| A cyclic peptide inhibitor of HIF-1 heterodimerization that inhibits hypoxia signaling in cancer cells E Miranda, IK Nordgren, AL Male, CE Lawrence, F Hoakwie, F Cuda, ... Journal of the American Chemical Society 135 (28), 10418-10425, 2013 | 228* | 2013 |
| Biocompatible artificial DNA linker that is read through by DNA polymerases and is functional in Escherichia coli AH El-Sagheer, AP Sanzone, R Gao, A Tavassoli, T Brown Proceedings of the National Academy of Sciences 108 (28), 11338-11343, 2011 | 219 | 2011 |
| Split-intein mediated circular ligation used in the synthesis of cyclic peptide libraries in E. coli A Tavassoli, SJ Benkovic Nature protocols 2 (5), 1126-1133, 2007 | 214 | 2007 |
| Inhibition of HIV Budding by a Genetically Selected Cyclic Peptide Targeting the Gag− TSG101 Interaction A Tavassoli, Q Lu, J Gam, H Pan, SJ Benkovic, SN Cohen ACS chemical biology 3 (12), 757-764, 2008 | 200 | 2008 |
| Methods for generating and screening libraries of genetically encoded cyclic peptides in drug discovery C Sohrabi, A Foster, A Tavassoli Nature Reviews Chemistry 4 (2), 90-101, 2020 | 191 | 2020 |
| Identification of borinic esters as inhibitors of bacterial cell growth and bacterial methyltransferases, CcrM and MenH SJ Benkovic, SJ Baker, MRK Alley, YH Woo, YK Zhang, T Akama, W Mao, ... Journal of medicinal chemistry 48 (23), 7468-7476, 2005 | 174 | 2005 |
| A lanthipeptide library used to identify a protein–protein interaction inhibitor X Yang, KR Lennard, C He, MC Walker, AT Ball, C Doigneaux, ... Nature Chemical Biology 14 (4), 375-380, 2018 | 156 | 2018 |
| SICLOPPS cyclic peptide libraries in drug discovery A Tavassoli Current Opinion in Chemical Biology 38, 30-35, 2017 | 149 | 2017 |
| Genetically selected cyclic‐peptide inhibitors of AICAR transformylase homodimerization A Tavassoli, SJ Benkovic Angewandte Chemie International Edition 44 (18), 2760-2763, 2005 | 132 | 2005 |
| Targeting Tumour Proliferation with a Small‐Molecule Inhibitor of AICAR Transformylase Homodimerization IB Spurr, CN Birts, F Cuda, SJ Benkovic, JP Blaydes, A Tavassoli ChemBioChem 13 (11), 1628-1634, 2012 | 117 | 2012 |
| Transcription of Click‐Linked DNA in Human Cells CN Birts, AP Sanzone, AH El‐Sagheer, JP Blaydes, T Brown, A Tavassoli Angewandte Chemie International Edition 53 (9), 2362-2365, 2014 | 103 | 2014 |
| Targeting tumour angiogenesis with small molecule inhibitors of hypoxia inducible factor IK Nordgren, A Tavassoli Chemical Society Reviews 40 (8), 4307-4317, 2011 | 99 | 2011 |
| A cyclic peptide inhibitor of C-terminal binding protein dimerization links metabolism with mitotic fidelity in breast cancer cells CN Birts, SK Nijjar, CA Mardle, F Hoakwie, PJ Duriez, JP Blaydes, ... Chemical Science 4 (8), 3046-3057, 2013 | 97 | 2013 |
| Assembly of a biocompatible triazole-linked gene by one-pot click-DNA ligation NM Kukwikila, N Gale, AH El-Sagheer, T Brown, A Tavassoli Nature Chemistry, 2017 | 96 | 2017 |
| AMPK Activation via Modulation of De Novo Purine Biosynthesis with an Inhibitor of ATIC Homodimerization DJ Asby, F Cuda, M Beyaert, FD Houghton, FR Cagampang, A Tavassoli Chemistry & biology 22 (7), 838-848, 2015 | 96 | 2015 |
| Peptides Come Round: Using SICLOPPS Libraries for Early Stage Drug Discovery KR Lennard, A Tavassoli Chemistry-A European Journal 20 (34), 10608-10614, 2014 | 87 | 2014 |
| Influenza A/Hong Kong/156/1997 (H5N1) virus NS1 gene mutations F103L and M106I both increase IFN antagonism, virulence and cytoplasmic localization but differ in binding to RIG … SK Dankar, E Miranda, NE Forbes, M Pelchat, A Tavassoli, M Selman, ... Virology journal 10 (1), 243, 2013 | 63 | 2013 |
| Fluorescent transmembrane anion transporters: shedding light on anionophoric activity in cells SN Berry, V Soto-Cerrato, ENW Howe, HJ Clarke, I Mistry, A Tavassoli, ... Chemical Science 7 (8), 5069-5077, 2016 | 60 | 2016 |
| Rational design, synthesis, evaluation, and crystal structure of a potent inhibitor of human GAR Tfase: 10-(trifluoroacetyl)-5, 10-dideazaacyclic-5, 6, 7, 8-tetrahydrofolic acid Y Zhang, J Desharnais, TH Marsilje, C Li, MP Hedrick, LT Gooljarsingh, ... Biochemistry 42 (20), 6043-6056, 2003 | 60 | 2003 |
| Assessing the biocompatibility of click-linked DNA in Escherichia coli AP Sanzone, AH El-Sagheer, T Brown, A Tavassoli Nucleic acids research 40 (20), 10567-10575, 2012 | 59 | 2012 |
