Machine-learning methods for ligand–protein molecular docking

K Crampon, A Giorkallos, M Deldossi, S Baud… - Drug discovery today, 2022‏ - Elsevier
Artificial intelligence (AI) is often presented as a new Industrial Revolution. Many domains
use AI, including molecular simulation for drug discovery. In this review, we provide an …

Artificial intelligence in the prediction of protein–ligand interactions: recent advances and future directions

A Dhakal, C McKay, JJ Tanner… - Briefings in …, 2022‏ - academic.oup.com
New drug production, from target identification to marketing approval, takes over 12 years
and can cost around $2.6 billion. Furthermore, the COVID-19 pandemic has unveiled the …

Interpretable bilinear attention network with domain adaptation improves drug–target prediction

P Bai, F Miljković, B John, H Lu - Nature Machine Intelligence, 2023‏ - nature.com
Predicting drug–target interaction is key for drug discovery. Recent deep learning-based
methods show promising performance, but two challenges remain: how to explicitly model …

CFSSynergy: combining feature-based and similarity-based methods for drug synergy prediction

F Rafiei, H Zeraati, K Abbasi, P Razzaghi… - Journal of chemical …, 2024‏ - ACS Publications
Drug synergy prediction plays a vital role in cancer treatment. Because experimental
approaches are labor-intensive and expensive, computational-based approaches get more …

[HTML][HTML] Comprehensive survey of recent drug discovery using deep learning

J Kim, S Park, D Min, W Kim - International Journal of Molecular Sciences, 2021‏ - mdpi.com
Drug discovery based on artificial intelligence has been in the spotlight recently as it
significantly reduces the time and cost required for develo** novel drugs. With the …

DeepTraSynergy: drug combinations using multimodal deep learning with transformers

F Rafiei, H Zeraati, K Abbasi, JB Ghasemi… - …, 2023‏ - academic.oup.com
Motivation Screening bioactive compounds in cancer cell lines receive more attention.
Multidisciplinary drugs or drug combinations have a more effective role in treatments and …

An effective self-supervised framework for learning expressive molecular global representations to drug discovery

P Li, J Wang, Y Qiao, H Chen, Y Yu… - Briefings in …, 2021‏ - academic.oup.com
How to produce expressive molecular representations is a fundamental challenge in
artificial intelligence-driven drug discovery. Graph neural network (GNN) has emerged as a …

Pharmacophoric-constrained heterogeneous graph transformer model for molecular property prediction

Y Jiang, S **, X **, X **ao, W Wu, X Liu… - Communications …, 2023‏ - nature.com
Informative representation of molecules is a crucial prerequisite in AI-driven drug design and
discovery. Pharmacophore information including functional groups and chemical reactions …

ZeroBind: a protein-specific zero-shot predictor with subgraph matching for drug-target interactions

Y Wang, Y **a, J Yan, Y Yuan, HB Shen… - Nature …, 2023‏ - nature.com
Existing drug-target interaction (DTI) prediction methods generally fail to generalize well to
novel (unseen) proteins and drugs. In this study, we propose a protein-specific meta …

Large language models in bioinformatics: applications and perspectives

J Liu, M Yang, Y Yu, H Xu, K Li, X Zhou - Ar**v, 2024‏ - pmc.ncbi.nlm.nih.gov
Large language models (LLMs) are a class of artificial intelligence models based on deep
learning, which have great performance in various tasks, especially in natural language …