| General enantioselective C− H activation with efficiently tunable cyclopentadienyl ligands ZJ Jia, C Merten, R Gontla, CG Daniliuc, AP Antonchick, H Waldmann Angewandte Chemie International Edition 56 (9), 2429-2434, 2017 | 295 | 2017 |
| Enantioselective Formal C(sp3)−H Bond Activation in the Synthesis of Bioactive Spiropyrazolone Derivatives H Li, R Gontla, J Flegel, C Merten, S Ziegler, AP Antonchick, H Waldmann Angewandte Chemie International Edition 58 (1), 307-311, 2019 | 121 | 2019 |
| Covalent‐allosteric kinase inhibitors J Weisner, R Gontla, L van der Westhuizen, S Oeck, J Ketzer, P Janning, ... Angewandte Chemie International Edition 54 (35), 10313-10316, 2015 | 114 | 2015 |
| Preclinical Efficacy of Covalent-Allosteric AKT Inhibitor Borussertib in Combination with Trametinib in KRAS-Mutant Pancreatic and Colorectal Cancer J Weisner, I Landel, C Reintjes, N Uhlenbrock, M Trajkovic-Arsic, ... Cancer research 79 (9), 2367-2378, 2019 | 89 | 2019 |
| Structural and chemical insights into the covalent-allosteric inhibition of the protein kinase Akt N Uhlenbrock, S Smith, J Weisner, I Landel, M Lindemann, TA Le, ... Chemical Science 10 (12), 3573-3585, 2019 | 59 | 2019 |
| B (C6F5) 3: an efficient catalyst for reductive alkylation of alkoxy benzenes and for synthesis of triarylmethanes using aldehydes S Chandrasekhar, S Khatun, G Rajesh, CR Reddy Tetrahedron Letters 50 (48), 6693-6697, 2009 | 36 | 2009 |
| Tris (pentafluorophenyl) borane: a mild and efficient catalyst for the chemoselective tritylation of alcohols CR Reddy, G Rajesh, SV Balaji, N Chethan Tetrahedron Letters 49 (6), 970-973, 2008 | 34 | 2008 |
| Palladium-catalyzed [4+ 2] annulation of aryl and alkenyl carboxamides with 1, 3-dienes via C–H functionalization: synthesis of 3, 4-dihydroisoquinolones and 5, 6 … M Sun, J Li, W Chen, H Wu, J Yang, Z Wang Synthesis 52 (08), 1253-1265, 2020 | 25 | 2020 |
| First total synthesis of achaetolide S Chandrasekhar, SV Balaji, G Rajesh Tetrahedron Letters 51 (39), 5164-5166, 2010 | 20 | 2010 |
| Enantioselective synthesis of the C5–C23 segment of biselyngbyaside S Chandrasekhar, G Rajesh, T Naresh Tetrahedron Letters 54 (3), 252-255, 2013 | 19 | 2013 |
| Kovalent‐allosterische Kinase‐Inhibitoren J Weisner, R Gontla, L van der Westhuizen, S Oeck, J Ketzer, P Janning, ... Angewandte Chemie 127 (35), 10452-10456, 2015 | 12 | 2015 |
| Avapritinib-based SAR studies unveil a binding pocket in KIT and PDGFRA A Teuber, T Schulz, BS Fletcher, R Gontla, T Mühlenberg, ML Zischinsky, ... Nature Communications 15 (1), 63, 2024 | 11 | 2024 |
| Variability of Rhodium (III)-Catalyzed Reactions of Aromatic Oximes with Alkenes EA Trifonova, AA Komarova, D Chusov, DS Perekalin Synlett 31 (11), 1117-1120, 2020 | 11 | 2020 |
| van der Westhuizen l, Oeck S, Ketzer J, Janning P, Richters A, Mühlenberg T, Fang z, Taher A, et al: Covalent‑allosteric kinase inhibitors J Weisner, R Gontla Angew Chem Int ed engl 54, 10313-10316, 2015 | 6 | 2015 |
| Correction: A high-throughput effector screen identifies a novel small molecule scaffold for inhibition of ten-eleven translocation dioxygenase 2 S Palei, J Weisner, M Vogt, R Gontla, B Buchmuller, C Ehrt, T Grabe, ... RSC Medicinal Chemistry 15 (2), 753-754, 2024 | 1 | 2024 |
| A high-throughput effector screen identifies a novel small molecule scaffold for inhibition of ten-eleven translocation dioxygenase 2 S Palei, J Weisner, M Vogt, R Gontla, B Buchmuller, C Ehrt, T Grabe, ... RSC Medicinal Chemistry 13 (12), 1540-1548, 2022 | 1 | 2022 |
| Design, Synthesis, and SAR of Covalent KIT and PDGFRA Inhibitors─ Exploring Their Potential in Targeting GIST T Schulz, R Gontla, A Teuber, M Beerbaum, BS Fletcher, T Mühlenberg, ... Journal of medicinal chemistry, 2025 | | 2025 |
| Kinase inhibitors and their use in cancer therapy D Rauh, R Gontla, J Weisner US Patent 10,550,114, 2020 | | 2020 |
