A field guide to foldamers

DJ Hill, MJ Mio, RB Prince, TS Hughes… - Chemical …, 2001‏ - ACS Publications
The breadth of structure and function displayed by the molecules of biology is remarkable.
Considering that there are only three major biopolymer backbones (proteins, ribonucleic …

DNA analogues: from supramolecular principles to biological properties

CJ Leumann - Bioorganic & medicinal chemistry, 2002‏ - Elsevier
Mainly driven by the needs of antisense research, a large number of oligonucleotide
analogues have been prepared and evaluated over the last 15 years. Besides minor …

Development of nucleic acid medicines based on chemical technology

Y Kawamoto, Y Wu, Y Takahashi, Y Takakura - Advanced Drug Delivery …, 2023‏ - Elsevier
Oligonucleotide-based therapeutics have attracted attention as an emerging modality that
includes the modulation of genes and their binding proteins related to diseases, allowing us …

α-l-ribo-Configured Locked Nucleic Acid (α-L-LNA):  Synthesis and Properties

MD Sørensen, L Kværnø, T Bryld… - Journal of the …, 2002‏ - ACS Publications
The syntheses of monomeric nucleosides and 3 '-O-phosphoramidite building blocks en
route to α-l-ribo-configured locked nucleic acids (α-L-LNA), composed entirely of α-L-LNA …

Oligonucleotide analogues

J Wengel, P Nielsen - US Patent 8,153,365, 2012‏ - Google Patents
US8153365B2 - Oligonucleotide analogues - Google Patents US8153365B2 -
Oligonucleotide analogues - Google Patents Oligonucleotide analogues Download PDF …

The eight stereoisomers of LNA (locked nucleic acid): a remarkable family of strong RNA binding molecules

VK Rajwanshi, AE Håkansson… - Angewandte …, 2000‏ - Wiley Online Library
1724 WILEY-VCH Verlag GmbH, D-69451 Weinheim, 2000 0044-8249/00/11209-1724
$17.50+. 50/0 Angew. Chem. 2000, 112, Nr. 9 towards both complementary DNA (ΔTm 3.08 …

LNA (locked nucleic acid)

J Wengel, A Koshkin, SK Singh, P Nielsen… - Nucleosides & …, 1999‏ - Taylor & Francis
Abstract LNA (Locked Nucleic Acid) forms duplexes with complementary DNA, RNA or LNA
with unprecedented thermal affinities. CD spectra show that duplexes involving fully …

C-Class CpG ODN: sequence requirements and characterization of immunostimulatory activities on mRNA level

M Jurk, B Schulte, A Kritzler, B Noll, E Uhlmann… - Immunobiology, 2004‏ - Elsevier
Synthetic oligodeoxynucleotides (ODN) containing unmethylated deoxycytosine–
deoxyguanosine (CpG) motifs are very potent inducers of the innate immune system …

Bicyclic nucleosides and conformational restriction of oligonucleotides

M Meldgaard, J Wengel - Journal of the Chemical Society, Perkin …, 2000‏ - pubs.rsc.org
Bicyclic nucleosides and conformational restriction of oligonucleotides - Journal of the Chemical
Society, Perkin Transactions 1 (RSC Publishing) DOI:10.1039/B000114G Royal Society of …

Chemistry of locked nucleic acids (LNA): Design, synthesis, and bio-physical properties

J Wengel, M Petersen, M Frieden, T Koch - Letters in Peptide Science, 2003‏ - Springer
Preparation of LNA nucleosides requires a number of synthetic steps but very efficient
procedures have been developed, as have protocols for synthesis of LNA oligonucleotides …