Pyrimidine-based EGFR TK inhibitors in targeted cancer therapy

A Ayati, S Moghimi, M Toolabi, A Foroumadi - European Journal of …, 2021‏ - Elsevier
Despite significant improvements of new treatment options, cancer continues to represent as
one of the most common and fatal disease. The EGFR signaling pathway is considered as a …

Signaling pathway and small-molecule drug discovery of FGFR: a comprehensive review

J Zheng, W Zhang, L Li, Y He, Y Wei, Y Dang… - Frontiers in …, 2022‏ - frontiersin.org
Targeted therapy is a groundbreaking innovation for cancer treatment. Among the receptor
tyrosine kinases, the fibroblast growth factor receptors (FGFRs) garnered substantial …

Therapeutic strategies of dual-target small molecules to overcome drug resistance in cancer therapy

J Ye, J Wu, B Liu - Biochimica et Biophysica Acta (BBA)-Reviews on …, 2023‏ - Elsevier
Despite some advances in targeted therapeutics of human cancers, curative cancer
treatment still remains a tremendous challenge due to the occurrence of drug resistance. A …

Development of dual inhibitors targeting epidermal growth factor receptor in cancer therapy

L Tan, J Zhang, Y Wang, X Wang, Y Wang… - Journal of Medicinal …, 2022‏ - ACS Publications
Epidermal growth factor receptor (EGFR) is of great significance in mediating cell signaling
transduction and tumor behaviors. Currently, third-generation inhibitors of EGFR, especially …

An outlook of docking analysis and structure-activity relationship of pyrimidine-based analogues as EGFR inhibitors against non-small cell lung cancer (NSCLC)

R Pal, G Teli, S Sengupta, L Maji… - Journal of …, 2024‏ - Taylor & Francis
Almost 80% of lung cancer diagnoses each year correspond to non-small cell lung cancer
(NSCLC). The percentage of NSCLC with EGFR overexpression ranges from 40% to 89 …

Recent advances in, and challenges of, anti-angiogenesis agents for tumor chemotherapy based on vascular normalization

K Wang, Q Chen, N Liu, J Zhang, X Pan - Drug discovery today, 2021‏ - Elsevier
A major problem associated with cancer treatment is resistance-prone chemotherapeutic
drugs. An increasing number of studies have documented that the occurrence of resistance …

Nitrogen‐Containing Heterocyclic Scaffolds as EGFR Inhibitors: Design Approaches, Molecular Docking, and Structure‐Activity Relationships

R Pal, G Teli, G Swamy Purawarga Matada… - …, 2023‏ - Wiley Online Library
Cancer is a wide collection of diseases and among the numerous pathways involved in
cancer pathogenesis, pathway involving epidermal growth factor receptor (EGFR) is one of …

Epidermal growth factor receptor inhibitors as potential anticancer agents: An update of recent progress

B Sharma, VJ Singh, PA Chawla - Bioorganic Chemistry, 2021‏ - Elsevier
Epidermal growth factor receptor (EGFR) is a vital intermediate in cell signaling pathway
including cell proliferation, angiogenesis, apoptosis, and metastatic spread and also having …

Discovery of anilino-1, 4-naphthoquinones as potent EGFR tyrosine kinase inhibitors: synthesis, biological evaluation, and comprehensive molecular modeling

P Mahalapbutr, R Leechaisit, A Thongnum… - ACS …, 2022‏ - ACS Publications
Epidermal growth factor receptor (EGFR) has been recognized as one of the attractive
targets for anticancer drug development. Herein, a set of anilino-1, 4-naphthoquinone …

Epidermal growth factor receptor dual-target inhibitors as a novel therapy for cancer: A review

C Wang, Y Zhang, T Zhang, J Xu, S Yan, B Liang… - International Journal of …, 2023‏ - Elsevier
Overexpression of the epidermal growth factor receptor (EGFR) has been linked to several
human cancers, including esophageal cancer, pancreatic cancer, anal cancer, breast …