2-substituted benzothiazoles as antiproliferative agents: Novel insights on structure-activity relationships

A Ammazzalorso, S Carradori, R Amoroso… - European Journal of …, 2020 - Elsevier
Given the wide spectrum of biological activities, benzothiazoles represent privileged
scaffolds in medicinal chemistry, useful in drug discovery programs to modulate biological …

Design, synthesis and biological activities of (thio) urea benzothiazole derivatives

JE Mendieta-Wejebe, MC Rosales-Hernández… - International Journal of …, 2023 - mdpi.com
(Thio) ureas ((T) Us) and benzothiazoles (BTs) each have demonstrated to have a great
variety of biological activities. When these groups come together, the 2-(thio) …

Antifungal Effect of Volatile Organic Compounds from Bacillus velezensis CT32 against Verticillium dahliae and Fusarium oxysporum

X Li, X Wang, X Shi, B Wang, M Li, Q Wang, S Zhang - Processes, 2020 - mdpi.com
The present study focuses on the inhibitory effect of volatile metabolites released by Bacillus
velezensis CT32 on Verticillium dahliae and Fusarium oxysporum, the causal agents of …

Modern approaches to the synthesis and transformations of practically valuable benzothiazole derivatives

LV Zhilitskaya, BA Shainyan, NO Yarosh - Molecules, 2021 - mdpi.com
The review is devoted to modern trends in the chemistry of 2-amino and 2-mercapto
substituted benzothiazoles covering the literature since 2015. The reviewed heterocycles …

Green design and synthesis of some novel thiazolidinone appended benzothiazole–triazole hybrids as antimicrobial agents

B Dwivedi, D Bhardwaj, D Choudhary - RSC advances, 2024 - pubs.rsc.org
The global increase in bacterial resistance poses a significant threat, jeopardizing the
effectiveness of antibiotics. Therefore, the development of new and efficient antimicrobial …

Synthesis of biologically active derivatives of 2-aminobenzothiazole

LV Zhilitskaya, NО Yarosh - Chemistry of Heterocyclic Compounds, 2021 - Springer
Synthesis of biologically active derivatives of 2-aminobenzothiazole | Chemistry of Heterocyclic
Compounds Skip to main content Springer Nature Link Account Menu Find a journal Publish …

Recent advances in the synthesis of perimidines and their applications

N Sahiba, S Agarwal - Topics in Current Chemistry, 2020 - Springer
Perimidines are versatile scaffolds and a fascinating class of N-heterocycles that have
evolved significantly in recent years due to their immense applications in life sciences …

TBHP/KI-promoted annulation of anilines, ethers, and elemental sulfur: access to 2-Aryl-, 2-heteroaryl-, or 2-alkyl-substituted benzothiazoles

J Zhang, X Zhao, P Liu, P Sun - The Journal of Organic Chemistry, 2019 - ACS Publications
An efficient TBHP/KI-promoted annulation of anilines with ethers and elemental sulfur has
been developed through the selective C–O bond cleavage of ethers under transition-metal …

Green and highly efficient MCR strategy for the synthesis of pyrimidine analogs in water via C–C and C–N bond formation and docking studies

A Sethiya, J Soni, A Manhas, PC Jha… - Research on Chemical …, 2021 - Springer
The current study deals with the synthesis of some novel pyrimidine derivatives by the
reaction of aromatic aldehydes, 2-aminobenzothiazole, and dimedone in the presence of …

Copper-coordinated thiazoles and benzothiazoles: A perfect alliance in the search for compounds with antibacterial and antifungal activity

R Colorado-Peralta, JL Olivares-Romero… - Inorganics, 2023 - mdpi.com
Throughout human history, bacteria and fungi have caused infections that are difficult to
combat. For this reason, countless research groups have developed novel compounds to …