[HTML][HTML] In vitro models replicating the human intestinal epithelium for absorption and metabolism studies: A systematic review

A Fedi, C Vitale, G Ponschin, S Ayehunie… - Journal of Controlled …, 2021‏ - Elsevier
Absorption, distribution, metabolism and excretion (ADME) studies represent a fundamental
step in the early stages of drug discovery. In particular, the absorption of orally administered …

An overview of in vitro, ex vivo and in vivo models for studying the transport of drugs across intestinal barriers

Y Xu, N Shrestha, V Préat, A Beloqui - Advanced Drug Delivery Reviews, 2021‏ - Elsevier
Oral administration is the most commonly used route for drug delivery owing to its cost-
effectiveness, ease of administration, and high patient compliance. However, the absorption …

Pharmaceutical cocrystals: walking the talk

G Bolla, A Nangia - Chemical communications, 2016‏ - pubs.rsc.org
Pharmaceutical cocrystals belong to a sub-class of cocrystals wherein one of the
components is a drug molecule (or an active pharmaceutical ingredient, API) and the …

[HTML][HTML] Current evidence on the bioavailability of food bioactive peptides

L Amigo, B Hernández-Ledesma - Molecules, 2020‏ - mdpi.com
Food protein-derived bioactive peptides are recognized as valuable ingredients of functional
foods and/or nutraceuticals to promote health and reduce the risk of chronic diseases …

[HTML][HTML] Oral absorption of peptides and nanoparticles across the human intestine: Opportunities, limitations and studies in human tissues

P Lundquist, P Artursson - Advanced drug delivery reviews, 2016‏ - Elsevier
In this contribution, we review the molecular and physiological barriers to oral delivery of
peptides and nanoparticles. We discuss the opportunities and predictivity of various in vitro …

[HTML][HTML] Intestinal permeability and drug absorption: predictive experimental, computational and in vivo approaches

D Dahlgren, H Lennernäs - Pharmaceutics, 2019‏ - mdpi.com
The main objective of this review is to discuss recent advancements in the overall
investigation and in vivo prediction of drug absorption. The intestinal permeability of an …

The delivery of sensitive food bioactive ingredients: Absorption mechanisms, influencing factors, encapsulation techniques and evaluation models

C Bao, P Jiang, J Chai, Y Jiang, D Li, W Bao… - Food Research …, 2019‏ - Elsevier
Food-sourced bioactive compounds have drawn much attention due to their health benefits
such as anti-oxidant, anti-cancer, anti-diabetes and cardiovascular disease-preventing …

Correlation between oral drug absorption in humans and apparent drug permeability coefficients in human intestinal epithelial (Caco-2) cells

P Artursson, J Karlsson - Biochemical and biophysical research …, 1991‏ - Elsevier
Monolayers of a well differentiated human intestinal epithelial cell line, Caco-2, were used
as a model to study passive drug absorption across the intestinal epithelium. Absorption rate …

Development of a human primary gut-on-a-chip to model inflammatory processes

C Beaurivage, A Kanapeckaite, C Loomans… - Scientific reports, 2020‏ - nature.com
Inflammatory bowel disease (IBD) is a complex multi-factorial disease for which
physiologically relevant in vitro models are lacking. Existing models are often a compromise …

The Caco-2 cell line as a model of the intestinal barrier: influence of cell and culture-related factors on Caco-2 cell functional characteristics

Y Sambuy, I De Angelis, G Ranaldi, ML Scarino… - Cell biology and …, 2005‏ - Springer
The human intestinal Caco-2 cell line has been extensively used over the last twenty years
as a model of the intestinal barrier. The parental cell line, originally obtained from a human …