| Discovery and preclinical characterization of [18F] PI-2620, a next-generation tau PET tracer for the assessment of tau pathology in Alzheimer’s disease and other tauopathies H Kroth, F Oden, J Molette, H Schieferstein, F Capotosti, A Mueller, ... European journal of nuclear medicine and molecular imaging 46 (10), 2178-2189, 2019 | 188 | 2019 |
| Radiolabeling of nanoparticles and polymers for PET imaging K Stockhofe, JM Postema, H Schieferstein, TL Ross Pharmaceuticals 7 (4), 392-418, 2014 | 175 | 2014 |
| 18F-labeling using click cycloadditions K Kettenbach, H Schieferstein, TL Ross BioMed research international 2014, 2014 | 61 | 2014 |
| A Simple, Rapid Method for the Preparation of [11C]Formaldehyde JM Hooker, M Schönberger, H Schieferstein, JS Fowler Angewandte Chemie International Edition 47 (32), 5989-5992, 2008 | 58 | 2008 |
| Considerations for Human ADME strategy and design paradigm shift (s)‐an Industry white paper GC Young, DK Spracklin, AD James, MG Hvenegaard, G Scarfe, ... Clinical Pharmacology & Therapeutics, 2022 | 23 | 2022 |
| 18 F-click labeling and preclinical evaluation of a new 18 F-folate for PET imaging H Schieferstein, T Betzel, CR Fischer, TL Ross EJNMMI research 3 (1), 1-10, 2013 | 20 | 2013 |
| PI-2620 Lead Optimization Highlights the Importance of Off-Target Assays to Develop a PET Tracer for the Detection of Pathological Aggregated Tau in Alzheimer’s … H Kroth, F Oden, J Molette, H Schieferstein, E Gabellieri, A Mueller, ... Journal of Medicinal Chemistry 64 (17), 12808-12830, 2021 | 19 | 2021 |
| Selective binding to monoamine oxidase A: In vitro and in vivo evaluation of 18F-labeled β-carboline derivatives H Schieferstein, M Piel, F Beyerlein, H Lüddens, N Bausbacher, ... Bioorganic & Medicinal Chemistry 23 (3), 612-623, 2015 | 18 | 2015 |
| 18F‐labeled folic acid derivatives for imaging of the folate receptor via positron emission tomography H Schieferstein, TL Ross Journal of Labelled Compounds and Radiopharmaceuticals 56 (9-10), 432-440, 2013 | 17 | 2013 |
| Characterization of the novel PET Tracer PI-2620 for the assessment of Tau pathology in Alzheimer’s disease and other tauopathies A Mueller, H Kroth, M Berndt, F Capotosti, J Molette, H Schieferstein, ... Journal of Nuclear Medicine 58 (supplement 1), 847-847, 2017 | 16 | 2017 |
| 18F‐Radiolabeling, Preliminary Evaluation of Folate‐pHPMA Conjugates via PET H Schieferstein, A Kelsch, A Reibel, K Koynov, M Barz, HG Buchholz, ... Macromolecular bioscience 14 (10), 1396-1405, 2014 | 16 | 2014 |
| Comparison Study of Two Differently Clicked 18F-Folates—Lipophilicity Plays a Key Role K Kettenbach, LM Reffert, H Schieferstein, S Pektor, R Eckert, M Miederer, ... Pharmaceuticals 11 (1), 30, 2018 | 15 | 2018 |
| Eine einfache und schnelle Methode zur Herstellung von [11C] Formaldehyd JM Hooker, M Schönberger, H Schieferstein, JS Fowler Angewandte Chemie 120 (32), 6078-6081, 2008 | 12 | 2008 |
| Identification of M4205─ A Highly Selective Inhibitor of KIT Mutations for Treatment of Unresectable Metastatic or Recurrent Gastrointestinal Stromal Tumors A Blum, D Dorsch, N Linde, S Brandstetter, HP Buchstaller, M Busch, ... Journal of Medicinal Chemistry, 2023 | 11 | 2023 |
| Synthesis and evaluation of boron folates for Boron-Neutron-Capture-Therapy (BNCT) K Kettenbach, H Schieferstein, C Grunewald, D Iffland, LM Reffert, ... Radiochimica Acta 103 (11), 799-809, 2015 | 10 | 2015 |
| A Polar 18F‐Labeled Amino Acid Derivative for Click Labeling of Biomolecules H Schieferstein, TL Ross European Journal of Organic Chemistry 2014 (17), 3546-3550, 2014 | 9 | 2014 |
| Discovery of 2-(4-(2-fluoroethoxy) piperidin-1-yl)-9-methyl-9H-pyrrolo [2, 3-b: 4, 5-c’] dipyridine ([18F] PI-2014) as PET tracer for the detection of pathological aggregated … E Gabellieri, F Capotosti, J Molette, N Sreenivasachary, A Mueller, ... European Journal of Medicinal Chemistry 204, 112615, 2020 | 7 | 2020 |
| Characterization of novel PET tracers for the assessment of tau pathology in Alzheimer’s disease and other tauopathies A Stephens, H Kroth, M Berndt, F Capotosti, A Mueller, J Molette, ... Neurodegener. Dis 17, 2017 | 7 | 2017 |
| Carbazole and carboline compounds for use in the diagnosis, treatment, alleviation or prevention of disorders associated with amyloid or amyloid-like proteins H Kroth, S Nampally, E Gabellieri, PAR BENDERITTER, W Froestl, ... US Patent 10,662,193, 2020 | 6 | 2020 |
| [IC‐P‐192]: PRECLINICAL CHARACTERIZATION OF PI‐2620, A NOVEL TAU PET TRACER FOR DETECTION OF TAU IN AD AND OTHER TAUOPATHIES A Mueller, H Kroth, H Schieferstein, M Berndt, F Oden, F Capotosti, ... Alzheimer's & Dementia 13 (7S_Part_3), P141-P142, 2017 | 5 | 2017 |
