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Grégory Upert
Grégory Upert
Bright Peak Therapeutics
Email verificata su brightpeaktx.com
Titolo
Citata da
Citata da
Anno
Chimeric peptidomimetic antibiotics against Gram-negative bacteria
A Luther, M Urfer, M Zahn, M Müller, SY Wang, M Mondal, A Vitale, ...
Nature 576 (7787), 452-458, 2019
2962019
Enamine catalysis with low catalyst loadings-high efficiency via kinetic studies
M Wiesner, G Upert, G Angelici, H Wennemers
Journal of the American Chemical Society 132 (1), 6-7, 2010
2182010
Emerging peptide antibiotics with therapeutic potential
G Upert, A Luther, D Obrecht, P Ermert
Medicine in drug discovery 9, 100078, 2021
722021
Peptidomic comparison and characterization of the major components of the venom of the giant ant Dinoponera quadriceps collected in four different areas of Brazil
CT Cologna, J dos Santos Cardoso, E Jourdan, M Degueldre, G Upert, ...
Journal of proteomics 94, 413-422, 2013
722013
Oligoprolines as scaffolds for the formation of silver nanoparticles in defined sizes: correlating molecular and nanoscopic dimensions
G Upert, F Bouillère, H Wennemers
Angewandte Chemie 17 (124), 4307-4310, 2012
692012
RgIA4 potently blocks mouse α9α10 nAChRs and provides long lasting protection against oxaliplatin-induced cold allodynia
SB Christensen, AJ Hone, I Roux, J Kniazeff, JP Pin, G Upert, D Servent, ...
Frontiers in cellular neuroscience 11, 219, 2017
682017
Silver nanoparticle formation in different sizes induced by peptides identified within split‐and‐mix libraries
K Belser, T Vig Slenters, C Pfumbidzai, G Upert, L Mirolo, KM Fromm, ...
Angewandte Chemie International Edition 48 (20), 3661-3664, 2009
682009
Antibiotic polymyxin arranges lipopolysaccharide into crystalline structures to solidify the bacterial membrane
S Manioglu, SM Modaresi, N Ritzmann, J Thoma, SA Overall, A Harms, ...
Nature communications 13 (1), 6195, 2022
662022
Identification, structural and pharmacological characterization of τ-CnVA, a conopeptide that selectively interacts with somatostatin sst3 receptor
C Petrel, HG Hocking, M Reynaud, G Upert, P Favreau, D Biass, ...
Biochemical pharmacology 85 (11), 1663-1671, 2013
512013
Zinc-selective inhibition of the promiscuous bacterial amide-hydrolase DapE: implications of metal heterogeneity for evolution and antibiotic drug design
NR Uda, G Upert, G Angelici, S Nicolet, T Schmidt, T Schwede, M Creus
Metallomics 6 (1), 88-95, 2014
312014
An efficient biodelivery system for antisense polyamide nucleic acid (PNA)
M Mehiri, G Upert, S Tripathi, A Di Giorgio, R Condom, VN Pandey, ...
Oligonucleotides 18 (3), 245-256, 2008
252008
Ancestral protein resurrection and engineering opportunities of the mamba aminergic toxins
G Blanchet, D Alili, A Protte, G Upert, N Gilles, L Tepshi, EA Stura, ...
Scientific Reports 7 (1), 2701, 2017
232017
New α-adrenergic property for synthetic MTβ and CM-3 three-finger fold toxins from black mamba
G Blanchet, G Upert, G Mourier, B Gilquin, N Gilles, D Servent
Toxicon 75, 160-167, 2013
232013
Combined use of ion mobility and collision-induced dissociation to investigate the opening of disulfide bridges by electron-transfer dissociation in peptides bearing two …
P Massonnet, G Upert, N Smargiasso, N Gilles, L Quinton, E De Pauw
Analytical chemistry 87 (10), 5240-5246, 2015
222015
Peptidomimetic antibiotics disrupt the lipopolysaccharide transport bridge of drug-resistant Enterobacteriaceae
M Schuster, E Brabet, KK Oi, N Desjonquères, K Moehle, K Le Poupon, ...
Science Advances 9 (21), eadg3683, 2023
202023
A venomics approach coupled to high-throughput toxin production strategies identifies the first venom-derived melanocortin receptor agonists
S Reynaud, J Ciolek, M Degueldre, NJ Saez, AF Sequeira, Y Duhoo, ...
Journal of medicinal chemistry 63 (15), 8250-8264, 2020
202020
Ion mobility-mass spectrometry as a tool for the structural characterization of peptides bearing intramolecular disulfide bond (s)
P Massonnet, JRN Haler, G Upert, M Degueldre, D Morsa, N Smargiasso, ...
Journal of The American Society for Mass Spectrometry 27 (10), 1637-1646, 2016
182016
Thieme chemistry journals awardees–where are they now? A stereoselective tripeptide catalyst for conjugate addition reactions of acetophenones to dicyanoolefins
T Schnitzer, H Wennemers
Synlett 28 (11), 1282-1286, 2017
172017
Effect of γ-substituted proline derivatives on the performance of the peptidic catalyst H-dPro-pro-Glu-NH2
T Schnitzer, H Wennemers
Synthesis 50 (22), 4377-4382, 2018
162018
A new Kunitz‐type snake toxin family associated with an original mode of interaction with the vasopressin 2 receptor
L Droctové, J Ciolek, C Mendre, A Chorfa, P Huerta, C Carvalho, C Gouin, ...
British Journal of Pharmacology 179 (13), 3470-3481, 2022
152022
Il sistema al momento non può eseguire l'operazione. Riprova più tardi.
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