A 1, 8-naphthyridone derivative targets the HIV-1 Tat-mediated transcription and potently inhibits the HIV-1 replication S Massari, D Daelemans, ML Barreca, A Knezevich, S Sabatini, ... Journal of medicinal chemistry 53 (2), 641-648, 2010 | 174 | 2010 |
6-Aminoquinolones as new potential anti-HIV agents V Cecchetti, C Parolin, S Moro, T Pecere, E Filipponi, A Calistri, ... Journal of medicinal chemistry 43 (20), 3799-3802, 2000 | 151 | 2000 |
Effects of novel 6-desfluoroquinolones and classic quinolones on pentylenetetrazole-induced seizures in mice A De Sarro, V Cecchetti, V Fravolini, F Naccari, O Tabarrini, G De Sarro Antimicrobial agents and chemotherapy 43 (7), 1729-1736, 1999 | 147 | 1999 |
Evolution from a Natural Flavones Nucleus to Obtain 2-(4-Propoxyphenyl)quinoline Derivatives As Potent Inhibitors of the S. aureus NorA Efflux Pump S Sabatini, F Gosetto, G Manfroni, O Tabarrini, GW Kaatz, D Patel, ... Journal of medicinal chemistry 54 (16), 5722-5736, 2011 | 124 | 2011 |
Quinolonecarboxylic acids. 2. Synthesis and antibacterial evaluation of 7-oxo-2, 3 dihydro-7H-pyrido [1, 2, 3-de][1, 4] benzothiazine-6-carboxylic acids V Cecchetti, A Fravolini, R Fringuelli, G Mascellani, P Pagella, M Palmioli, ... Journal of medicinal chemistry 30 (3), 465-473, 1987 | 121 | 1987 |
A broad anti-influenza hybrid small molecule that potently disrupts the interaction of polymerase acidic protein–basic protein 1 (PA-PB1) subunits S Massari, G Nannetti, J Desantis, G Muratore, S Sabatini, G Manfroni, ... Journal of Medicinal Chemistry 58 (9), 3830-3842, 2015 | 108 | 2015 |
Pyrazolo[4,3-c][1,2]benzothiazines 5,5-Dioxide: A Promising New Class of Staphylococcus aureus NorA Efflux Pump Inhibitors S Sabatini, F Gosetto, S Serritella, G Manfroni, O Tabarrini, N Iraci, ... Journal of Medicinal Chemistry 55 (7), 3568-3572, 2012 | 105 | 2012 |
Synthesis and anti-BVDV activity of acridones as new potential antiviral agents O Tabarrini, G Manfroni, A Fravolini, V Cecchetti, S Sabatini, E De Clercq, ... Journal of medicinal chemistry 49 (8), 2621-2627, 2006 | 103 | 2006 |
Studies on 6-aminoquinolones: synthesis and antibacterial evaluation of 6-amino-8-methylquinolones V Cecchetti, A Fravolini, MC Lorenzini, O Tabarrini, P Terni, T Xin Journal of medicinal chemistry 39 (2), 436-445, 1996 | 97 | 1996 |
Velnacrine thiaanalogues as potential agents for treating alzheimer's disease O Tabarrini, V Cecchetti, A Temperini, E Filipponi, MG Lamperti, ... Bioorganic & medicinal chemistry 9 (11), 2921-2928, 2001 | 94 | 2001 |
New anti-human immunodeficiency virus type 1 6-aminoquinolones: mechanism of action C Parolin, B Gatto, C Del Vecchio, T Pecere, E Tramontano, V Cecchetti, ... Antimicrobial agents and chemotherapy 47 (3), 889-896, 2003 | 92 | 2003 |
Structure− activity relationship study on anti-HIV 6-desfluoroquinolones O Tabarrini, S Massari, D Daelemans, M Stevens, G Manfroni, S Sabatini, ... Journal of medicinal chemistry 51 (17), 5454-5458, 2008 | 89 | 2008 |
Mg2+-mediated binding of 6-Substituted quinolones to DNA: Relevance to biological activity C Sissi, M Andreolli, V Cecchetti, A Fravolini, B Gatto, M Palumbo Bioorganic & medicinal chemistry 6 (9), 1555-1561, 1998 | 83 | 1998 |
Design and synthesis of modified quinolones as antitumoral acridones O Tabarrini, V Cecchetti, A Fravolini, G Nocentini, A Barzi, S Sabatini, ... Journal of medicinal chemistry 42 (12), 2136-2144, 1999 | 78 | 1999 |
Highly Potent 1,4-Benzothiazine Derivatives as KATP-Channel Openers V Cecchetti, V Calderone, O Tabarrini, S Sabatini, E Filipponi, L Testai, ... Journal of medicinal chemistry 46 (17), 3670-3679, 2003 | 74 | 2003 |
Pharmacophore-Based Repositioning of Approved Drugs as Novel Staphylococcus aureus NorA Efflux Pump Inhibitors A Astolfi, T Felicetti, N Iraci, G Manfroni, S Massari, D Pietrella, O Tabarrini, ... Journal of medicinal chemistry 60 (4), 1598-1604, 2017 | 71 | 2017 |
6-Aminoquinolones: a new class of quinolone antibacterials? V Cecchetti, S Clementi, G Cruciani, A Fravolini, PG Pagella, A Savino, ... Journal of medicinal chemistry 38 (6), 973-982, 1995 | 69 | 1995 |
Targeting flavivirus RNA dependent RNA polymerase through a pyridobenzothiazole inhibitor D Tarantino, R Cannalire, E Mastrangelo, R Croci, G Querat, ML Barreca, ... Antiviral research 134, 226-235, 2016 | 68 | 2016 |
Studies on anti-HIV quinolones: new insights on the C-6 position S Massari, D Daelemans, G Manfroni, S Sabatini, O Tabarrini, ... Bioorganic & medicinal chemistry 17 (2), 667-674, 2009 | 67 | 2009 |
Structural investigation of cycloheptathiophene-3-carboxamide derivatives targeting influenza virus polymerase assembly S Massari, G Nannetti, L Goracci, L Sancineto, G Muratore, S Sabatini, ... Journal of Medicinal Chemistry 56 (24), 10118-10131, 2013 | 66 | 2013 |