[HTML][HTML] Targeting Wnt signaling for the treatment of gastric cancer

S Koushyar, AG Powell, E Vincan… - International Journal of …, 2020 - mdpi.com
The Wnt signaling pathway is evolutionarily conserved, regulating both embryonic
development and maintaining adult tissue homeostasis. Wnt signaling controls several …

[HTML][HTML] Nobiletin and xanthohumol sensitize colorectal cancer stem cells to standard chemotherapy

A Turdo, A Glaviano, G Pepe, F Calapà, S Raimondo… - Cancers, 2021 - mdpi.com
Simple Summary Colorectal cancer stem cells (CR-CSCs) play a pivotal role in the therapy
resistance and relapse of CRC patients. Herein we demonstrate that new treatment …

Evaluation of AXIN1 and AXIN2 as targets of tankyrase inhibition in hepatocellular carcinoma cell lines

W Wang, P Liu, M Lavrijsen, S Li, R Zhang, S Li… - Scientific Reports, 2021 - nature.com
AXIN1 mutations are observed in 8–10% of hepatocellular carcinomas (HCCs) and
originally were considered to support tumor growth by aberrantly enhancing β-catenin …

[HTML][HTML] A small-molecule tankyrase inhibitor reduces glioma stem cell proliferation and sphere formation

KS Kierulf-Vieira, CJ Sandberg, J Waaler, K Lund… - Cancers, 2020 - mdpi.com
Evidence suggests that the growth and therapeutic resistance of glioblastoma (GBM) may be
enabled by a population of glioma stem cells (GSCs) that are regulated by typical stem cell …

Identification of response signatures for tankyrase inhibitor treatment in tumor cell lines

L Mygland, SA Brinch, MF Strand, PA Olsen… - Iscience, 2021 - cell.com
Small-molecule tankyrase 1 and tankyrase 2 (TNKS1/2) inhibitors are effective antitumor
agents in selected tumor cell lines and mouse models. Here, we characterized the response …