| Highly Selective Dopamine D3 Receptor (D3R) Antagonists and Partial Agonists Based on Eticlopride and the D3R Crystal Structure: New Leads for Opioid … V Kumar, A Bonifazi, MP Ellenberger, TM Keck, E Pommier, R Rais, ... Journal of medicinal chemistry 59 (16), 7634-7650, 2016 | 101 | 2016 |
| Evidence for noncanonical neurotransmitter activation: norepinephrine as a dopamine D2-like receptor agonist M Sánchez-Soto, A Bonifazi, NS Cai, MP Ellenberger, AH Newman, ... Molecular pharmacology 89 (4), 457-466, 2016 | 84 | 2016 |
| Novel and high affinity 2-[(diphenylmethyl) sulfinyl] acetamide (modafinil) analogues as atypical dopamine transporter inhibitors J Cao, RD Slack, OM Bakare, C Burzynski, R Rais, BS Slusher, T Kopajtic, ... Journal of medicinal chemistry 59 (23), 10676-10691, 2016 | 72 | 2016 |
| Toward Understanding the Structural Basis of Partial Agonism at the Dopamine D3 Receptor M Michino, CA Boateng, P Donthamsetti, H Yano, OM Bakare, A Bonifazi, ... Journal of medicinal chemistry 60 (2), 580-593, 2017 | 56 | 2017 |
| Synthesis and pharmacological characterization of novel trans-cyclopropylmethyl-linked bivalent ligands that exhibit selectivity and allosteric pharmacology at the dopamine D3 … V Kumar, AE Moritz, TM Keck, A Bonifazi, MP Ellenberger, CD Sibley, ... Journal of medicinal chemistry 60 (4), 1478-1494, 2017 | 49 | 2017 |
| Novel Bivalent Ligands Based on the Sumanirole Pharmacophore Reveal Dopamine D2 Receptor (D2R) Biased Agonism A Bonifazi, H Yano, MP Ellenberger, L Muller, V Kumar, MF Zou, NS Cai, ... Journal of medicinal chemistry 60 (7), 2890-2907, 2017 | 47 | 2017 |
| Dopamine D4 Receptor-Selective Compounds Reveal Structure–Activity Relationships that Engender Agonist Efficacy TM Keck, RB Free, MM Day, SL Brown, MS Maddaluna, G Fountain, ... Journal of medicinal chemistry 62 (7), 3722-3740, 2019 | 36 | 2019 |
| Development of Novel Tools for Dissection of Central Versus Peripheral Dopamine D2-Like Receptor Signaling in Dysglycemia A Bonifazi, M Ellenberger, ZJ Farino, D Aslanoglou, R Rais, S Pereira, ... Diabetes 73 (9), 1411-1425, 2024 | 1 | 2024 |
| 1299-P: Novel Tools to Dissect the Metabolic Roles of Central and Peripheral Dopamine D2-Like Receptors A Bonifazi, MP Ellenberger, Z Farino, R Rais, J Mantilla-Rivas, ... Diabetes 71 (Supplement_1), 2022 | | 2022 |
| Structural basis of partial agonism at the dopamine D3 receptor M Michino, C Boateng, P Donthamsetti, O Bakare, A Bonifazi, ... ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 251, 2016 | | 2016 |
| DOPAMINE D2, D3, AND D4 RECEPTOR AFFINITIES OF 77-LH-28-1 AND ITS ANALOGUES A Piergentili, F DEL BELLO, M Giannella, G Giorgioni, W Quaglia, ... 33 rd Camerino-Cyprus Symposium. Receptor Chemistry: Reality and Vision, 89-89, 2016 | | 2016 |
Newman Amy HauckNational Institue on Drug Abuse-Intramural Research Program, NIHDirección de correo verificada de intra.nida.nih.gov
