| Click chemistry reactions in medicinal chemistry: Applications of the 1, 3‐dipolar cycloaddition between azides and alkynes GC Tron, T Pirali, RA Billington, PL Canonico, G Sorba, AA Genazzani Medicinal research reviews 28 (2), 278-308, 2008 | 1313 | 2008 |
| Medicinal chemistry of combretastatin A4: present and future directions GC Tron, T Pirali, G Sorba, F Pagliai, S Busacca, AA Genazzani Journal of medicinal chemistry 49 (11), 3033-3044, 2006 | 783 | 2006 |
| To each his own: isonitriles for all flavors. Functionalized isocyanides as valuable tools in organic synthesis M Giustiniano, A Basso, V Mercalli, A Massarotti, E Novellino, GC Tron, ... Chemical Society Reviews 46 (5), 1295-1357, 2017 | 386 | 2017 |
| Visible light photocatalysis in the late-stage functionalization of pharmaceutically relevant compounds R Cannalire, S Pelliccia, L Sancineto, E Novellino, GC Tron, ... Chemical Society Reviews 50 (2), 766-897, 2021 | 329 | 2021 |
| Rapid synthesis of triazole-modified resveratrol analogues via click chemistry F Pagliai, T Pirali, E Del Grosso, R Di Brisco, GC Tron, G Sorba, ... Journal of medicinal chemistry 49 (2), 467-470, 2006 | 294 | 2006 |
| One-pot synthesis of macrocycles by a tandem three-component reaction and intramolecular [3+ 2] cycloaddition T Pirali, GC Tron, J Zhu Organic Letters 8 (18), 4145-4148, 2006 | 168 | 2006 |
| Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors U Galli, C Travelli, A Massarotti, G Fakhfouri, R Rahimian, GC Tron, ... Journal of medicinal chemistry 56 (16), 6279-6296, 2013 | 167 | 2013 |
| Are 1, 4‐and 1, 5‐Disubstituted 1, 2, 3‐Triazoles Good Pharmacophoric Groups? A Massarotti, S Aprile, V Mercalli, E Del Grosso, G Grosa, G Sorba, ... ChemMedChem 9 (11), 2497-2508, 2014 | 163 | 2014 |
| Synthesis and cytotoxic evaluation of combretafurazans GC Tron, F Pagliai, E Del Grosso, AA Genazzani, G Sorba Journal of medicinal chemistry 48 (9), 3260-3268, 2005 | 150 | 2005 |
| Chemoselective esterification of phenolic acids and alcohols G Appendino, A Minassi, N Daddario, F Bianchi, GC Tron Organic Letters 4 (22), 3839-3841, 2002 | 135 | 2002 |
| A novel potent nicotinamide phosphoribosyltransferase inhibitor synthesized via click chemistry G Colombano, C Travelli, U Galli, A Caldarelli, MG Chini, PL Canonico, ... Journal of medicinal chemistry 53 (2), 616-623, 2010 | 129 | 2010 |
| Macrocyclic Diterpenoids from Euphorbia semiperfoliata G Appendino, S Jakupovic, GC Tron, J Jakupovic, V Milon, M Ballero Journal of natural products 61 (6), 749-756, 1998 | 127 | 1998 |
| Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus M Bassetto, T De Burghgraeve, L Delang, A Massarotti, A Coluccia, ... Antiviral research 98 (1), 12-18, 2013 | 126 | 2013 |
| Recent advances in NAMPT inhibitors: a novel immunotherapic strategy U Galli, G Colombo, C Travelli, GC Tron, AA Genazzani, AA Grolla Frontiers in pharmacology 11, 656, 2020 | 122 | 2020 |
| In vitro metabolism study of combretastatin A-4 in rat and human liver microsomes S Aprile, E Del Grosso, GC Tron, G Grosa Drug metabolism and disposition 35 (12), 2252-2261, 2007 | 111 | 2007 |
| A mimicry of primary amines by bis-secondary diamines as components in the Ugi four-component reaction GB Giovenzana, GC Tron, S Di Paola, IG Menegotto, T Pirali Angewandte Chemie-International Edition 45 (7), 1099-1102, 2006 | 110 | 2006 |
| Replacement of the lactone moiety on podophyllotoxin and steganacin analogues with a 1, 5-disubstituted 1, 2, 3-triazole via ruthenium-catalyzed click chemistry D Imperio, T Pirali, U Galli, F Pagliai, L Cafici, PL Canonico, G Sorba, ... Bioorganic & medicinal chemistry 15 (21), 6748-6757, 2007 | 108 | 2007 |
| An Expeditious Procedure for the Isolation of Ingenol from the Seeds of Euphorbia lathyris G Appendino, GC Tron, G Cravotto, G Palmisano, J Jakupovic Journal of natural products 62 (1), 76-79, 1999 | 108 | 1999 |
| Medicinal chemistry of isocyanides A Massarotti, F Brunelli, S Aprile, M Giustiniano, GC Tron Chemical Reviews 121 (17), 10742-10788, 2021 | 104 | 2021 |
| Regioselective Suzuki coupling of dihaloheteroaromatic compounds as a rapid strategy to synthesize potent rigid combretastatin analogues S Theeramunkong, A Caldarelli, A Massarotti, S Aprile, D Caprioglio, ... Journal of medicinal chemistry 54 (14), 4977-4986, 2011 | 104 | 2011 |