| Homologation chemistry with nucleophilic α-substituted organometallic reagents: chemocontrol, new concepts and (solved) challenges L Castoldi, S Monticelli, R Senatore, L Ielo, V Pace Chemical Communications 54 (50), 6692-6704, 2018 | 81 | 2018 |
| Exploiting the 1-(4-fluorobenzyl) piperazine fragment for the development of novel tyrosinase inhibitors as anti-melanogenic agents: Design, synthesis, structural insights and … L Ielo, B Deri, MP Germano, S Vittorio, S Mirabile, R Gitto, A Rapisarda, ... European journal of medicinal chemistry 178, 380-389, 2019 | 74 | 2019 |
| Telescoped, Divergent, Chemoselective C1 and C1‐C1 Homologation of Imine Surrogates: Access to Quaternary Chloro‐and Halomethyl‐Trifluoromethyl Aziridines L Ielo, S Touqeer, A Roller, T Langer, W Holzer, V Pace Angewandte Chemie 131 (8), 2501-2506, 2019 | 71 | 2019 |
| Weinreb amides as privileged acylating agents for accessing α-substituted ketones R Senatore, L Ielo, S Monticelli, L Castoldi, V Pace Synthesis 51 (14), 2792-2808, 2019 | 54 | 2019 |
| Expeditious and chemoselective synthesis of α-aryl and α-alkyl selenomethylketones via homologation chemistry R Senatore, L Castoldi, L Ielo, W Holzer, V Pace Organic Letters 20 (9), 2685-2688, 2018 | 52 | 2018 |
| Targeting tyrosinase: development and structural insights of novel inhibitors bearing arylpiperidine and arylpiperazine fragments S Ferro, B Deri, MP Germanò, R Gitto, L Ielo, MR Buemi, G Certo, ... Journal of medicinal chemistry 61 (9), 3908-3917, 2018 | 48 | 2018 |
| Chemical exploration of 4-(4-fluorobenzyl) piperidine fragment for the development of new tyrosinase inhibitors S Ferro, L De Luca, MP Germanò, MR Buemi, L Ielo, G Certo, M Kanteev, ... European journal of medicinal chemistry 125, 992-1001, 2017 | 47 | 2017 |
| Recent advances in the accessibility, synthetic utility, and biological applications of aziridines C Dank, L Ielo Organic & Biomolecular Chemistry 21 (22), 4553-4573, 2023 | 44 | 2023 |
| Chemoselective Homologation–Deoxygenation Strategy Enabling the Direct Conversion of Carbonyls into (n+1)-Halomethyl-Alkanes M Miele, A Citarella, T Langer, E Urban, M Zehl, W Holzer, L Ielo, V Pace Organic Letters 22 (19), 7629-7634, 2020 | 37 | 2020 |
| Merging lithium carbenoid homologation and enzymatic reduction: A combinative approach to the HIV-protease inhibitor nelfinavir L Castoldi, L Ielo, P Hoyos, MJ Hernáiz, L De Luca, AR Alcántara, ... Tetrahedron 74 (18), 2211-2217, 2018 | 33 | 2018 |
| The synthetic versatility of the Tiffeneau–Demjanov chemistry in homologation tactics SM Kohlbacher, VS Ionasz, L Ielo, V Pace Monatshefte für Chemie-Chemical Monthly 150, 2011-2019, 2019 | 26 | 2019 |
| Heterocyclic compounds as synthetic tyrosinase inhibitors: recent advances S Vittorio, C Dank, L Ielo International journal of molecular sciences 24 (10), 9097, 2023 | 23 | 2023 |
| Direct Access to 9-Chloro-1H-benzo[b]furo[3,4-e]azepin-1-ones via Palladium(II)-Catalyzed Intramolecular syn-Oxypalladation/Olefin Insertion/sp2-C–H Bond … M Karuppasamy, BS Vachan, P Vinoth, I Muthukrishnan, S Nagarajan, ... Organic Letters 21 (15), 5784-5788, 2019 | 23 | 2019 |
| Halogen‐Imparted Reactivity in Lithium Carbenoid Mediated Homologations of Imine Surrogates: Direct Assembly of bis‐Trifluoromethyl‐β‐Diketiminates and the Dual Role of LiCH2I L Ielo, L Castoldi, S Touqeer, J Lombino, A Roller, C Prandi, W Holzer, ... Angewandte Chemie 132 (47), 21038-21043, 2020 | 22 | 2020 |
| Substituted α‐Sulfur Methyl Carbanions: Effective Homologating Agents for the Chemoselective Preparation of β‐Oxo Thioethers from Weinreb Amides R Senatore, L Ielo, E Urban, W Holzer, V Pace European Journal of Organic Chemistry 2018 (20-21), 2466-2470, 2018 | 22 | 2018 |
| A Combination of pharmacophore and docking‐based virtual screening to discover new tyrosinase inhibitors S Vittorio, T Seidel, MP Germanò, R Gitto, L Ielo, A Garon, A Rapisarda, ... Molecular Informatics 39 (3), 1900054, 2020 | 21 | 2020 |
| Straightforward chemoselective access to unsymmetrical dithioacetals through a thiosulfonate homologation-nucleophilic substitution sequence L Ielo, V Pillari, N Gajic, W Holzer, V Pace Chemical Communications 56 (82), 12395-12398, 2020 | 21 | 2020 |
| 4‐Fluorobenzylpiperazine‐containing derivatives as efficient inhibitors of mushroom tyrosinase S Vittorio, L Ielo, S Mirabile, R Gitto, A Fais, S Floris, A Rapisarda, ... ChemMedChem 15 (18), 1757-1764, 2020 | 19 | 2020 |
| Inhibition of HIV-1 RT activity by a new series of 3-(1, 3, 4-thiadiazol-2-yl) thiazolidin-4-one derivatives MR Buemi, R Gitto, L Ielo, C Pannecouque, L De Luca Bioorganic & Medicinal Chemistry 28 (8), 115431, 2020 | 19 | 2020 |
| Carbenoid-Mediated Homologation Tactics for Assembling (Fluorinated) Epoxides and Aziridines L Ielo, V Pillari, M Miele, D Castiglione, V Pace Synlett 32 (06), 551-560, 2021 | 18 | 2021 |
