| Design, synthesis, modeling studies and biological evaluation of thiazolidine derivatives containing pyrazole core as potential anti-diabetic PPAR-γ agonists and anti … KRA Abdellatif, WAA Fadaly, GM Kamel, YAMM Elshaier, MA El-Magd Bioorganic chemistry 82, 86-99, 2019 | 107 | 2019 |
| New 1, 2, 4-triazole/pyrazole hybrids linked to oxime moiety as nitric oxide donor celecoxib analogs: Synthesis, cyclooxygenase inhibition anti-inflammatory, ulcerogenicity … WAA Fadaly, YAMM Elshaier, EHM Hassanein, KRA Abdellatif Bioorganic Chemistry 98, 103752, 2020 | 81 | 2020 |
| Non-acidic 1, 3, 4-trisubstituted-pyrazole derivatives as lonazolac analogs with promising COX-2 selectivity, anti-inflammatory activity and gastric safety profile KRA Abdellatif, WAA Fadaly, YAMM Elshaier, WAM Ali, GM Kamel Bioorganic Chemistry 77, 568-578, 2018 | 65 | 2018 |
| Synthesis, cyclooxygenase inhibition, anti-inflammatory evaluation and ulcerogenic liability of new 1, 3, 5-triarylpyrazoline and 1, 5-diarylpyrazole derivatives as selective … KRA Abdellatif, EKA Abdelall, WAA Fadaly, GM Kamel Bioorganic & Medicinal Chemistry Letters 26 (2), 406-412, 2016 | 58 | 2016 |
| Thiohydantoin derivatives incorporating a pyrazole core: Design, synthesis and biological evaluation as dual inhibitors of topoisomerase-I and cycloxygenase-2 with anti-cancer … KRA Abdellatif, WAA Fadaly, YA Mostafa, DM Zaher, HA Omar Bioorganic Chemistry 91, 103132, 2019 | 53 | 2019 |
| Synthesis, cyclooxygenase inhibition, and anti-inflammatory evaluation of novel diarylheterocycles with a central pyrazole, pyrazoline, or pyridine ring KRA Abdellatif, EKA Abdelall, WAA Fadaly, GM Kamel Medicinal Chemistry Research 24, 2632-2644, 2015 | 46 | 2015 |
| New 1, 2-diaryl-4-substituted-benzylidene-5-4H-imidazolone derivatives: Design, synthesis and biological evaluation as potential anti-inflammatory and analgesic agents KRA Abdellatif, WAA Fadaly Bioorganic Chemistry 72, 123-129, 2017 | 30 | 2017 |
| Design, synthesis, cyclooxygenase inhibition and biological evaluation of new 1, 3, 5-triaryl-4, 5-dihydro-1H-pyrazole derivatives possessing amino/methanesulfonyl pharmacophore KRA Abdellatif, WAA Fadaly Bioorganic Chemistry 70, 57-66, 2017 | 27 | 2017 |
| Synthesis of novel halogenated triarylpyrazoles as selective COX-2 inhibitors: anti-inflammatory activity, histopatholgical profile and in-silico studies KRA Abdellatif, EKA Abdelall, MB Labib, WAA Fadaly, TH Zidan Bioorganic Chemistry 105, 104418, 2020 | 25 | 2020 |
| Design, synthesis, modeling studies and biological evaluation of pyrazole derivatives linked to oxime and nitrate moieties as nitric oxide donor selective COX-2 and aromatase … WAA Fadaly, YAMM Elshaier, MTM Nemr, KRA Abdellatif Bioorganic Chemistry 134, 106428, 2023 | 21 | 2023 |
| Synthesis, cyclooxygenase inhibition, anti-inflammatory evaluation and ulcerogenic liability of new 1, 5-diarylpyrazole derivatives KRA Abdellatif, WAA Fadaly, WAM Ali, GM Kamel Journal of enzyme inhibition and medicinal chemistry 31 (sup3), 54-60, 2016 | 21 | 2016 |
| Chemistry of 2-vinylindoles: synthesis and applications YAAM Elshaier, MTM Nemr, MS Refaey, WAA Fadaly, A Barakat New Journal of Chemistry 46 (28), 13383-13400, 2022 | 19 | 2022 |
| New pyrazolyl-thiazolidinone/thiazole derivatives as celecoxib/dasatinib analogues with selective COX-2, HER-2 and EGFR inhibitory effects: design, synthesis, anti-inflammatory … WAA Fadaly, TH Zidan, NM Kahk, FEA Mohamed, MM Abdelhakeem, ... Journal of enzyme inhibition and medicinal chemistry 38 (1), 2281262, 2023 | 18 | 2023 |
| New 1,2,3-triazole/1,2,4-triazole hybrids linked to oxime moiety as nitric oxide donor selective COX-2, aromatase, B-RAFV600E and EGFR inhibitors celecoxib … WAA Fadaly, MTM Nemr, TH Zidan, FEA Mohamed, MM Abdelhakeem, ... Journal of Enzyme Inhibition and Medicinal Chemistry 38 (1), 2290461, 2023 | 15 | 2023 |
| Design, synthesis of celecoxib-tolmetin drug hybrids as selective and potent COX-2 inhibitors KRA Abdellatif, EKA Abdelall, MB Labib, WAA Fadaly, TH Zidan Bioorganic chemistry 90, 103029, 2019 | 15 | 2019 |
| Discovery of novel pyrazole based Urea/Thiourea derivatives as multiple targeting VEGFR-2, EGFRWT, EGFRT790M tyrosine kinases and COX-2 Inhibitors, with anti-cancer and anti … WAA Fadaly, MTM Nemr, NM Kahk Bioorganic chemistry 147, 107403, 2024 | 14 | 2024 |
| Synthesis, Cyclooxygenase Inhibition, Anti‐Inflammatory Evaluation, and Ulcerogenic Liability of New 1, 3, 5‐Triarylpyrazoline Derivatives Possessing a Methanesulfonyl … KRA Abdellatif, WAA Fadaly, AA Azouz Archiv der Pharmazie 349 (10), 801-807, 2016 | 13 | 2016 |
| Vicinal diaryl pyrazole with tetrazole/urea scaffolds as selective angiotensin converting enzyme‐1/cyclooxygenase‐2 inhibitors: Design, synthesis, anti‐hypertensive, anti … WAA Fadaly, YAMM Elshaier, FEM Ali, AH El‐Bahrawy, KRA Abdellatif, ... Drug Development Research 85 (4), e22217, 2024 | 6 | 2024 |
| Discovery of novel thiazole derivatives containing pyrazole scaffold as PPAR-γ Agonists, α-Glucosidase, α-Amylase and COX-2 inhibitors; Design, synthesis and in silico study WAA Fadaly, A Elshewy, MTM Nemr, K Abdou, AM Sayed, NM Kahk Bioorganic Chemistry 152, 107760, 2024 | 3 | 2024 |
| Novel benzenesulfonamide derivatives as potential selective carbonic anhydrase IX, XII inhibitors with anti-proliferative activity: Design, synthesis and in silico studies WAA Fadaly, FEA Mohamed, MTM Nemr, AM Sayed, RG Khalil, TH Zidan Bioorganic Chemistry 153, 107881, 2024 | 2 | 2024 |