| Key Green Chemistry research areas from a pharmaceutical manufacturers’ perspective revisited MC Bryan, PJ Dunn, D Entwistle, F Gallou, SG Koenig, JD Hayler, ... Green Chemistry 20 (22), 5082-5103, 2018 | 542 | 2018 |
| Pharmaceutical roundtable study demonstrates the value of continuous manufacturing in the design of greener processes P Poechlauer, J Colberg, E Fisher, M Jansen, MD Johnson, SG Koenig, ... Organic Process Research & Development 17 (12), 1472-1478, 2013 | 173 | 2013 |
| Targeted drug delivery through the traceless release of tertiary and heteroaryl amines from antibody–drug conjugates LR Staben, SG Koenig, SM Lehar, R Vandlen, D Zhang, J Chuh, SF Yu, ... Nature chemistry 8 (12), 1112-1119, 2016 | 166 | 2016 |
| A deeper shade of green: inspiring sustainable drug manufacturing F Roschangar, J Colberg, PJ Dunn, F Gallou, JD Hayler, SG Koenig, ... Green Chemistry 19 (1), 281-285, 2017 | 126 | 2017 |
| GNE-781, a highly advanced potent and selective bromodomain inhibitor of cyclic adenosine monophosphate response element binding protein, binding protein (CBP) FA Romero, J Murray, KW Lai, V Tsui, BK Albrecht, L An, MH Beresini, ... Journal of Medicinal Chemistry 60 (22), 9162-9183, 2017 | 115 | 2017 |
| An efficient synthesis of enamides from ketones H Zhao, CP Vandenbossche, SG Koenig, SP Singh, RP Bakale Organic Letters 10 (3), 505-507, 2008 | 99 | 2008 |
| Introduction of a process mass intensity metric for biologics K Budzinski, M Blewis, P Dahlin, D D'Aquila, J Esparza, J Gavin, SV Ho, ... New biotechnology 49, 37-42, 2019 | 97 | 2019 |
| Sustainability challenges and opportunities in oligonucleotide manufacturing BI Andrews, FD Antia, SB Brueggemeier, LJ Diorazio, SG Koenig, ... The Journal of Organic Chemistry 86 (1), 49-61, 2020 | 93 | 2020 |
| Inspiring process innovation via an improved green manufacturing metric: iGAL F Roschangar, Y Zhou, DJC Constable, J Colberg, DP Dickson, PJ Dunn, ... Green Chemistry 20 (10), 2206-2211, 2018 | 89 | 2018 |
| Chemoselective sp2-sp3 Cross-Couplings: Iron-Catalyzed Alkyl Transfer to Dihaloaromatics S Malhotra, PS Seng, SG Koenig, AJ Deese, KA Ford Organic letters 15 (14), 3698-3701, 2013 | 67 | 2013 |
| A Transient N− O-Linked Pauson− Khand Strategy for the Synthesis of the Deschloro Carbocyclic Core of the Palau'amines and Styloguanidines SG Koenig, SM Miller, KA Leonard, RS Löwe, BC Chen, DJ Austin Organic Letters 5 (13), 2203-2206, 2003 | 60 | 2003 |
| Visible-light-induced trifluoromethylation of highly functionalized arenes and heteroarenes in continuous flow I Abdiaj, C Bottecchia, J Alcazar, T Noёl Synthesis 49 (22), 4978-4985, 2017 | 59 | 2017 |
| A facile deprotection of secondary acetamides SG Koenig, CP Vandenbossche, H Zhao, P Mousaw, SP Singh, ... Organic Letters 11 (2), 433-436, 2009 | 58 | 2009 |
| The PMI Predictor app to enable green-by-design chemical synthesis A Borovika, J Albrecht, J Li, AS Wells, C Briddell, BR Dillon, LJ Diorazio, ... Nature Sustainability 2 (11), 1034-1040, 2019 | 56 | 2019 |
| Improved iGAL 2.0 metric empowers pharmaceutical scientists to make meaningful contributions to united nations sustainable development goal 12 F Roschangar, J Li, Y Zhou, W Aelterman, A Borovika, J Colberg, ... ACS Sustainable Chemistry & Engineering 10 (16), 5148-5162, 2021 | 52 | 2021 |
| Evaluating the impact of a decade of funding from the green chemistry institute pharmaceutical roundtable SG Koenig, DK Leahy, AS Wells Organic Process Research & Development 22 (10), 1344-1359, 2018 | 48 | 2018 |
| Metal‐Catalyzed Organic Reactions by Resonant Acoustic Mixing L Gonnet, CB Lennox, JL Do, I Malvestiti, SG Koenig, K Nagapudi, ... Angewandte Chemie International Edition 61 (13), e202115030, 2022 | 47 | 2022 |
| A green chemistry continuum for a robust and sustainable active pharmaceutical ingredient supply chain SG Koenig, C Bee, A Borovika, C Briddell, J Colberg, GR Humphrey, ... ACS Sustainable Chemistry & Engineering 7 (20), 16937-16951, 2019 | 47 | 2019 |
| Synthesis of indole-2-carboxylate derivatives via palladium-catalyzed aerobic amination of aryl C–H bonds K Clagg, H Hou, AB Weinstein, D Russell, SS Stahl, SG Koenig Organic letters 18 (15), 3586-3589, 2016 | 47 | 2016 |
| Development of a Large-Scale Stereoselective Process for (1R,4S)-4-(3,4-Dichlorophenyl)-1,2,3,4-tetrahydronaphthalen-1-amine Hydrochloride Z Han, SG Koenig, H Zhao, X Su, SP Singh, RP Bakale Organic process research & development 11 (4), 726-730, 2007 | 44 | 2007 |