| Late-stage difluoromethylation: concepts, developments and perspective JBI Sap, CF Meyer, NJW Straathof, N Iwumene, CW Am Ende, ... Chemical Society Reviews 50 (14), 8214-8247, 2021 | 264 | 2021 |
| Organophotoredox hydrodefluorination of trifluoromethylarenes with translational applicability to drug discovery JBI Sap, NJW Straathof, T Knauber, CF Meyer, M Médebielle, L Buglioni, ... Journal of the American Chemical Society 142 (20), 9181-9187, 2020 | 160 | 2020 |
| Light-driven post-translational installation of reactive protein side chains B Josephson, C Fehl, PG Isenegger, S Nadal, TH Wright, AWJ Poh, ... Nature 585 (7826), 530-537, 2020 | 141 | 2020 |
| Hydrosulfonylation of alkenes with sulfonyl chlorides under visible light activation SM Hell, CF Meyer, A Misale, JBI Sap, KE Christensen, MC Willis, ... Angewandte Chemie International Edition 59 (28), 11620-11626, 2020 | 124 | 2020 |
| Manual and automated Cu-mediated radiosynthesis of the PARP inhibitor [18F]olaparib F Guibbal, PG Isenegger, TC Wilson, A Pacelli, D Mahaut, JBI Sap, ... Nature protocols 15 (4), 1525-1541, 2020 | 52 | 2020 |
| Hydrofluoromethylation of alkenes with fluoroiodomethane and beyond SM Hell, CF Meyer, S Ortalli, JBI Sap, X Chen, V Gouverneur Chemical Science 12 (36), 12149-12155, 2021 | 47 | 2021 |
| [18F]Difluorocarbene for positron emission tomography JBI Sap, CF Meyer, J Ford, NJW Straathof, AB Dürr, MJ Lelos, SJ Paisey, ... Nature 606 (7912), 102-108, 2022 | 43 | 2022 |
| Synthesis of 18 F-difluoromethylarenes using aryl boronic acids, ethyl bromofluoroacetate and [18 F] fluoride JBI Sap, TC Wilson, CW Kee, NJW Straathof, CW Am Ende, P Mukherjee, ... Chemical Science 10 (11), 3237-3241, 2019 | 41 | 2019 |
| Multi-patient dose synthesis of [18F]Flumazenil via a copper-mediated 18F-fluorination T Gendron, G Destro, NJW Straathof, JBI Sap, F Guibbal, C Vriamont, ... EJNMMI Radiopharmacy and Chemistry 7 (1), 5, 2022 | 11 | 2022 |
| Radiosynthesis of [18F]ArylSCF2H Using Aryl Boronic Acids, S-(Chlorofluoromethyl)benzenesulfonothioate and [18F]Fluoride Q Zhao, PG Isenegger, TC Wilson, JBI Sap, F Guibbal, L Lu, ... CCS Chemistry 3 (7), 1921-1028, 2021 | 9 | 2021 |
| Hydrochlorofluoromethylation of unactivated alkenes with chlorofluoroacetic acid CF Meyer, SM Hell, JBI Sap, A Misale, A Peschiulli, D Oehlrich, ... Tetrahedron 75 (47), 130679, 2019 | 9 | 2019 |
| Light‐Driven Radiochemistry with Fluorine‐18, Carbon‐11 and Zirconium‐89 D Lin, LM Lechermann, MP Huestis, J Marik, JBI Sap Angewandte Chemie International Edition 63 (14), e202317136, 2024 | 6 | 2024 |
| Mechanochemical difluoromethylation of (thio)phenols and N‐heterocycles J Ford, B Hopkin, JBI Sap, V Gouverneur Israel Journal of Chemistry 63 (10-11), e202300109, 2023 | 3 | 2023 |
| Expedient Access to 18F‐Fluoroheteroarenes via Deaminative Radiofluorination of Aniline‐Derived Pyridinium Salts J Ford, S Ortalli, Z Chen, JBI Sap, M Tredwell, V Gouverneur Angewandte Chemie, e202404945, 2024 | 1 | 2024 |
| Isostere 18F-protein post-translational editing enables dynamic tracking of neurodegeneration biomarkers N Yang, AWJ Poh, AM Giltrap, PG Isenegger, JBI Sap, J Ford, ... bioRxiv, 2025.01. 26.634877, 2025 | | 2025 |
| DIFLUOROCARBENE RADIOSYNTHESIS VEBM Gouverneur, CF Meyer, JBI Sap US Patent App. 18/694,241, 2024 | | 2024 |
| The evaluation of enzyme-mediated forms of [18F] AlF-RESCA-VHH5v2 exemplified with human CD8 PET imaging H Gill, S Sriraman, A Ogasawara, J Sap, J Tinianow, S Lim, P Holder, ... Nuclear Medicine and Biology 126, 108706, 2023 | | 2023 |
| Photoredox protein modification PG Isenegger, BG Davis, B Josephson, V Gouverneur, C Fehl, AWJ Poh, ... US Patent App. 18/005,519, 2023 | | 2023 |
| Multi-patient dose synthesis of [18F] Flumazenil via a copper-mediated 18F-fluorination G Thibault, D Gianluca, SN JW, JB Sap, G Florian, C Vriamont, C Caygill, ... EJNMMI Radiopharmacy and Chemistry 7 (1), 2022 | | 2022 |
| New late-stage strategies towards difluoromethylarenes JBI Sap University of Oxford, 2020 | | 2020 |