Recent advances in the medicinal chemistry of aurones R Haudecoeur, A Boumendjel Current medicinal chemistry 19 (18), 2861-2875, 2012 | 150 | 2012 |
Discovery of naturally occurring aurones that are potent allosteric inhibitors of hepatitis C virus RNA-dependent RNA polymerase R Haudecoeur, A Ahmed-Belkacem, W Yi, A Fortuné, R Brillet, C Belle, ... Journal of medicinal chemistry 54 (15), 5395-5402, 2011 | 138 | 2011 |
Advances in the design of genuine human tyrosinase inhibitors for targeting melanogenesis and related pigmentations B Roulier, B Pérès, R Haudecoeur Journal of medicinal chemistry 63 (22), 13428-13443, 2020 | 103 | 2020 |
A model of smart G-quadruplex ligand R Haudecoeur, L Stefan, F Denat, D Monchaud Journal of the American Chemical Society 135 (2), 550-553, 2013 | 99 | 2013 |
Occurrences, biosynthesis and properties of aurones as high-end evolutionary products B Boucherle, M Peuchmaur, A Boumendjel, R Haudecoeur Phytochemistry 142, 92-111, 2017 | 95 | 2017 |
Refinement of arylthiosemicarbazone pharmacophore in inhibition of mushroom tyrosinase W Yi, C Dubois, S Yahiaoui, R Haudecoeur, C Belle, H Song, R Hardré, ... European journal of medicinal chemistry 46 (9), 4330-4335, 2011 | 81 | 2011 |
Traditional uses, phytochemistry and pharmacological properties of African Nauclea species: A review R Haudecoeur, M Peuchmaur, B Pérès, M Rome, GS Taïwe, ... Journal of Ethnopharmacology 212, 106-136, 2018 | 76 | 2018 |
Are human tyrosinase and related proteins suitable targets for melanoma therapy? E Buitrago, R Hardre, R Haudecoeur, H Jamet, C Belle, A Boumendjel, ... Current topics in medicinal chemistry 16 (27), 3033-3047, 2016 | 73 | 2016 |
Occurrence of the synthetic analgesic tramadol in an African medicinal plant. A Boumendjel, G Sotoing Taïwe, E Ngo Bum, T Chabrol, C Beney, ... Angewandte Chemie International Edition 52 (45), 2013 | 73 | 2013 |
Aurone derivatives as promising antibacterial agents against resistant Gram-positive pathogens H Olleik, S Yahiaoui, B Roulier, E Courvoisier-Dezord, J Perrier, B Pérès, ... European journal of medicinal chemistry 165, 133-141, 2019 | 67 | 2019 |
Nauclea latifolia: biological activity and alkaloid phytochemistry of a West African tree B Boucherle, R Haudecoeur, EF Queiroz, M De Waard, JL Wolfender, ... Natural product reports 33 (9), 1034-1043, 2016 | 67 | 2016 |
β-Carboline as a privileged scaffold for multitarget strategies in Alzheimer’s disease therapy A Beato, A Gori, B Boucherle, M Peuchmaur, R Haudecoeur Journal of Medicinal Chemistry 64 (3), 1392-1422, 2021 | 66 | 2021 |
Structure–activity relationships in the development of allosteric hepatitis c virus rna‐dependent rna polymerase inhibitors: ten years of research R Haudecoeur, M Peuchmaur, A Ahmed‐Belkacem, JM Pawlotsky, ... Medicinal research reviews 33 (5), 934-984, 2013 | 59 | 2013 |
2-Hydroxypyridine-N-oxide-Embedded Aurones as Potent Human Tyrosinase Inhibitors R Haudecoeur, M Carotti, A Gouron, M Maresca, E Buitrago, R Hardré, ... ACS medicinal chemistry letters 8 (1), 55-60, 2017 | 57 | 2017 |
B-ring modified aurones as promising allosteric inhibitors of hepatitis C virus RNA-dependent RNA polymerase A Meguellati, A Ahmed-Belkacem, W Yi, R Haudecoeur, M Crouillère, ... European journal of medicinal chemistry 80, 579-592, 2014 | 54 | 2014 |
Versatile effects of aurone structure on mushroom tyrosinase activity C Dubois, R Haudecoeur, M Orio, C Belle, C Bochot, A Boumendjel, ... ChemBioChem 13 (4), 559-565, 2012 | 48 | 2012 |
Investigation of binding‐site homology between mushroom and bacterial Tyrosinases by using Aurones as effectors R Haudecoeur, A Gouron, C Dubois, H Jamet, M Lightbody, R Hardré, ... ChemBioChem 15 (9), 1325-1333, 2014 | 47 | 2014 |
Porphyrin-templated synthetic G-quartet (PorphySQ): a second prototype of G-quartet-based G-quadruplex ligand HJ Xu, L Stefan, R Haudecoeur, S Vuong, P Richard, F Denat, JM Barbe, ... Organic & Biomolecular Chemistry 10 (27), 5212-5218, 2012 | 37 | 2012 |
Recombinant Tyrosinase from Polyporus arcularius: Overproduction in Escherichia coli, Characterization, and Use in a Study of Aurones as Tyrosinase Effectors E Marková, M Kotik, A Křenková, P Man, R Haudecoeur, A Boumendjel, ... Journal of Agricultural and Food Chemistry 64 (14), 2925-2931, 2016 | 36 | 2016 |
Glycosyl‐Substituted Dicarboxylates as Detergents for the Extraction, Overstabilization, and Crystallization of Membrane Proteins KA Nguyen, M Peuchmaur, S Magnard, R Haudecoeur, C Boyère, ... Angewandte Chemie International Edition 57 (11), 2948-2952, 2018 | 34 | 2018 |