The substitution of primary or secondary alcohols with nucleophiles mediated by a redox
combination of a trialkylor triarylphosphine and a dialkyl azodicarboxylate is popularly …

Ruthenium complexes are an important class that has multiple catalytic and biological
applications. Ruthenium has a remarkably broad and diversified chemical spectrum. In the …

The Mitsunobu reaction is a widely used and versatile method for the dehydrative oxidation–
reduction condensation of an acid/pronucleophile usually with a primary or secondary …

This manuscript describes a new strategy for prodrug synthesis in which a relatively inert
ether group is introduced at an early stage in a synthetic sequence and functionalized in the …

A vanadium-catalyzed method for the oxidative kinetic resolution of α-hydroxyesters, using
oxygen as the terminal oxidant, is described. The catalyst is generated in situ from vanadium …

Aim To investigate whether modifications of prostate-specific membrane antigen (PSMA)-
targeted radiolabeled urea-based inhibitors could reduce salivary gland uptake and thus …

The preparation of depsi-peptides, amide-to-ester-substituted peptides used to probe the
role of hydrogen bonding in protein folding energetics, is accomplished by replacing specific …

Development of new methods for the synthesis of β-amino acids is important as polymers of
these compounds are promising peptidomimetic candidates in medicinal chemistry. We …

Furan is a rodent hepatotoxicant and carcinogen. Because this compound is an important
industrial intermediate and has been detected in heat-processed foods and smoke, humans …

Cross-dehydrogenative C–O coupling of N-hydroxyimides with ketones, esters, and
carboxylic acids was achieved employing the di-tert-butyl peroxide as a source of free …