Structure–Activity Relationship Studies of Acetazolamide-Based Carbonic Anhydrase Inhibitors with Activity against Neisseria gonorrhoeae CS Hewitt, NS Abutaleb, AEM Elhassanny, A Nocentini, X Cao, DP Amos, ... ACS infectious diseases 7 (7), 1969-1984, 2021 | 71 | 2021 |
Structure-activity relationship studies for inhibitors for vancomycin-resistant Enterococcus and human carbonic anhydrases W An, KJ Holly, A Nocentini, RD Imhoff, CS Hewitt, NS Abutaleb, X Cao, ... Journal of Enzyme Inhibition and Medicinal Chemistry 37 (1), 1838-1844, 2022 | 31 | 2022 |
Structural Characterization of Thiadiazolesulfonamide Inhibitors Bound to Neisseria gonorrhoeae α-Carbonic Anhydrase AK Marapaka, A Nocentini, MS Youse, W An, KJ Holly, C Das, R Yadav, ... ACS Medicinal Chemistry Letters 14 (1), 103-109, 2022 | 19 | 2022 |
Discovery and validation of a novel inhibitor of HYPE-mediated AMPylation A Camara, H Chugh, A George, L Dolidze, K Ryu, KJ Holly, DP Flaherty, ... Cell Stress and Chaperones 29 (3), 404-424, 2024 | 1 | 2024 |
Unguarded liabilities: Borrelia burgdorferi’s complex amino acid dependence exposes unique avenues of inhibition KJ Holly, A Kataria, DP Flaherty, AM Groshong Frontiers in Antibiotics 3, 1395425, 2024 | 1 | 2024 |
Enterococci carbonic anhydrase inhibition KJ Holly, MS Youse, DP Flaherty Bacterial Carbonic Anhydrases 55, 283, 2024 | | 2024 |
Neisseria gonorrhoeae carbonic anhydrase inhibition MS Youse, KJ Holly, DP Flaherty Bacterial Carbonic Anhydrases 55, 243, 2024 | | 2024 |