Discovery of soluble epoxide hydrolase inhibitors from chemical synthesis and natural products

CP Sun, XY Zhang, C Morisseau… - Journal of medicinal …, 2020‏ - ACS Publications
Soluble epoxide hydrolase (sEH) is an α/β hydrolase fold protein and widely distributed in
numerous organs including the liver, kidney, and brain. The inhibition of sEH can effectively …

Structures and bioactive properties of myrtucommulones and related acylphloroglucinols from Myrtaceae

R Nicoletti, MM Salvatore, P Ferranti, A Andolfi - Molecules, 2018‏ - mdpi.com
Myrtaceae are a group of plants that include a number of renowned species used in
ethnomedicine in many areas worldwide. Their valuable therapeutic properties have …

Discovery of glycosidated glycyrrhetinic acid derivatives: Natural product-based soluble epoxide hydrolase inhibitors

Q Liu, YX Wang, ZH Ge, MZ Zhu, J Ding… - European Journal of …, 2024‏ - Elsevier
There are few reports on soluble epoxide hydrolase (sEH) structure-activity relationship
studies using natural product-based scaffolds. In this study, we discovered that C-30 urea …

Highly Potent Antiausterity Agents from Callistemon citrinus and Their Mechanism of Action against the PANC-1 Human Pancreatic Cancer Cell Line

AM Tawila, S Sun, MJ Kim, AM Omar… - Journal of Natural …, 2020‏ - ACS Publications
Human pancreatic cancer cells display remarkable tolerance to nutrition starvation that help
them to survive in a hypovascular tumor microenvironment, a phenomenon known as …

Chemical constituents of Callistemon citrinus from Egypt and their antiausterity activity against PANC-1 human pancreatic cancer cell line

AM Tawila, S Sun, MJ Kim, AM Omar, DF Dibwe… - Bioorganic & Medicinal …, 2020‏ - Elsevier
Human pancreatic cancer is resistant to almost all conventional chemotherapeutic agents. It
is known to proliferate aggressively within hypovascular tumor microenvironment by …

Establishment of pressurized-liquid extraction by response surface methodology approach coupled to HPLC-DAD-TOF-MS for the determination of phenolic …

E Díaz-de-Cerio, D Arráez-Román… - Analytical and …, 2018‏ - Springer
Myrtus communis L.(myrtle) is native to the Mediterranean region and Western Asia. Its
leaves have demonstrated its potential effect towards different bioactivities like anti-diabetic …

Kaempferia diterpenoids and flavonoids: an overview on phytochemistry, biosynthesis, synthesis, pharmacology, and pharmacokinetics

C Anh Van, DX Duc, NT Son - Medicinal Chemistry Research, 2024‏ - Springer
Kaempferia species have contained various crucial ethnobotanical features, and are being
used as traditional folk medicines in some Southeast Asia. This review tends to highlight …

Callistemon genus- a review on phytochemistry and biological activities

EM Abdelmalek, MA Ramadan, FM Darwish… - Medicinal Chemistry …, 2021‏ - Springer
Callistemon is an important genus in the family Myrtaceae which contains about 34 species.
The members of this genus are known for their ornamental potentials, in addition to their …

Acylphloroglucinols from the leaves of Callistemon viminalis

HX Liu, YC Chen, Y Liu, WM Zhang, JW Wu, HB Tan… - Fitoterapia, 2016‏ - Elsevier
A phytochemical study on the leaves of Callistemon viminalis, a widely distributed
ornamental and medicinal plant of agricultural importance in China, resulted in the isolation …

Antiplasmodial β-Triketone–Flavanone Hybrids from the Flowers of the Australian Tree Corymbia torelliana

SPD Senadeera, L Lucantoni, S Duffy… - Journal of Natural …, 2018‏ - ACS Publications
The methanol extract of the flowers of the Australian eucalypt tree Corymbia torelliana
yielded six new β-triketone–flavanone hybrids, torellianones A–F (1–6), the …