The symbiotic relationship between drug discovery and organic chemistry OO Grygorenko, DM Volochnyuk, SV Ryabukhin, DB Judd Chemistry–A European Journal 26 (6), 1196-1237, 2020 | 165 | 2020 |
Bicyclic conformationally restricted diamines OO Grygorenko, DS Radchenko, DM Volochnyuk, AA Tolmachev, ... Chemical Reviews 111 (9), 5506-5568, 2011 | 120 | 2011 |
Combinatorial knoevenagel reactions SV Ryabukhin, AS Plaskon, DM Volochnyuk, SE Pipko, AN Shivanyuk, ... Journal of Combinatorial Chemistry 9 (6), 1073-1078, 2007 | 111 | 2007 |
N-Substituted ureas and thioureas in Biginelli reaction promoted by chlorotrimethylsilane: Convenient synthesis of N1-alkyl-, N1-aryl-, and N1, N3-dialkyl-3, 4-dihydropyrimidin … SV Ryabukhin, AS Plaskon, EN Ostapchuk, DM Volochnyuk, ... Synthesis 2007 (03), 417-427, 2007 | 107 | 2007 |
Synthesis of fused imidazoles and benzothiazoles from (hetero) aromatic ortho-diamines or ortho-aminothiophenol and aldehydes promoted by chlorotrimethylsilane SV Ryabukhin, AS Plaskon, DM Volochnyuk, AA Tolmachev Synthesis 2006 (21), 3715-3726, 2006 | 100 | 2006 |
Evolution of commercially available compounds for HTS DM Volochnyuk, SV Ryabukhin, YS Moroz, O Savych, A Chuprina, ... Drug Discovery Today 24 (2), 390-402, 2019 | 81 | 2019 |
Emerging building blocks for medicinal chemistry: recent synthetic advances OO Grygorenko, DM Volochnyuk, BV Vashchenko European Journal of Organic Chemistry 2021 (47), 6478-6510, 2021 | 72 | 2021 |
Electron-rich amino heterocycles for regiospecific synthesis of trifluoromethyl-containing fused pyridines DM Volochnyuk, AO Pushechnikov, DG Krotko, DA Sibgatulin, ... Synthesis 2003 (10), 1531-1540, 2003 | 71 | 2003 |
Effect of gem‐Difluorination on the Key Physicochemical Properties Relevant to Medicinal Chemistry: The Case of Functionalized Cycloalkanes S Holovach, KP Melnykov, A Skreminskiy, M Herasymchuk, O Tavlui, ... Chemistry–A European Journal 28 (19), e202200331, 2022 | 68 | 2022 |
Saturated boronic acids, boronates, and trifluoroborates: an update on their synthetic and medicinal chemistry DM Volochnyuk, AO Gorlova, OO Grygorenko Chemistry–A European Journal 27 (62), 15277-15326, 2021 | 66 | 2021 |
A close-up look at the chemical space of commercially available building blocks for medicinal chemistry Y Zabolotna, DM Volochnyuk, SV Ryabukhin, D Horvath, KS Gavrilenko, ... Journal of chemical information and modeling 62 (9), 2171-2185, 2021 | 63 | 2021 |
Cyclobutane-derived diamines: synthesis and molecular structure DS Radchenko, SO Pavlenko, OO Grygorenko, DM Volochnyuk, ... The Journal of Organic Chemistry 75 (17), 5941-5952, 2010 | 63 | 2010 |
Catalytic undirected borylation of tertiary C–H bonds in bicyclo [1.1. 1] pentanes and bicyclo [2.1. 1] hexanes IF Yu, JL Manske, A Diéguez-Vázquez, A Misale, AE Pashenko, ... Nature chemistry 15 (5), 685-693, 2023 | 62 | 2023 |
Synthesis of quinolines from 3-formylchromone AS Plaskon, SV Ryabukhin, DM Volochnyuk, KS Gavrilenko, ... The Journal of Organic Chemistry 73 (15), 6010-6013, 2008 | 62 | 2008 |
3-Methoxalylchromone—a novel versatile reagent for the regioselective purine isostere synthesis S Mkrtchyan, VO Iaroshenko, S Dudkin, A Gevorgyan, M Vilches-Herrera, ... Organic & Biomolecular Chemistry 8 (23), 5280-5284, 2010 | 57 | 2010 |
Aminoheterocycles as synthons for combinatorial Biginelli reactions SV Ryabukhin, AS Plaskon, SY Boron, DM Volochnyuk, AA Tolmachev Molecular diversity 15, 189-195, 2011 | 56 | 2011 |
CF3-substituted 1, 3-dicarbonyl compounds in the Biginelli reaction promoted by chlorotrimethylsilane SV Ryabukhin, AS Plaskon, EN Ostapchuk, DM Volochnyuk, OV Shishkin, ... Journal of Fluorine Chemistry 129 (7), 625-631, 2008 | 52 | 2008 |
Synthesis of Trifluoromethyl-Substituted 3-Azabicyclo [n. 1.0] alkanes: Advanced Building Blocks for Drug Discovery. OS Artamonov, EY Slobodyanyuk, DM Volochnyuk, IV Komarov, ... European Journal of Organic Chemistry 2014 (17), 2014 | 50 | 2014 |
2, 3-Unsubstituted chromones and their enaminone precursors as versatile reagents for the synthesis of fused pyridines VO Iaroshenko, S Mkrtchyan, A Gevorgyan, M Miliutina, A Villinger, ... Organic & Biomolecular Chemistry 10 (4), 890-894, 2012 | 48 | 2012 |
Approach to the library of fused pyridine-4-carboxylic acids by Combes-type reaction of acyl pyruvates and electron-rich amino heterocycles DM Volochnyuk, SV Ryabukhin, AS Plaskon, YV Dmytriv, OO Grygorenko, ... Journal of Combinatorial Chemistry 12 (4), 510-517, 2010 | 48 | 2010 |