Chimeric peptidomimetic antibiotics against Gram-negative bacteria A Luther, M Urfer, M Zahn, M Müller, SY Wang, M Mondal, A Vitale, ... Nature 576 (7787), 452-458, 2019 | 296 | 2019 |
Enamine catalysis with low catalyst loadings-high efficiency via kinetic studies M Wiesner, G Upert, G Angelici, H Wennemers Journal of the American Chemical Society 132 (1), 6-7, 2010 | 218 | 2010 |
Emerging peptide antibiotics with therapeutic potential G Upert, A Luther, D Obrecht, P Ermert Medicine in drug discovery 9, 100078, 2021 | 72 | 2021 |
Peptidomic comparison and characterization of the major components of the venom of the giant ant Dinoponera quadriceps collected in four different areas of Brazil CT Cologna, J dos Santos Cardoso, E Jourdan, M Degueldre, G Upert, ... Journal of proteomics 94, 413-422, 2013 | 72 | 2013 |
Oligoprolines as scaffolds for the formation of silver nanoparticles in defined sizes: correlating molecular and nanoscopic dimensions G Upert, F Bouillère, H Wennemers Angewandte Chemie 17 (124), 4307-4310, 2012 | 69 | 2012 |
RgIA4 potently blocks mouse α9α10 nAChRs and provides long lasting protection against oxaliplatin-induced cold allodynia SB Christensen, AJ Hone, I Roux, J Kniazeff, JP Pin, G Upert, D Servent, ... Frontiers in cellular neuroscience 11, 219, 2017 | 68 | 2017 |
Silver nanoparticle formation in different sizes induced by peptides identified within split‐and‐mix libraries K Belser, T Vig Slenters, C Pfumbidzai, G Upert, L Mirolo, KM Fromm, ... Angewandte Chemie International Edition 48 (20), 3661-3664, 2009 | 68 | 2009 |
Antibiotic polymyxin arranges lipopolysaccharide into crystalline structures to solidify the bacterial membrane S Manioglu, SM Modaresi, N Ritzmann, J Thoma, SA Overall, A Harms, ... Nature communications 13 (1), 6195, 2022 | 66 | 2022 |
Identification, structural and pharmacological characterization of τ-CnVA, a conopeptide that selectively interacts with somatostatin sst3 receptor C Petrel, HG Hocking, M Reynaud, G Upert, P Favreau, D Biass, ... Biochemical pharmacology 85 (11), 1663-1671, 2013 | 51 | 2013 |
Zinc-selective inhibition of the promiscuous bacterial amide-hydrolase DapE: implications of metal heterogeneity for evolution and antibiotic drug design NR Uda, G Upert, G Angelici, S Nicolet, T Schmidt, T Schwede, M Creus Metallomics 6 (1), 88-95, 2014 | 31 | 2014 |
An efficient biodelivery system for antisense polyamide nucleic acid (PNA) M Mehiri, G Upert, S Tripathi, A Di Giorgio, R Condom, VN Pandey, ... Oligonucleotides 18 (3), 245-256, 2008 | 25 | 2008 |
Ancestral protein resurrection and engineering opportunities of the mamba aminergic toxins G Blanchet, D Alili, A Protte, G Upert, N Gilles, L Tepshi, EA Stura, ... Scientific Reports 7 (1), 2701, 2017 | 23 | 2017 |
New α-adrenergic property for synthetic MTβ and CM-3 three-finger fold toxins from black mamba G Blanchet, G Upert, G Mourier, B Gilquin, N Gilles, D Servent Toxicon 75, 160-167, 2013 | 23 | 2013 |
Combined use of ion mobility and collision-induced dissociation to investigate the opening of disulfide bridges by electron-transfer dissociation in peptides bearing two … P Massonnet, G Upert, N Smargiasso, N Gilles, L Quinton, E De Pauw Analytical chemistry 87 (10), 5240-5246, 2015 | 22 | 2015 |
Peptidomimetic antibiotics disrupt the lipopolysaccharide transport bridge of drug-resistant Enterobacteriaceae M Schuster, E Brabet, KK Oi, N Desjonquères, K Moehle, K Le Poupon, ... Science Advances 9 (21), eadg3683, 2023 | 20 | 2023 |
A venomics approach coupled to high-throughput toxin production strategies identifies the first venom-derived melanocortin receptor agonists S Reynaud, J Ciolek, M Degueldre, NJ Saez, AF Sequeira, Y Duhoo, ... Journal of medicinal chemistry 63 (15), 8250-8264, 2020 | 20 | 2020 |
Ion mobility-mass spectrometry as a tool for the structural characterization of peptides bearing intramolecular disulfide bond (s) P Massonnet, JRN Haler, G Upert, M Degueldre, D Morsa, N Smargiasso, ... Journal of The American Society for Mass Spectrometry 27 (10), 1637-1646, 2016 | 18 | 2016 |
Thieme chemistry journals awardees–where are they now? A stereoselective tripeptide catalyst for conjugate addition reactions of acetophenones to dicyanoolefins T Schnitzer, H Wennemers Synlett 28 (11), 1282-1286, 2017 | 17 | 2017 |
Effect of γ-substituted proline derivatives on the performance of the peptidic catalyst H-dPro-pro-Glu-NH2 T Schnitzer, H Wennemers Synthesis 50 (22), 4377-4382, 2018 | 16 | 2018 |
A new Kunitz‐type snake toxin family associated with an original mode of interaction with the vasopressin 2 receptor L Droctové, J Ciolek, C Mendre, A Chorfa, P Huerta, C Carvalho, C Gouin, ... British Journal of Pharmacology 179 (13), 3470-3481, 2022 | 15 | 2022 |