Novel bioactive natural products from bacteria via bioprospecting, genome mining and metabolic engineering

ON Sekurova, O Schneider… - Microbial biotechnology, 2019 - Wiley Online Library
For over seven decades, bacteria served as a valuable source of bioactive natural products
some of which were eventually developed into drugs to treat infections, cancer and immune …

Carboxylic acid reductase enzymes (CARs)

M Winkler - Current opinion in chemical biology, 2018 - Elsevier
Highlights•Carboxylate reductases (CARs) catalyze the selective one step reduction of an
acid to an aldehyde.•The substrate scope of CARs is broad.•CARs have been implemented …

De novo design and engineering of non-ribosomal peptide synthetases

KAJ Bozhüyük, F Fleischhacker, A Linck, F Wesche… - Nature …, 2018 - nature.com
Peptides derived from non-ribosomal peptide synthetases (NRPSs) represent an important
class of pharmaceutically relevant drugs. Methods to generate novel non-ribosomal …

Modification and de novo design of non-ribosomal peptide synthetases using specific assembly points within condensation domains

KAJ Bozhüyük, A Linck, A Tietze, J Kranz, F Wesche… - Nature …, 2019 - nature.com
Non-ribosomal peptide synthetases (NRPSs) are giant enzyme machines that activate
amino acids in an assembly line fashion. As NRPSs are not restricted to the incorporation of …

Ribosomally derived lipopeptides containing distinct fatty acyl moieties

F Hubrich, NM Bösch, C Chepkirui… - Proceedings of the …, 2022 - National Acad Sciences
Lipopeptides represent a large group of microbial natural products that include important
antibacterial and antifungal drugs and some of the most-powerful known biosurfactants. The …

Structural diversity and biological activities of cyclic depsipeptides from fungi

X Wang, X Gong, P Li, D Lai, L Zhou - Molecules, 2018 - mdpi.com
Cyclic depsipeptides (CDPs) are cyclopeptides in which amide groups are replaced by
corresponding lactone bonds due to the presence of a hydroxylated carboxylic acid in the …

Beyond peptide bond formation: the versatile role of condensation domains in natural product biosynthesis

S Dekimpe, J Masschelein - Natural product reports, 2021 - pubs.rsc.org
Covering: up to the end of 2020 Nonribosomal peptide synthetases are remarkable
molecular machines that produce a wide range of structurally complex peptide natural …

Engineering of the Filamentous Fungus Penicillium chrysogenum as Cell Factory for Natural Products

F Guzmán-Chávez, RD Zwahlen… - Frontiers in …, 2018 - frontiersin.org
Penicillium chrysogenum (renamed P. rubens) is the most studied member of a family of
more than 350 Penicillium species that constitute the genus. Since the discovery of penicillin …

Bacteria as genetically programmable producers of bioactive natural products

JJ Hug, D Krug, R Müller - Nature Reviews Chemistry, 2020 - nature.com
Next to plants, bacteria account for most of the biomass on Earth. They are found
everywhere, although certain species thrive only in specific ecological niches. These …

Structural advances toward understanding the catalytic activity and conformational dynamics of modular nonribosomal peptide synthetases

KD Patel, MR MacDonald, SF Ahmed, J Singh… - Natural Product …, 2023 - pubs.rsc.org
Covering: up to fall 2022. Nonribosomal peptide synthetases (NRPSs) are a family of
modular, multidomain enzymes that catalyze the biosynthesis of important peptide natural …