| Allosteric modulation of neurotransmitter transporters as a therapeutic strategy M Niello, R Gradisch, CJ Loland, T Stockner, HH Sitte Trends in Pharmacological Sciences 41 (7), 446-463, 2020 | 61 | 2020 |
| Structural basis of organic cation transporter-3 inhibition B Khanppnavar, J Maier, F Herborg, R Gradisch, E Lazzarin, D Luethi, ... Nature communications 13 (1), 6714, 2022 | 55 | 2022 |
| The role of the degenerate nucleotide binding site in type I ABC exporters T Stockner, R Gradisch, L Schmitt FEBS letters 594 (23), 3815-3838, 2020 | 45 | 2020 |
| Occlusion of the human serotonin transporter is mediated by serotonin-induced conformational changes in the bundle domain R Gradisch, D Szöllősi, M Niello, E Lazzarin, HH Sitte, T Stockner Journal of Biological Chemistry 298 (3), 2022 | 21 | 2022 |
| Persistent binding at dopamine transporters determines sustained psychostimulant effects M Niello, S Sideromenos, R Gradisch, R O´ Shea, J Schwazer, J Maier, ... Proceedings of the National Academy of Sciences 120 (6), e2114204120, 2023 | 14 | 2023 |
| Ligand coupling mechanism of the human serotonin transporter differentiates substrates from inhibitors R Gradisch, K Schlögl, E Lazzarin, M Niello, J Maier, FP Mayer, ... Nature Communications 15 (1), 417, 2024 | 8 | 2024 |
| De novo variants in GABRA4 are associated with a neurological phenotype including developmental delay, behavioral abnormalities and epilepsy SA Sajan, R Gradisch, FD Vogel, AJ Coffey, D Salyakina, D Soler, ... European Journal of Human Genetics 32 (8), 912-919, 2024 | 5 | 2024 |
| Unveiling the crucial role of betaine: modulation of GABA homeostasis via SLC6A1 transporter (GAT1) M Bhatt, E Lazzarin, AS Alberto-Silva, G Domingo, R Zerlotti, R Gradisch, ... Cellular and Molecular Life Sciences 81 (1), 269, 2024 | 3 | 2024 |
| Free energy profile of the substrate‐induced occlusion of the human serotonin transporter L Alves da Silva, E Lazzarin, R Gradisch, A Clarke, T Stockner Journal of Neurochemistry 168 (9), 1993-2006, 2024 | 1 | 2024 |
| Interaction of GAT1 with sodium ions: from efficient recruitment to stabilisation of substrate and conformation E Lazzarin, R Gradisch, SMC Skopec, L Alves da Silva, ... bioRxiv, 2023.10. 10.561652, 2023 | 1 | 2023 |
Assoc.Prof. Thomas StocknerMedical University of ViennaZweryfikowany adres z meduniwien.ac.at