The nuts and bolts of AGC protein kinases

LR Pearce, D Komander, DR Alessi - Nature reviews Molecular cell …, 2010 - nature.com
The AGC kinase subfamily of protein kinases contains 60 members, including PKA, PKG
and PKC. The family comprises some intensely examined protein kinases (such as Akt, S6K …

Protein kinase C (PKC) isoforms in cancer, tumor promotion and tumor suppression

N Isakov - Seminars in cancer biology, 2018 - Elsevier
The AGC family of serine/threonine kinases (PKA, PKG, PKC) includes more than 60
members that are critical regulators of numerous cellular functions, including cell cycle and …

[HTML][HTML] Cancer-associated protein kinase C mutations reveal kinase's role as tumor suppressor

CE Antal, AM Hudson, E Kang, C Zanca, C Wirth… - Cell, 2015 - cell.com
Protein kinase C (PKC) isozymes have remained elusive cancer targets despite the
unambiguous tumor promoting function of their potent ligands, phorbol esters, and the …

Emerging insights into the molecular and cellular basis of glioblastoma

GP Dunn, ML Rinne, J Wykosky… - Genes & …, 2012 - genesdev.cshlp.org
Glioblastoma is both the most common and lethal primary malignant brain tumor. Extensive
multiplatform genomic characterization has provided a higher-resolution picture of the …

The PTEN/PI3K/AKT signalling pathway in cancer, therapeutic implications

A Carnero, C Blanco-Aparicio, O Renner… - Current cancer drug …, 2008 - ingentaconnect.com
PTEN/PI3K/AKT constitutes an important pathway regulating the signaling of multiple
biological processes such as apoptosis, metabolism, cell proliferation and cell growth. PTEN …

Structural basis of protein kinase C isoform function

SF Steinberg - Physiological reviews, 2008 - journals.physiology.org
Protein kinase C (PKC) isoforms comprise a family of lipid-activated enzymes that have
been implicated in a wide range of cellular functions. PKCs are modular enzymes comprised …

The PI3K–PDK1 connection: more than just a road to PKB

B Vanhaesebroeck, DR Alessi - Biochemical Journal, 2000 - portlandpress.com
Phosphoinositide 3-kinases (PI3Ks) generate specific inositol lipids that have been
implicated in the regulation of cell growth, proliferation, survival, differentiation and …

[HTML][HTML] Regulation of elongation factor 2 kinase by p90RSK1 and p70 S6 kinase

X Wang, W Li, M Williams, N Terada, DR Alessi… - The EMBO …, 2001 - embopress.org
Elongation factor 2 kinase (eEF2k) phosphorylates and inactivates eEF2. Insulin induces
dephosphorylation of eEF2 and inactivation of eEF2 kinase, and these effects are blocked …

mTORC2 controls the activity of PKC and Akt by phosphorylating a conserved TOR interaction motif

TR Baffi, G Lordén, JM Wozniak, A Feichtner… - Science …, 2021 - science.org
The complex mTORC2 is accepted to be the kinase that controls the phosphorylation of the
hydrophobic motif, a key regulatory switch for AGC kinases, although whether mTOR directly …

Protein kinase SGK mediates survival signals by phosphorylating the forkhead transcription factor FKHRL1 (FOXO3a)

A Brunet, J Park, H Tran, LS Hu… - … and cellular biology, 2001 - Am Soc Microbiol
Serum-and glucocorticoid-inducible kinases (SGKs) form a novel family of serine/threonine
kinases that are activated in response to a variety of extracellular stimuli. SGKs are related to …