| Discovery of ARD-69 as a highly potent proteolysis targeting chimera (PROTAC) degrader of androgen receptor (AR) for the treatment of prostate cancer X Han, C Wang, C Qin, W Xiang, E Fernandez-Salas, CY Yang, M Wang, ... Journal of medicinal chemistry 62 (2), 941-964, 2019 | 385 | 2019 |
| Discovery of QCA570 as an exceptionally potent and efficacious proteolysis targeting chimera (PROTAC) degrader of the bromodomain and extra-terminal (BET) proteins capable of … C Qin, Y Hu, B Zhou, E Fernandez-Salas, CY Yang, L Liu, D McEachern, ... Journal of medicinal chemistry 61 (15), 6685-6704, 2018 | 277 | 2018 |
| Discovery of highly potent and efficient PROTAC degraders of androgen receptor (AR) by employing weak binding affinity VHL E3 ligase ligands X Han, L Zhao, W Xiang, C Qin, B Miao, T Xu, M Wang, CY Yang, ... Journal of medicinal chemistry 62 (24), 11218-11231, 2019 | 208 | 2019 |
| Iron-Facilitated Direct Oxidative C− H Transformation of Allylarenes or Alkenes to Alkenyl Nitriles C Qin, N Jiao Journal of the American Chemical Society 132 (45), 15893-15895, 2010 | 195 | 2010 |
| Silver-Catalyzed Nitrogenation of Alkynes: A Direct Approach to Nitriles through C C Bond Cleavage. T Shen, T Wang, C Qin, N Jiao Angewandte Chemie 125 (26), 2013 | 191 | 2013 |
| Ru (ii)-catalyzed intermolecular C–H amidation of weakly coordinating ketones QZ Zheng, YF Liang, C Qin, N Jiao Chemical Communications 49 (50), 5654-5656, 2013 | 155 | 2013 |
| Iron-catalyzed CH and CC bond cleavage: a direct approach to amides from simple hydrocarbons. C Qin, W Zhou, F Chen, Y Ou, N Jiao Angewandte Chemie (International ed. in English) 50 (52), 12595-12599, 2011 | 130 | 2011 |
| Discovery of ARD-2585 as an exceptionally potent and orally active PROTAC degrader of androgen receptor for the treatment of advanced prostate cancer W Xiang, L Zhao, X Han, C Qin, B Miao, D McEachern, Y Wang, ... Journal of medicinal chemistry 64 (18), 13487-13509, 2021 | 126 | 2021 |
| Small-molecule PROTAC degraders of the Bromodomain and Extra Terminal (BET) proteins—A review CY Yang, C Qin, L Bai, S Wang Drug Discovery Today: Technologies 31, 43-51, 2019 | 120 | 2019 |
| Strategies toward discovery of potent and orally bioavailable proteolysis targeting chimera degraders of androgen receptor for the treatment of prostate cancer X Han, L Zhao, W Xiang, C Qin, B Miao, D McEachern, Y Wang, ... Journal of medicinal chemistry 64 (17), 12831-12854, 2021 | 117 | 2021 |
| Selective C (sp2)-C (sp) bond cleavage: the nitrogenation of alkynes to amides. C Qin, P Feng, Y Ou, T Shen, T Wang, N Jiao Angewandte Chemie (International ed. in English) 52 (30), 7850-7854, 2013 | 97 | 2013 |
| Implanting Nitrogen into Hydrocarbon Molecules through C H and C C Bond Cleavages: A Direct Approach to Tetrazoles F Chen, C Qin, Y Cui, N Jiao Angewandte Chemie International Edition 50 (48), 11487-11491, 2011 | 83 | 2011 |
| Splitting a Substrate into Three Parts: Gold‐Catalyzed Nitrogenation of Alkynes by C C and C C Bond Cleavage C Qin, Y Su, T Shen, X Shi, N Jiao Angewandte Chemie 128 (1), 358-362, 2016 | 82 | 2016 |
| FeCl2‐Promoted Cleavage of the Unactivated C C Bond of Alkylarenes and Polystyrene: Direct Synthesis of Arylamines C Qin, T Shen, C Tang, N Jiao ChemInform 43 (51), no, 2012 | 73 | 2012 |
| Без заголовка WO Patent 2018052945:A1, 0 | 34* | |
| Discovery of ARD-1676 as a highly potent and orally efficacious AR PROTAC degrader with a broad activity against AR mutants for the treatment of AR+ human prostate cancer W Xiang, L Zhao, X Han, T Xu, S Kregel, M Wang, B Miao, C Qin, M Wang, ... Journal of Medicinal Chemistry 66 (18), 13280-13303, 2023 | 31 | 2023 |
| Oxygenation of simple olefins through selective allylic C− C bond cleavage: a direct approach to cinnamyl aldehydes J Liu, X Wen, C Qin, X Li, X Luo, A Sun, B Zhu, S Song, N Jiao Angewandte Chemie International Edition 56 (39), 11940-11944, 2017 | 30 | 2017 |
| Discovery of ARD-2051 as a potent and orally efficacious proteolysis targeting chimera (PROTAC) degrader of androgen receptor for the treatment of advanced prostate cancer X Han, L Zhao, W Xiang, B Miao, C Qin, M Wang, T Xu, D McEachern, ... Journal of Medicinal Chemistry 66 (13), 8822-8843, 2023 | 28 | 2023 |
| PROTAC degraders of androgen receptor‐integrated dissolving microneedles for androgenetic alopecia and recrudescence treatment via single topical administration R Wang, T Zhong, Q Bian, S Zhang, X Ma, L Li, Y Xu, Y Gu, A Yuan, W Hu, ... Small Methods 7 (1), 2201293, 2023 | 27 | 2023 |
| Discovery of BWA-522, a First-in-Class and Orally Bioavailable PROTAC Degrader of the Androgen Receptor Targeting N-Terminal Domain for the Treatment of … B Zhang, C Liu, Z Yang, S Zhang, X Hu, B Li, M Mao, X Wang, Z Li, S Ma, ... Journal of medicinal chemistry 66 (16), 11158-11186, 2023 | 21 | 2023 |