 6 (93), 90754-90759, 2016 | 17 | 2016 |
A strategy for ortho-phenylenediamine synthesis via dearomative-rearomative coupling of nitrobenzenes and amines R Sánchez-Bento, B Roure, J Llaveria, A Ruffoni, D Leonori Chem 9 (12), 3685-3695, 2023 | 15 | 2023 |
A Photochemical Strategy for ortho‐Aminophenol Synthesis via Dearomative‐Rearomative Coupling Between Aryl Azides and Alcohols B Li, A Ruffoni, D Leonori Angewandte Chemie International Edition 62 (52), e202310540, 2023 | 13 | 2023 |