Synthesis, biological evaluation and molecular modeling study of new (1, 2, 4-triazole or 1, 3, 4-thiadiazole)-methylthio-derivatives of quinazolin-4 (3H)-one as DHFR inhibitors YI El-Gazzar, HH Georgey, SM El-Messery, HA Ewida, GS Hassan, ... Bioorganic Chemistry 72, 282-292, 2017 | 55 | 2017 |
Thiazolo [4, 5-d] pyridazine analogues as a new class of dihydrofolate reductase (DHFR) inhibitors: Synthesis, biological evaluation and molecular modeling study MA Ewida, DA Abou El Ella, DS Lasheen, HA Ewida, YI El-Gazzar, ... Bioorganic chemistry 74, 228-237, 2017 | 28 | 2017 |
Imidazo [2′, 1′: 2, 3] thiazolo [4, 5-d] pyridazinone as a new scaffold of DHFR inhibitors: Synthesis, biological evaluation and molecular modeling study MA Ewida, DA Abou El Ella, DS Lasheen, HA Ewida, YI El-Gazzar, ... Bioorganic Chemistry 80, 11-23, 2018 | 27 | 2018 |
New quinazolinone‐based derivatives as DHFR/EGFR‐TK inhibitors: synthesis, molecular modeling simulations, and anticancer activity YI El‐Gazzar, HR Ghaiad, AM El Kerdawy, RF George, HH Georgey, ... Archiv der Pharmazie 356 (1), 2200417, 2023 | 12 | 2023 |
Synthesis, biological evaluation and molecular modeling study of new (1, 2, 4-triazole or 1, 3, 4-thiadiazole)-methylthio-derivatives of quinazolin-4 (3H)-one as DHFR inhibitors MM Rafaat, YI El-Gazzar, HH Georgey, SM El-Messery, HA Ewida, ... ELSEVIER, Bioorganic Chemistry, 2017 | | 2017 |