| Synthesis and reactivity of propargylamines in organic chemistry K Lauder, A Toscani, N Scalacci, D Castagnolo Chemical reviews 117 (24), 14091-14200, 2017 | 453 | 2017 |
| Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones D Castagnolo, F Manetti, M Radi, B Bechi, M Pagano, A De Logu, ... Bioorganic & medicinal chemistry 17 (15), 5716-5721, 2009 | 212 | 2009 |
| Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis D Castagnolo, A De Logu, M Radi, B Bechi, F Manetti, M Magnani, ... Bioorganic & medicinal chemistry 16 (18), 8587-8591, 2008 | 190 | 2008 |
| Guanylated diamines, triamines, and polyamines: chemistry and biological properties D Castagnolo, S Schenone, M Botta Chemical reviews 111 (9), 5247-5300, 2011 | 137 | 2011 |
| Antimicrobial drugs bearing guanidine moieties: A review SH Kim, D Semenya, D Castagnolo European Journal of Medicinal Chemistry 216, 113293, 2021 | 111 | 2021 |
| Synthesis and biological evaluation of new taxoids derived from 2-deacetoxytaxinine J M Botta, S Armaroli, D Castagnolo, G Fontana, P Pera, E Bombardelli Bioorganic & medicinal chemistry letters 17 (6), 1579-1583, 2007 | 109 | 2007 |
| Tuberculosis drug discovery: challenges and new horizons GFS Fernandes, AM Thompson, D Castagnolo, WA Denny, ... Journal of Medicinal Chemistry 65 (11), 7489-7531, 2022 | 106 | 2022 |
| Microwave-assisted organocatalytic multicomponent Knoevenagel/hetero Diels–Alder reaction for the synthesis of 2, 3-dihydropyran [2, 3-c] pyrazoles M Radi, V Bernardo, B Bechi, D Castagnolo, M Pagano, M Botta Tetrahedron Letters 50 (47), 6572-6575, 2009 | 103 | 2009 |
| Photo‐biocatalytic one‐pot cascades for the enantioselective synthesis of 1, 3‐mercaptoalkanol volatile sulfur compounds K Lauder, A Toscani, Y Qi, J Lim, SJ Charnock, K Korah, D Castagnolo Angewandte Chemie 130 (20), 5905-5909, 2018 | 91 | 2018 |
| Synthesis of New Linear Guanidines and Macrocyclic Amidinourea Derivatives Endowed with High Antifungal Activity against Candida spp. and Aspergillus spp. F Manetti, D Castagnolo, F Raffi, AT Zizzari, S Rajamaki, S D’Arezzo, ... Journal of medicinal chemistry 52 (23), 7376-7379, 2009 | 82 | 2009 |
| Unveiling the biocatalytic aromatizing activity of monoamine oxidases MAO-N and 6-HDNO: development of chemoenzymatic cascades for the synthesis of pyrroles N Scalacci, GW Black, G Mattedi, NL Brown, NJ Turner, D Castagnolo ACS Catalysis 7 (2), 1295-1300, 2017 | 80 | 2017 |
| Synthesis and biological evaluation of new enantiomerically pure azole derivatives as inhibitors of Mycobacterium tuberculosis D Castagnolo, M Radi, F Dessì, F Manetti, M Saddi, R Meleddu, ... Bioorganic & medicinal chemistry letters 19 (8), 2203-2205, 2009 | 71 | 2009 |
| Discovery of multitarget antivirals acting on both the Dengue virus NS5-NS3 interaction and the host Src/Fyn kinases P Vincetti, F Caporuscio, S Kaptein, A Gioiello, V Mancino, Y Suzuki, ... Journal of medicinal chemistry 58 (12), 4964-4975, 2015 | 65 | 2015 |
| Ligand‐Based Virtual Screening, Parallel Solution‐Phase and Microwave‐Assisted Synthesis as Tools to Identify and Synthesize New Inhibitors of Mycobacterium tuberculosis F Manetti, M Magnani, D Castagnolo, L Passalacqua, M Botta, F Corelli, ... ChemMedChem: Chemistry Enabling Drug Discovery 1 (9), 973-989, 2006 | 62 | 2006 |
| Synthesis of 1, 2, 3-substituted pyrroles from propargylamines via a one-pot tandem enyne cross metathesis–cyclization reaction H Chachignon, N Scalacci, E Petricci, D Castagnolo The Journal of Organic Chemistry 80 (10), 5287-5295, 2015 | 60 | 2015 |
| Design and Synthesis of 1-((1,5-Bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N′-((E)-3,7 … S Bhakta, N Scalacci, A Maitra, AK Brown, S Dasugari, D Evangelopoulos, ... Journal of medicinal chemistry 59 (6), 2780-2793, 2016 | 56 | 2016 |
| Domino alkylation-cyclization reaction of propargyl bromides with thioureas/thiopyrimidinones: a new facile synthesis of 2-aminothiazoles and 5H-thiazolo [3, 2-a] pyrimidin-5-ones D Castagnolo, M Pagano, M Bernardini, M Botta Synlett 2009 (13), 2093-2096, 2009 | 55 | 2009 |
| Pyrimidine derivatives with antitubercular activity V Finger, M Kufa, O Soukup, D Castagnolo, J Roh, J Korabecny European Journal of Medicinal Chemistry 246, 114946, 2023 | 52 | 2023 |
| Intramolecular arylation of amino acid enolates RC Atkinson, DJ Leonard, J Maury, D Castagnolo, N Volz, J Clayden Chemical Communications 49 (84), 9734-9736, 2013 | 52 | 2013 |
| Crotylation versus propargylation: two routes for the synthesis of the C13− C18 fragment of the antibiotic branimycin W Felzmann, D Castagnolo, D Rosenbeiger, J Mulzer The Journal of Organic Chemistry 72 (6), 2182-2186, 2007 | 52 | 2007 |
