PI3K isoforms in cell signalling and vesicle trafficking

B Bilanges, Y Posor, B Vanhaesebroeck - Nature reviews Molecular …, 2019‏ - nature.com
PI3Ks are a family of lipid kinases that phosphorylate intracellular inositol lipids to regulate
signalling and intracellular vesicular traffic. Mammals have eight isoforms of PI3K, divided …

Phosphoinositides: tiny lipids with giant impact on cell regulation

T Balla - Physiological reviews, 2013‏ - journals.physiology.org
Phosphoinositides (PIs) make up only a small fraction of cellular phospholipids, yet they
control almost all aspects of a cell's life and death. These lipids gained tremendous research …

The emerging mechanisms of isoform-specific PI3K signalling

B Vanhaesebroeck, J Guillermet-Guibert… - … reviews Molecular cell …, 2010‏ - nature.com
Abstract Phosphoinositide 3-kinases (PI3Ks) function early in intracellular signal
transduction pathways and affect many biological functions. A further level of complexity …

Classes of phosphoinositide 3-kinases at a glance

S Jean, AA Kiger - Journal of cell science, 2014‏ - journals.biologists.com
ABSTRACT The phosphoinositide 3-kinase (PI3K) family is important to nearly all aspects of
cell and tissue biology and central to human cancer, diabetes and aging. PI3Ks are spatially …

Targeting PI3K signalling in cancer: opportunities, challenges and limitations

JA Engelman - Nature Reviews Cancer, 2009‏ - nature.com
There are ample genetic and laboratory studies that suggest the PI3K–Akt pathway is vital to
the growth and survival of cancer cells. Inhibitors targeting this pathway are entering the …

Aberrant T cell signaling and subsets in systemic lupus erythematosus

T Katsuyama, GC Tsokos, VR Moulton - Frontiers in immunology, 2018‏ - frontiersin.org
Systemic lupus erythematosus (SLE) is a chronic multi-organ debilitating autoimmune
disease, which mainly afflicts women in the reproductive years. A complex interaction of …

[HTML][HTML] Efficacy of PI3K inhibitors in advanced breast cancer

B Verret, J Cortes, T Bachelot, F Andre, M Arnedos - Annals of Oncology, 2019‏ - Elsevier
Abstract The phosphoinositide 3 (PI3)-kinase/Akt signaling pathway has always been a
focus of interest in breast cancer due to its role in cell growth, cell proliferation, cell migration …

The PTEN/PI3K/AKT signalling pathway in cancer, therapeutic implications

A Carnero, C Blanco-Aparicio, O Renner… - Current cancer drug …, 2008‏ - ingentaconnect.com
PTEN/PI3K/AKT constitutes an important pathway regulating the signaling of multiple
biological processes such as apoptosis, metabolism, cell proliferation and cell growth. PTEN …

[HTML][HTML] A pharmacological map of the PI3-K family defines a role for p110α in insulin signaling

ZA Knight, B Gonzalez, ME Feldman, ER Zunder… - Cell, 2006‏ - cell.com
Summary Phosphoinositide 3-kinases (PI3-Ks) are an important emerging class of drug
targets, but the unique roles of PI3-K isoforms remain poorly defined. We describe here an …

Phosphatidylinositol 3-kinase-δ inhibitor CAL-101 shows promising preclinical activity in chronic lymphocytic leukemia by antagonizing intrinsic and extrinsic cellular …

SEM Herman, AL Gordon, AJ Wagner… - Blood, The Journal …, 2010‏ - ashpublications.org
Targeted therapy with imatinib in chronic myeloid leukemia (CML) prompted a new
treatment paradigm. Unlike CML, chronic lymphocytic leukemia (CLL) lacks an aberrant …