| The role of natural products in drug discovery and development against neglected tropical diseases PM Cheuka, G Mayoka, P Mutai, K Chibale Molecules 22 (1), 58, 2016 | 256 | 2016 |
| Plasmepsin inhibitors in antimalarial drug discovery: medicinal chemistry and target validation (2000 to present) PM Cheuka, G Dziwornu, J Okombo, K Chibale Journal of medicinal chemistry 63 (9), 4445-4467, 2020 | 44 | 2020 |
| New Amidated 3,6-Diphenylated Imidazopyridazines with Potent Antiplasmodium Activity Are Dual Inhibitors of Plasmodium Phosphatidylinositol-4-kinase and … PM Cheuka, L Centani, LB Arendse, S Fienberg, L Wambua, SS Renga, ... ACS Infectious Diseases 7 (1), 34-46, 2020 | 17 | 2020 |
| Cocrystal and salt forms of an imidazopyridazine antimalarial drug lead TJ Noonan, K Chibale, PM Cheuka, SA Bourne, MR Caira Journal of pharmaceutical sciences 108 (7), 2349-2357, 2019 | 16 | 2019 |
| Antiplasmodial imidazopyridazines: structure–activity relationship studies lead to the identification of analogues with improved solubility and hERG profiles PM Cheuka, N Lawrence, D Taylor, S Wittlin, K Chibale Medchemcomm 9 (10), 1733-1745, 2018 | 14 | 2018 |
| Phytochemical screening and in vitro antibacterial activity of Odontonema strictum (Acanthaceae) against selected bacteria LP Luhata, NM Munkombwe, PM Cheuka, H Sikanyika International Journal of Development Research 5 (6), 4655-59, 2015 | 12 | 2015 |
| Structure activity relationship (SAR) of some benzoic acid derivatives from plant origin that exhibit anti-sickling properties in vitro LL Pierre, NM Moses, CM Peter Nat Prod Chem Res 3 (176), 2, 2015 | 12 | 2015 |
| Activity of N-phenylbenzamide analogs against the neglected disease pathogen, Schistosoma mansoni M Kanyanta, C Lengwe, D Mambwe, KR Francisco, LJ Liu, YU Sun, ... Bioorganic & medicinal chemistry letters 82, 129164, 2023 | 9 | 2023 |
| Five solid forms of a potent imidazopyridazine antimalarial drug lead: A preformulation study TJ Noonan, K Chibale, PM Cheuka, M Kumar, SA Bourne, MR Caira Crystal Growth & Design 19 (8), 4683-4697, 2019 | 8 | 2019 |
| Medicinal chemistry progression of antimalarial hits from phenotypic whole cell screening of SoftFocus libraries PM Cheuka, G Mayoka, J Okombo, K Chibale Annual reports in medicinal chemistry 53, 25-71, 2019 | 8 | 2019 |
| Structure–activity relationship studies of antiplasmodial aminomethylthiazoles PM Cheuka, DG Cabrera, T Paquet, K Chibale Bioorganic & Medicinal Chemistry Letters 24 (22), 5207-5211, 2014 | 8 | 2014 |
| Drug discovery and target identification against schistosomiasis: A reality check on progress and future prospects PM Cheuka Current Topics in Medicinal Chemistry 22 (19), 1595-1610, 2022 | 7 | 2022 |
| Emerging Drug Targets for Antimalarial Drug Discovery: Validation and Insights into Molecular Mechanisms of Function PM Cheuka, P Njaria, G Mayoka, E Funjika Journal of Medicinal Chemistry 67 (2), 838-863, 2024 | 5 | 2024 |
| Medicinal Chemistry and Target Identification of Synthetic Clinical and Advanced Preclinical Antimalarial Candidates (2000-2022) PM Cheuka, D Mambwe, G Mayoka Current Topics in Medicinal Chemistry 23 (3), 227-247, 2023 | 5 | 2023 |
| Phytochemical and pharmacological profiles of the genus Odontonema (Acanthaceae) LP Luhata, NM Munkombwe, PM Cheuka, H Sikanyika British Journal of Pharmaceutical Research 14 (1), 1-7, 2016 | 4 | 2016 |
| Critical Study of Phytochemical and Pharmacological Profiles of the Genus Odontonema (Acanthaceae) LP Luhata, PM Cheuka BP International, 2021 | 2 | 2021 |
| Exploring the transmission-blocking activity of antiplasmodial 3, 6-diarylated imidazopyridazines D Coertzen, J Reader, ME van der Watt, MM Leshabane, H Langeveld, ... Transactions of the Royal Society of South Africa 76 (3), 225-233, 2021 | 1 | 2021 |
| Antimalarial imidazopyridazines and aminopyrazines: synthesis, physicochemical optimization and structure-activity relationships PM Cheuka | 1 | 2018 |
| Synthesis of aminomethylthiazole analogues for evaluation as antiplasmodial agents PM Cheuka | 1 | 2014 |
| Structure activity relationships of antischistosomal N-phenylbenzamides by incorporation of electron-withdrawing functionalities AM Dawoodjee, J Sichinga, H Banda, S Mbaya, E Funjika, G Mayoka, ... Results in Chemistry 12, 101890, 2024 | | 2024 |
