[HTML][HTML] Antidiabetic agents as a novel treatment for Alzheimer's and Parkinson's disease

J Nowell, E Blunt, D Gupta, P Edison - Ageing research reviews, 2023‏ - Elsevier
Therapeutic strategies for neurodegenerative disorders have commonly targeted individual
aspects of the disease pathogenesis to little success. Neurodegenerative diseases …

[HTML][HTML] Human protein tyrosine phosphatase 1B (PTP1B): from structure to clinical inhibitor perspectives

R Liu, C Mathieu, J Berthelet, W Zhang… - International Journal of …, 2022‏ - mdpi.com
Phosphorylation is an essential process in biological events and is considered critical for
biological functions. In tissues, protein phosphorylation mainly occurs on tyrosine (Tyr) …

Fructose and hepatic insulin resistance

S Softic, KL Stanhope, J Boucher… - Critical reviews in …, 2020‏ - Taylor & Francis
Excessive caloric intake in a form of high-fat diet (HFD) was long thought to be the major risk
factor for development of obesity and its complications, such as fatty liver disease and …

Update on GLUT4 vesicle traffic: a cornerstone of insulin action

JR Jaldin-Fincati, M Pavarotti, S Frendo-Cumbo… - Trends in Endocrinology …, 2017‏ - cell.com
Glucose transport is rate limiting for dietary glucose utilization by muscle and fat. The
glucose transporter GLUT4 is dynamically sorted and retained intracellularly and …

The role of protein tyrosine phosphatase 1B (PTP1B) in the pathogenesis of type 2 diabetes mellitus and its complications

M Teimouri, H Hosseini, Z ArabSadeghabadi… - Journal of physiology …, 2022‏ - Springer
Insulin resistance, the most important characteristic of the type 2 diabetes mellitus (T2DM), is
mostly caused by impairment in the insulin receptor (IR) signal transduction pathway …

Coumarins as potential antidiabetic agents

H Li, Y Yao, L Li - Journal of Pharmacy and Pharmacology, 2017‏ - academic.oup.com
Objectives Even with great advances in modern medicine and therapeutic agent
development, the search for effective antidiabetic drugs remains challenging. Coumarins are …

Turn and face the strange: § a new view on phosphatases

M Köhn - ACS central science, 2020‏ - ACS Publications
Phosphorylation as a post-translational modification is critical for cellular homeostasis.
Kinases and phosphatases regulate phosphorylation levels by adding or removing …

[HTML][HTML] Protein tyrosine phosphatase 1B (PTP1B) as a potential therapeutic target for neurological disorders

J Olloquequi, A Cano, E Sanchez-López… - Biomedicine & …, 2022‏ - Elsevier
Protein tyrosine phosphatase 1B (PTP1B) is a typical member of the PTP family, considered
a direct negative regulator of several receptor and receptor-associated tyrosine kinases …

Recent updates on development of protein-tyrosine phosphatase 1B inhibitors for treatment of diabetes, obesity and related disorders

S Singh, AS Grewal, R Grover, N Sharma, B Chopra… - Bioorganic …, 2022‏ - Elsevier
The aim of this review was to discuss an overview of type 2 diabetes; biology of PTP1B; role
of PTP1B in metabolic disorders; and recent updates in the development of PTP1B inhibitors …

Connecting Alzheimer's disease to diabetes: underlying mechanisms and potential therapeutic targets

MNN Vieira, RAS Lima-Filho, FG De Felice - Neuropharmacology, 2018‏ - Elsevier
Alzheimer's disease (AD) is a risk factor for type 2 diabetes and vice versa, and a growing
body of evidence indicates that these diseases are connected both at epidemiological …